SI2849758T1 - Compositions comprising zoledronic acid or related compounds for relieving inflammatory pain and related conditions - Google Patents

Compositions comprising zoledronic acid or related compounds for relieving inflammatory pain and related conditions Download PDF

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Publication number
SI2849758T1
SI2849758T1 SI201330993T SI201330993T SI2849758T1 SI 2849758 T1 SI2849758 T1 SI 2849758T1 SI 201330993 T SI201330993 T SI 201330993T SI 201330993 T SI201330993 T SI 201330993T SI 2849758 T1 SI2849758 T1 SI 2849758T1
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Slovenia
Prior art keywords
zoledronic acid
use according
administered
preparation
mammal
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Application number
SI201330993T
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English (en)
Slovenian (sl)
Inventor
Herriot Tabuteau
Original Assignee
Anatecip Bioventures Ii Llc
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Application filed by Anatecip Bioventures Ii Llc filed Critical Anatecip Bioventures Ii Llc
Publication of SI2849758T1 publication Critical patent/SI2849758T1/en

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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/66Phosphorus compounds
    • A61K31/675Phosphorus compounds having nitrogen as a ring hetero atom, e.g. pyridoxal phosphate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/66Phosphorus compounds
    • A61K31/662Phosphorus acids or esters thereof having P—C bonds, e.g. foscarnet, trichlorfon
    • A61K31/663Compounds having two or more phosphorus acid groups or esters thereof, e.g. clodronic acid, pamidronic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

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  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Physiology (AREA)
  • Nutrition Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
SI201330993T 2012-05-14 2013-05-14 Compositions comprising zoledronic acid or related compounds for relieving inflammatory pain and related conditions SI2849758T1 (en)

Applications Claiming Priority (13)

Application Number Priority Date Filing Date Title
US201261646538P 2012-05-14 2012-05-14
US201261647478P 2012-05-15 2012-05-15
US201261654383P 2012-06-01 2012-06-01
US201261654292P 2012-06-01 2012-06-01
US201261655527P 2012-06-05 2012-06-05
US201261655541P 2012-06-05 2012-06-05
US201361762225P 2013-02-07 2013-02-07
US201361764563P 2013-02-14 2013-02-14
US201361767676P 2013-02-21 2013-02-21
US201361767647P 2013-02-21 2013-02-21
US201361803721P 2013-03-20 2013-03-20
PCT/US2013/040939 WO2013173330A1 (en) 2012-05-14 2013-05-14 Compositions comprising zoledronic acid or related compounds for relieving inflammatory pain and related conditions
EP13791356.2A EP2849758B1 (en) 2012-05-14 2013-05-14 Compositions comprising zoledronic acid or related compounds for relieving inflammatory pain and related conditions

Publications (1)

Publication Number Publication Date
SI2849758T1 true SI2849758T1 (en) 2018-07-31

Family

ID=49549077

Family Applications (1)

Application Number Title Priority Date Filing Date
SI201330993T SI2849758T1 (en) 2012-05-14 2013-05-14 Compositions comprising zoledronic acid or related compounds for relieving inflammatory pain and related conditions

Country Status (21)

Country Link
US (5) US20130303486A1 (https=)
EP (2) EP2849758B1 (https=)
JP (2) JP2015518828A (https=)
KR (3) KR20150035597A (https=)
CN (2) CN109331027A (https=)
AU (3) AU2013262995B2 (https=)
CA (2) CA2987470A1 (https=)
CY (1) CY1120503T1 (https=)
DK (1) DK2849758T3 (https=)
ES (1) ES2667535T3 (https=)
HK (1) HK1255373A1 (https=)
HR (1) HRP20180606T1 (https=)
HU (1) HUE038905T2 (https=)
LT (1) LT2849758T (https=)
NZ (1) NZ702414A (https=)
PL (1) PL2849758T3 (https=)
PT (1) PT2849758T (https=)
RS (1) RS57294B1 (https=)
SI (1) SI2849758T1 (https=)
SM (1) SMT201800212T1 (https=)
WO (1) WO2013173330A1 (https=)

