SI2406253T1 - Derivati benzofuranila, uporabljeni kot inhibitorji glukokinaze - Google Patents

Derivati benzofuranila, uporabljeni kot inhibitorji glukokinaze

Info

Publication number
SI2406253T1
SI2406253T1 SI201030278T SI201030278T SI2406253T1 SI 2406253 T1 SI2406253 T1 SI 2406253T1 SI 201030278 T SI201030278 T SI 201030278T SI 201030278 T SI201030278 T SI 201030278T SI 2406253 T1 SI2406253 T1 SI 2406253T1
Authority
SI
Slovenia
Prior art keywords
derivatives used
glucokinase inhibitors
benzofuranyl derivatives
benzofuranyl
glucokinase
Prior art date
Application number
SI201030278T
Other languages
English (en)
Inventor
Anthony Lai Ling
Jeffrey Allen Pfefferkorn
Original Assignee
Pfizer Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=42124287&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SI2406253(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer Inc. filed Critical Pfizer Inc.
Publication of SI2406253T1 publication Critical patent/SI2406253T1/sl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4965—Non-condensed pyrazines
    • A61K31/497—Non-condensed pyrazines containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
SI201030278T 2009-03-11 2010-03-04 Derivati benzofuranila, uporabljeni kot inhibitorji glukokinaze SI2406253T1 (sl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US15909909P 2009-03-11 2009-03-11
EP10708644.9A EP2406253B1 (en) 2009-03-11 2010-03-04 Benzofuranyl derivatives used as glucokinase inhibitors
PCT/IB2010/050943 WO2010103437A1 (en) 2009-03-11 2010-03-04 Benzofuranyl derivatives used as glucokinase inhibitors

Publications (1)

Publication Number Publication Date
SI2406253T1 true SI2406253T1 (sl) 2013-09-30

Family

ID=42124287

Family Applications (1)

Application Number Title Priority Date Filing Date
SI201030278T SI2406253T1 (sl) 2009-03-11 2010-03-04 Derivati benzofuranila, uporabljeni kot inhibitorji glukokinaze

Country Status (38)

Country Link
US (2) US8455496B2 (sl)
EP (2) EP2406253B1 (sl)
JP (1) JP5086480B2 (sl)
KR (1) KR101295937B1 (sl)
CN (1) CN102388038B (sl)
AP (1) AP3179A (sl)
AR (1) AR075729A1 (sl)
AU (1) AU2010222589B2 (sl)
BR (1) BRPI1013246B1 (sl)
CA (1) CA2754681C (sl)
CL (1) CL2011002185A1 (sl)
CO (1) CO6430427A2 (sl)
CR (1) CR20110467A (sl)
CU (1) CU24036B1 (sl)
DK (1) DK2406253T3 (sl)
DO (1) DOP2011000279A (sl)
EA (1) EA018894B1 (sl)
EC (1) ECSP11011306A (sl)
ES (1) ES2427279T3 (sl)
GE (1) GEP20156239B (sl)
HK (1) HK1164281A1 (sl)
HR (1) HRP20130661T1 (sl)
IL (1) IL214942A (sl)
MA (1) MA33119B1 (sl)
MY (1) MY151246A (sl)
NI (1) NI201100166A (sl)
NZ (1) NZ595024A (sl)
PE (1) PE20120668A1 (sl)
PL (1) PL2406253T3 (sl)
PT (1) PT2406253E (sl)
RS (1) RS52903B (sl)
SI (1) SI2406253T1 (sl)
TN (1) TN2011000454A1 (sl)
TW (1) TWI383981B (sl)
UA (1) UA99882C2 (sl)
UY (1) UY32480A (sl)
WO (1) WO2010103437A1 (sl)
ZA (1) ZA201106632B (sl)

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RS52903B (en) 2014-02-28
EP2604604A1 (en) 2013-06-19
AU2010222589A1 (en) 2011-09-22
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NI201100166A (es) 2012-01-23
DK2406253T3 (da) 2013-08-12
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WO2010103437A1 (en) 2010-09-16
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MA33119B1 (fr) 2012-03-01
US20100234285A1 (en) 2010-09-16
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TN2011000454A1 (fr) 2013-03-27
BRPI1013246B1 (pt) 2019-10-01
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