SI2766381T1 - Postopek za pripravo 17-substituiranih steroidov - Google Patents

Postopek za pripravo 17-substituiranih steroidov

Info

Publication number
SI2766381T1
SI2766381T1 SI201230729A SI201230729A SI2766381T1 SI 2766381 T1 SI2766381 T1 SI 2766381T1 SI 201230729 A SI201230729 A SI 201230729A SI 201230729 A SI201230729 A SI 201230729A SI 2766381 T1 SI2766381 T1 SI 2766381T1
Authority
SI
Slovenia
Prior art keywords
preparing
substituted steroids
steroids
substituted
Prior art date
Application number
SI201230729A
Other languages
English (en)
Inventor
Yvon Derrien
Patricia Poirier
Massimiliano Forcato
Tony Pintus
Livius Cotarca
Sebastien Meunier
Laurence Graindorge
Original Assignee
Zach System, Z.I.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Zach System, Z.I. filed Critical Zach System, Z.I.
Publication of SI2766381T1 publication Critical patent/SI2766381T1/sl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J43/003—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0051—Estrane derivatives
    • C07J1/0059—Estrane derivatives substituted in position 17 by a keto group
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J31/00—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
    • C07J31/003—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring the S atom directly linked to a ring carbon atom of the cyclopenta(a)hydrophenanthrene skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J31/00—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
    • C07J31/006—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring not covered by C07J31/003

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
SI201230729A 2011-10-10 2012-10-09 Postopek za pripravo 17-substituiranih steroidov SI2766381T1 (sl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP11306310 2011-10-10
EP12774995.0A EP2766381B1 (en) 2011-10-10 2012-10-09 Process for preparing 17-substituted steroids
PCT/EP2012/069937 WO2013053691A1 (en) 2011-10-10 2012-10-09 Process for preparing 17-substituted steroids

Publications (1)

Publication Number Publication Date
SI2766381T1 true SI2766381T1 (sl) 2016-11-30

Family

ID=47045010

Family Applications (1)

Application Number Title Priority Date Filing Date
SI201230729A SI2766381T1 (sl) 2011-10-10 2012-10-09 Postopek za pripravo 17-substituiranih steroidov

Country Status (14)

Country Link
US (1) US9353145B2 (sl)
EP (1) EP2766381B1 (sl)
JP (1) JP6091510B2 (sl)
CN (1) CN104066744B (sl)
BR (1) BR112014008671B1 (sl)
CA (1) CA2851330C (sl)
ES (1) ES2590753T3 (sl)
HR (1) HRP20161256T1 (sl)
HU (1) HUE029523T2 (sl)
IL (1) IL231995A (sl)
PL (1) PL2766381T3 (sl)
RS (1) RS55223B1 (sl)
SI (1) SI2766381T1 (sl)
WO (1) WO2013053691A1 (sl)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SG191724A1 (en) 2011-01-11 2013-08-30 Glaxosmithkline Llc Combination
ITMI20121788A1 (it) * 2012-10-22 2014-04-23 Olon Spa Procedimento per la purificazione di abiraterone acetato
EP2945960A2 (en) * 2013-01-18 2015-11-25 Cortendo AB (publ) Abiraterone and analogs thereof for the treatment of diseases associated with cortisol overproduction
EP2792682B1 (en) 2013-04-19 2016-11-09 Zach System Process for producing a solid form of abiraterone acetate
ES2705579T3 (es) 2013-06-28 2019-03-26 Scinopharm Taiwan Ltd Procedimiento de preparación de abiraterona e intermedios de la misma
CN106061481B (zh) * 2013-10-01 2019-08-16 诺华股份有限公司 用于治疗癌症的雄激素受体抑制剂与akt抑制剂的组合
US9556219B2 (en) 2014-01-28 2017-01-31 Olon S.P.A. Procedure for the preparation of abiraterone acetate and intermediates thereof
US10722527B2 (en) 2015-04-10 2020-07-28 Capsugel Belgium Nv Abiraterone acetate lipid formulations
ITUB20155309A1 (it) * 2015-10-27 2017-04-27 Olon Spa Procedimento per la preparazione di abiraterone acetato e suoi intermedi
CN105503992A (zh) * 2016-01-22 2016-04-20 江苏联环药业股份有限公司 一种醋酸阿比特龙的制备方法
WO2018071544A1 (en) * 2016-10-11 2018-04-19 Zhuhai Beihai Biotech Co., Ltd. Abiraterone derivative and formulations thereof
CN108948120A (zh) * 2018-07-07 2018-12-07 张正光 一种醋酸阿比特龙中间体的制备方法
CN111349138B (zh) * 2018-12-24 2023-06-16 江苏恒瑞医药股份有限公司 制备醋酸阿比特龙的方法
CN114026106A (zh) 2019-03-06 2022-02-08 普洛拉治疗公司 阿比特龙前药
CN112812147A (zh) * 2019-11-15 2021-05-18 江苏佳尔科药业集团股份有限公司 一种醋酸阿比特龙的合成方法及其中间体
CA3207282A1 (en) 2021-02-15 2022-08-18 Matthew J. Sharp Abiraterone prodrugs