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US10350227B2 (en) 2012-05-14 2019-07-16 Antecip Bioventures Ii Llc Neridronic acid for treating complex regional pain syndrome
US9956234B2 (en) 2012-05-14 2018-05-01 Antecip Bioventures Ii Llc Osteoclast inhibitors for joint conditions
US9669040B2 (en) 2012-05-14 2017-06-06 Antecip Bioventures Ii Llc Compositions for oral administration of zoledronic acid or related compounds for treating complex regional pain syndrome
US9675626B2 (en) 2012-05-14 2017-06-13 Antecip Bioventures Ii Llc Compositions for oral administration of zoledronic acid or related compounds for treating complex regional pain syndrome
US10092581B2 (en) 2014-05-15 2018-10-09 Antecip Bioventures Ii Llc Osteoclast inhibitors such as zoledronic acid for low back pain treatment
US10028969B2 (en) 2012-05-14 2018-07-24 Antecip Bioventures Ii Llc Compositions for oral administration of zoledronic acid or related compounds for treating complex regional pain syndrome
US10413561B2 (en) 2012-05-14 2019-09-17 Antecip Bioventures Ii Llc Neridronic acid and other bisphosphonates for treating complex regional pain syndrome and other diseases
US9770457B2 (en) 2012-05-14 2017-09-26 Antecip Bioventures Ii Llc Neridronic acid for treating bone marrow lesion
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US9795622B2 (en) 2012-05-14 2017-10-24 Antecip Bioventures Ii Llc Neridronic acid for treating pain associated with a joint
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US9694023B2 (en) 2012-05-14 2017-07-04 Antecip Bioventures Ii Llc Methods for the safe administration of imidazole or imidazolium compounds
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US9861648B2 (en) 2012-05-14 2018-01-09 Antecip Boiventures Ii Llc Osteoclast inhibitors for knee conditions
US9662343B2 (en) 2012-05-14 2017-05-30 Antecip Bioventures Ii Llc Compositions for oral administration of zoledronic acid or related compounds for treating complex regional pain syndrome
US9211257B2 (en) 2012-05-14 2015-12-15 Antecip Bioventures Ii Llc Osteoclast inhibitors for knee conditions
US9789128B2 (en) 2012-05-14 2017-10-17 Antecip Bioventures Ii Llc Compositions for oral administration of zoledronic acid or related compounds for treating complex regional pain syndrome
US10111837B2 (en) 2012-05-14 2018-10-30 Antecip Bioventures Ii Llc Dosage forms for oral administration of zoledronic acid or related compounds
US9616078B2 (en) 2012-05-14 2017-04-11 Antecip Bioventures Ii Llc Dosage forms for oral administration of zoledronic acid or related compounds for treating disease
US9867840B2 (en) 2014-05-27 2018-01-16 Antecip Bioventures Ii Llc Compositions for oral administration of zoledronic acid or related compounds for treating complex regional pain syndrome
US10173986B2 (en) 2012-05-14 2019-01-08 Antecip Bioventures Ii Llc Methods for the safe administration of imidazole or imidazolium compounds
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US9700570B2 (en) 2014-05-27 2017-07-11 Antecip Bioventures Ii Llc Compositions for oral administration of zoledronic acid or related compounds for treating complex regional pain syndrome
US10004756B2 (en) 2014-05-15 2018-06-26 Antecip Bioventures Ii Llc Compositions for oral administration of zoledronic acid or related compounds for treating complex regional pain syndrome
US9867839B2 (en) 2012-05-14 2018-01-16 Antecip Bioventures Ii Llc Osteoclast inhibitors for joint conditions
US8802658B2 (en) * 2012-05-14 2014-08-12 Antecip Bioventures Ii Llc Compositions for oral administration of zoledronic acid or related compounds for treating disease
US10034890B2 (en) 2012-05-14 2018-07-31 Antecip Bioventures Ii Llc Compositions for oral administration of zoledronic acid or related compounds for treating complex regional pain syndrome
US9289441B2 (en) 2014-08-08 2016-03-22 Antecip Bioventures Ii Llc Osteoclast inhibitors such as zoledronic acid for low back pain treatment
US9827256B2 (en) 2014-05-27 2017-11-28 Antecip Bioventures Ii Llc Compositions for administration of zoledronic acid or related compounds for treating lower back pain
US9949993B2 (en) 2012-05-14 2018-04-24 Antecip Bioventures Ii Llc Compositions for administration of zoledronic acid or related compounds for treating low back pain
US9655908B2 (en) 2012-05-14 2017-05-23 Antecip Bioventures Ii Llc Neridronic acid molecular complex for treating complex regional pain syndrome
US9956237B2 (en) 2012-05-14 2018-05-01 Antecip Bioventures Ii Llc Osteoclast inhibitors for knee conditions
US10463682B2 (en) 2012-05-14 2019-11-05 Antecip Bioventures Ii Llc Compositions for oral administration of zoledronic acid or related compounds for treating low back pain
US9956238B2 (en) 2014-05-15 2018-05-01 Antecip Bioventures Ii Llc Compositions for administration of zoledronic acid or related compounds for treating low back pain
US10080765B2 (en) 2012-05-14 2018-09-25 Antecip Bioventures Ii Llc Neridronic acid for treating complex regional pain syndrome
US10016445B2 (en) 2012-05-14 2018-07-10 Antecip Bioventures Ii Llc Compositions for oral administration of zoledronic acid or related compounds for treating complex regional pain syndrome
US9782421B1 (en) 2012-05-14 2017-10-10 Antecip Bioventures Ii Llc Neridronic acid molecular complex for treating complex regional pain syndrome
US9895383B2 (en) 2012-05-14 2018-02-20 Antecip Bioventures Ii Llc Compositions for oral administration of zoledronic acid or related compounds for treating complex regional pain syndrome
US8865757B1 (en) 2014-05-28 2014-10-21 Antecip Bioventures Ii Llp Therapeutic compositions comprising imidazole and imidazolium compounds
US9707245B2 (en) 2012-05-14 2017-07-18 Antecip Bioventures Ii Llc Neridronic acid for treating complex regional pain syndrome
US9820999B2 (en) 2012-05-14 2017-11-21 Antecip Bioventures Ii Llc Neridronic acid for treating complex regional pain syndrome
US9901589B2 (en) 2012-05-14 2018-02-27 Antecip Bioventures Ii Llc Compositions for oral administration of zoledronic acid or related compounds for treating complex regional pain syndrome
WO2015184003A1 (en) * 2014-05-27 2015-12-03 Antecip Bioventures Ii Llp Osteoclast inhibitors for pain
US9844559B2 (en) 2012-05-14 2017-12-19 Antecip Bioventures Ii Llc Neridronic acid for treating bone marrow lesions
US9427403B2 (en) 2012-05-14 2016-08-30 Antecip Bioventures Ii Llc Methods for the safe administration of imidazole or imidazolium compounds
US9877977B2 (en) 2012-05-14 2018-01-30 Antecip Bioventures Ii Llc Compositions for oral administration of zoledronic acid or related compounds for treating complex regional pain syndrome
US10016446B2 (en) 2012-05-14 2018-07-10 Antecip Bioventures Ii Llc Compositions for oral administration of zoledronic acid or related compounds for treating Paget's disease of bone
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US9827192B2 (en) 2012-05-14 2017-11-28 Antecip Bioventures Ii Llc Compositions for oral administration of zoledronic acid or related compounds for treating complex regional pain syndrome
US9707247B2 (en) 2012-05-14 2017-07-18 Antecip Bioventures Ii Llc Compositions for administration of zoledronic acid or related compounds for treating low back pain
US9717747B2 (en) 2012-05-14 2017-08-01 Antecip Bioventures Ii Llc Osteoclast inhibitors for knee conditions
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KR20190009428A (ko) * 2013-10-25 2019-01-28 안테씨프 바이오벤쳐스 투 엘엘씨 질병의 치료를 위한, 졸레드론산 또는 관련 화합물의 경구 투여용 조성물
US9079927B1 (en) 2014-05-27 2015-07-14 Antecip Bioventures Ii Llc Substituted imidazolium compounds for treating disease
US20170182072A1 (en) * 2014-05-27 2017-06-29 Antecip Bioventures Ii Llc Compositions for oral administration of zoledronic acid or related compounds for treating complex regional pain syndrome
CN106456610A (zh) * 2014-05-27 2017-02-22 安泰赛普生物风投二代有限责任公司 用于疼痛的破骨细胞抑制剂
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Also Published As

