SI2848610T1 - Inhibitors of kinase activity - Google Patents

Inhibitors of kinase activity Download PDF

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Publication number
SI2848610T1
SI2848610T1 SI200731975T SI200731975T SI2848610T1 SI 2848610 T1 SI2848610 T1 SI 2848610T1 SI 200731975 T SI200731975 T SI 200731975T SI 200731975 T SI200731975 T SI 200731975T SI 2848610 T1 SI2848610 T1 SI 2848610T1
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SI
Slovenia
Prior art keywords
diseases
disease
compound
pharmaceutical composition
kinase
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SI200731975T
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English (en)
Slovenian (sl)
Inventor
Christopher John Burns
Michael Francis Harte
James T. Palmer
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Ym Biosciences Australia Pty Ltd
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Priority claimed from AU2006906359A external-priority patent/AU2006906359A0/en
Application filed by Ym Biosciences Australia Pty Ltd filed Critical Ym Biosciences Australia Pty Ltd
Publication of SI2848610T1 publication Critical patent/SI2848610T1/en

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    • C07D241/10—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
    • C07D241/14—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D241/20—Nitrogen atoms
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    • A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D213/75—Amino or imino radicals, acylated by carboxylic or carbonic acids, or by sulfur or nitrogen analogues thereof, e.g. carbamates
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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D241/24—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D241/26—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals with nitrogen atoms directly attached to ring carbon atoms
    • C07D241/28—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals with nitrogen atoms directly attached to ring carbon atoms in which said hetero-bound carbon atoms have double bonds to oxygen, sulfur or nitrogen atoms
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SI200731975T 2006-11-15 2007-11-15 Inhibitors of kinase activity SI2848610T1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
AU2006906359A AU2006906359A0 (en) 2006-11-15 Inhibitors of kinase activity
US90151207P 2007-02-14 2007-02-14
EP14181447.5A EP2848610B1 (en) 2006-11-15 2007-11-15 Inhibitors of kinase activity

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SI2848610T1 true SI2848610T1 (en) 2018-02-28

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SI200731975T SI2848610T1 (en) 2006-11-15 2007-11-15 Inhibitors of kinase activity

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US (2) US8461161B2 (enExample)
EP (3) EP2099774A4 (enExample)
JP (5) JP5461189B2 (enExample)
AU (1) AU2007321719B2 (enExample)
CA (1) CA2701959C (enExample)
CY (1) CY1119528T1 (enExample)
DK (1) DK2848610T3 (enExample)
ES (1) ES2645947T3 (enExample)
HK (1) HK1225722A1 (enExample)
HU (1) HUE035868T2 (enExample)
LT (1) LT2848610T (enExample)
PL (1) PL2848610T3 (enExample)
PT (1) PT2848610T (enExample)
SI (1) SI2848610T1 (enExample)
WO (1) WO2008058341A1 (enExample)

Families Citing this family (58)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2431927B (en) 2005-11-04 2010-03-17 Amira Pharmaceuticals Inc 5-Lipoxygenase-activating protein (FLAP) inhibitors
US7977359B2 (en) 2005-11-04 2011-07-12 Amira Pharmaceuticals, Inc. 5-lipdxygenase-activating protein (FLAP) inhibitors
US8399666B2 (en) 2005-11-04 2013-03-19 Panmira Pharmaceuticals, Llc 5-lipoxygenase-activating protein (FLAP) inhibitors
EP2099774A4 (en) * 2006-11-15 2010-11-24 Ym Biosciences Australia Pty L INHIBITORS OF KINASEACTIVITY
WO2008063888A2 (en) 2006-11-22 2008-05-29 Plexxikon, Inc. Compounds modulating c-fms and/or c-kit activity and uses therefor
US20100190777A1 (en) 2007-07-17 2010-07-29 Plexxikon Inc. Compounds and methods for kinase modulation, and indications therefor
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