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2742331B2 (ja) * 1992-03-31 1998-04-22 ブリテイツシユ・テクノロジー・グループ・リミテツド 癌治療に有用な１７位置換ステロイド
GB2282377B (en) 1993-09-30 1997-09-03 British Tech Group Synthesis of 17-(3-pyridyl) steroids
PL1781683T3 (pl) 2004-08-24 2012-04-30 Btg Int Ltd Sposób wytwarzania 17-winylo-trifluorometanosulfonianów jako związków pośrednich
GB0418900D0 (en) 2004-08-24 2004-09-29 Btg Int Ltd Novel salt forms
CN101768199B (zh) 2009-12-24 2014-03-26 深圳万乐药业有限公司 醋酸阿比特龙的多晶型物及其制备方法

Also Published As

Publication number Publication date
CN104066744B (zh) 2017-03-22
CA2851330A1 (en) 2013-04-18
IL231995A (en) 2016-05-31
JP6091510B2 (ja) 2017-03-08
JP2014528461A (ja) 2014-10-27
EP2766381B1 (en) 2016-07-27
WO2013053691A1 (en) 2013-04-18
CA2851330C (en) 2019-07-16
BR112014008671B1 (pt) 2022-07-12
HRP20161256T1 (hr) 2016-11-18
US20140256932A1 (en) 2014-09-11
US9353145B2 (en) 2016-05-31
BR112014008671A2 (pt) 2017-04-18
ES2590753T3 (es) 2016-11-23
EP2766381A1 (en) 2014-08-20
CN104066744A (zh) 2014-09-24
RS55223B1 (sr) 2017-02-28
PL2766381T3 (pl) 2016-12-30
HUE029523T2 (en) 2017-03-28

Similar Documents

Publication Publication Date Title
PL2766381T3 (pl) Sposób wytwarzania steroidów podstawionych w pozycji 17
EP2940004A4 (en) PROCESS FOR PRODUCING OXIME
EP2699534A4 (en) PROCESS FOR PRODUCING TRANS-1233zd
GB201103499D0 (en) Process
GB201107072D0 (en) Process
PT2751073T (pt) Processo para a preparação de isocianatos
IL227872A0 (en) A process for the preparation of n-converted phenylhydroxylamines
GB201101370D0 (en) Process
EP2922820A4 (en) PROCESS FOR PREPARING CRYSTALLINE SORAFENIB TOSYLATE
ZA201402624B (en) Process for preparing buprenorphine
ZA201207386B (en) Process for preparing benzoxaboroles
EP2841444A4 (en) PROCESS FOR PREPARING 17-SUBSTITUTED STEROIDS
ZA201403736B (en) Process for the preparation of sterol derivatives
GB201107073D0 (en) Process
EP2740719A4 (en) PROCESS FOR THE PREPARATION OF A-FLUOROALDEHYDE
EP2619174A4 (en) PROCESS FOR THE PREPARATION OF L-PHENYL-3-DIMETHYLAMINOPROPANE DERIVATIVES
EP2585436A4 (en) PROCESS FOR THE PREPARATION OF 4-HYDROXYPYRIDINES
EP2669293A4 (en) PROCESS FOR THE PRODUCTION OF ROCURONIUM
EP2855433A4 (en) PROCESS FOR THE PREPARATION OF DIHALOPYRIDINES
EP2819995A4 (en) PROCESS FOR THE PREPARATION OF 3-METHYLSULFONYLPROPIONITRIL
IL223145A0 (en) Process for preparing dithiine-tetracarboxy-diimides
EP2938625A4 (en) PROCESS FOR ABIRATERONACETATE
EP2940000A4 (en) PROCESS FOR THE PREPARATION OF METHYL ACETATE
GB201103092D0 (en) Process
IL233626A (en) Process for making chloroamines