Publication number Publication date
US20130303485A1 (en) 2013-11-14
CA2873742A1 (en) 2013-11-21
EP2849758B1 (en) 2018-04-04
HK1255373A1 (en) 2019-08-16
EP3323418A1 (en) 2018-05-23
HRP20180606T1 (hr) 2018-06-29
AU2018214132B2 (en) 2019-07-11
US20130303486A1 (en) 2013-11-14
JP2015518828A (ja) 2015-07-06
PL2849758T3 (pl) 2018-08-31
NZ702414A (en) 2016-10-28
AU2018214132A1 (en) 2018-08-30
ES2667535T3 (es) 2018-05-11
CA2873742C (en) 2018-01-16
DK2849758T3 (en) 2018-05-14
US20130303488A1 (en) 2013-11-14
SMT201800212T1 (it) 2018-07-17
JP2018127477A (ja) 2018-08-16
CY1120503T1 (el) 2019-07-10
US20160151398A1 (en) 2016-06-02
WO2013173330A1 (en) 2013-11-21
PT2849758T (pt) 2018-05-09
KR20190004381A (ko) 2019-01-11
CA2987470A1 (en) 2013-11-21
KR20160139050A (ko) 2016-12-06
AU2013262995B2 (en) 2016-09-01
CN104349781A (zh) 2015-02-11
EP2849758A4 (en) 2015-12-30
RS57294B1 (sr) 2018-08-31
LT2849758T (lt) 2018-07-25
HUE038905T2 (hu) 2018-12-28
EP2849758A1 (en) 2015-03-25
CN109331027A (zh) 2019-02-15
AU2013262995A1 (en) 2014-12-18
AU2016256701A1 (en) 2016-11-24
US20130303487A1 (en) 2013-11-14
AU2016256701B2 (en) 2018-05-10
KR20150035597A (ko) 2015-04-06

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