SI3206684T1 - Iz pirazolina izhajajoča spojina in njena uporaba v tedenskem režimu odmerjanja proti vnetju in bolečini izhajajočih iz degenerativne bolezni sklepov pri sesalcih - Google Patents

Iz pirazolina izhajajoča spojina in njena uporaba v tedenskem režimu odmerjanja proti vnetju in bolečini izhajajočih iz degenerativne bolezni sklepov pri sesalcih

Info

Publication number
SI3206684T1
SI3206684T1 SI201531302T SI201531302T SI3206684T1 SI 3206684 T1 SI3206684 T1 SI 3206684T1 SI 201531302 T SI201531302 T SI 201531302T SI 201531302 T SI201531302 T SI 201531302T SI 3206684 T1 SI3206684 T1 SI 3206684T1
Authority
SI
Slovenia
Prior art keywords
derived
pyrazoline
mammals
dosage regimen
joint disease
Prior art date
Application number
SI201531302T
Other languages
English (en)
Slovenian (sl)
Inventor
Josep Homedes-Beguer
David Sabate-Elias
Original Assignee
Ecuphar N.V.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ecuphar N.V. filed Critical Ecuphar N.V.
Publication of SI3206684T1 publication Critical patent/SI3206684T1/sl

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pain & Pain Management (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Rheumatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Immunology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
SI201531302T 2014-10-16 2015-10-13 Iz pirazolina izhajajoča spojina in njena uporaba v tedenskem režimu odmerjanja proti vnetju in bolečini izhajajočih iz degenerativne bolezni sklepov pri sesalcih SI3206684T1 (sl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP14382396.1A EP3009137A1 (en) 2014-10-16 2014-10-16 Pyrazoline-derived compound and its use in a weekly dosage regime against inflammation and pain derived from degenerative joint disease in mammals
PCT/EP2015/073635 WO2016059028A1 (en) 2014-10-16 2015-10-13 Pyrazoline-derived compound and its use in a weekly dosage regime against inflammation and pain derived from degenerative joint disease in mammals
EP15778958.7A EP3206684B1 (en) 2014-10-16 2015-10-13 Pyrazoline-derived compound and its use in a weekly dosage regimen against inflammation and pain derived from degenerative joint disease in mammals

Publications (1)

Publication Number Publication Date
SI3206684T1 true SI3206684T1 (sl) 2020-11-30

Family

ID=51844648

Family Applications (1)

Application Number Title Priority Date Filing Date
SI201531302T SI3206684T1 (sl) 2014-10-16 2015-10-13 Iz pirazolina izhajajoča spojina in njena uporaba v tedenskem režimu odmerjanja proti vnetju in bolečini izhajajočih iz degenerativne bolezni sklepov pri sesalcih

Country Status (20)

Country Link
US (1) US11154536B2 (enExample)
EP (2) EP3009137A1 (enExample)
JP (1) JP6655625B2 (enExample)
CN (2) CN107257684A (enExample)
AR (1) AR102295A1 (enExample)
CA (1) CA2964428C (enExample)
CY (1) CY1123243T1 (enExample)
DK (1) DK3206684T3 (enExample)
ES (1) ES2828435T3 (enExample)
HR (1) HRP20201233T1 (enExample)
HU (1) HUE050511T2 (enExample)
LT (1) LT3206684T (enExample)
MX (1) MX376725B (enExample)
PL (1) PL3206684T3 (enExample)
PT (1) PT3206684T (enExample)
RS (1) RS60777B1 (enExample)
SI (1) SI3206684T1 (enExample)
SM (1) SMT202000415T1 (enExample)
TW (1) TWI707678B (enExample)
WO (1) WO2016059028A1 (enExample)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN109303784B (zh) * 2018-09-30 2020-06-23 山东省文登整骨医院 痛风性关节炎动物模型的构建方法
AU2020267953A1 (en) * 2019-05-08 2021-11-18 Novartis Ag Anti-CD40 antibodies for use in treatment of T1DM and insulitis
EP4029502A1 (en) 2021-01-15 2022-07-20 Ecuphar N.V. Pyrazoline-derived compound (enflicoxib) for use in the prevention and/or treatment of pain and inflammation associated to surgery in mammals
US12208085B2 (en) 2022-05-31 2025-01-28 Ecuphar Nv Pyrazoline-derived compound for use in the prevention and/or treatment of pain and inflammation associated to surgery in mammals

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU773615B2 (en) * 1997-05-05 2004-05-27 Pfizer Inc. COX-2 selective carprofen for treating pain and inflammation in dogs
ES2137138B1 (es) * 1998-05-29 2000-09-16 Esteve Labor Dr Derivados de pirazolinas, su preparacion y su aplicacion como medicamentos.
US20050131028A1 (en) * 2003-09-11 2005-06-16 Pharmacia Corporation Methods and compositions for the extended duration treatment of pain, inflammation and inflammation-related disorders
MX2007010922A (es) * 2005-03-10 2007-10-12 Genentech Inc Metodos y composiciones para modular la integridad vascular.

Also Published As

Publication number Publication date
LT3206684T (lt) 2020-10-12
EP3206684B1 (en) 2020-06-17
EP3009137A1 (en) 2016-04-20
DK3206684T3 (da) 2020-08-10
HRP20201233T1 (hr) 2020-11-13
PT3206684T (pt) 2020-08-24
EP3206684A1 (en) 2017-08-23
JP6655625B2 (ja) 2020-02-26
RS60777B1 (sr) 2020-10-30
PL3206684T3 (pl) 2021-01-11
HUE050511T2 (hu) 2020-12-28
CA2964428C (en) 2022-01-04
CA2964428A1 (en) 2016-04-21
CY1123243T1 (el) 2021-10-29
AR102295A1 (es) 2017-02-15
TWI707678B (zh) 2020-10-21
TW201625239A (zh) 2016-07-16
JP2017531042A (ja) 2017-10-19
US11154536B2 (en) 2021-10-26
ES2828435T3 (es) 2021-05-26
US20170231961A1 (en) 2017-08-17
CN115154465A (zh) 2022-10-11
CN107257684A (zh) 2017-10-17
WO2016059028A1 (en) 2016-04-21
MX2017004899A (es) 2018-02-12
MX376725B (es) 2025-03-07
SMT202000415T1 (it) 2020-11-10

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