SI2167502T1 - Derivati oskadizola in njihova uporaba kot ojačevalci -842 receptorja metabotropskega glutamata - Google Patents

Derivati oskadizola in njihova uporaba kot ojačevalci -842 receptorja metabotropskega glutamata

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Publication number
SI2167502T1
SI2167502T1 SI200830807T SI200830807T SI2167502T1 SI 2167502 T1 SI2167502 T1 SI 2167502T1 SI 200830807 T SI200830807 T SI 200830807T SI 200830807 T SI200830807 T SI 200830807T SI 2167502 T1 SI2167502 T1 SI 2167502T1
Authority
SI
Slovenia
Prior art keywords
glutamate receptor
metabotropic glutamate
oxadiazole derivatives
receptor potentiators
potentiators
Prior art date
Application number
SI200830807T
Other languages
English (en)
Slovenian (sl)
Inventor
Joshua Clayton
Ian Egle
James Empfield
James Folmer
Methvin Isaac
Fupeng Ma
Abdelmalik Slassi
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=40093925&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SI2167502(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of SI2167502T1 publication Critical patent/SI2167502T1/sl

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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
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    • A61P13/00—Drugs for disorders of the urinary system
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    • A61P19/00—Drugs for skeletal disorders
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    • A61P21/00—Drugs for disorders of the muscular or neuromuscular system
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00—Drugs for disorders of the muscular or neuromuscular system
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    • A—HUMAN NECESSITIES
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    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
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    • A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
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    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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    • A61P35/00—Antineoplastic agents
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    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/12—Antidiuretics, e.g. drugs for diabetes insipidus
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    • A61P9/00—Drugs for disorders of the cardiovascular system
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08—Bridged systems

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  • Health & Medical Sciences (AREA)
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  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Addiction (AREA)
  • Urology & Nephrology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Psychology (AREA)
  • Cardiology (AREA)
  • Diabetes (AREA)
  • Hospice & Palliative Care (AREA)
  • Vascular Medicine (AREA)
  • Anesthesiology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Rheumatology (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Epidemiology (AREA)
SI200830807T 2007-06-07 2008-06-05 Derivati oskadizola in njihova uporaba kot ojačevalci -842 receptorja metabotropskega glutamata SI2167502T1 (sl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US94255307P 2007-06-07 2007-06-07
PCT/SE2008/050666 WO2008150233A1 (en) 2007-06-07 2008-06-05 Oxadiazole derivatives and their use as metabotropic glutamate receptor potentiators - 842
EP08779348.5A EP2167502B3 (en) 2007-06-07 2008-06-05 Oxadiazole derivatives and their use as metabotropic glutamate receptor potentiators - 842

Publications (1)

Publication Number Publication Date
SI2167502T1 true SI2167502T1 (sl) 2012-12-31

Family

ID=40093925

Family Applications (2)

Application Number Title Priority Date Filing Date
SI200830807T SI2167502T1 (sl) 2007-06-07 2008-06-05 Derivati oskadizola in njihova uporaba kot ojačevalci -842 receptorja metabotropskega glutamata
SI200831385T SI2444399T1 (sl) 2007-06-07 2008-06-05 Derivati oksadizola in njihova uporaba kot potenciator metabotropskega receptorja glutamata -842

Family Applications After (1)

Application Number Title Priority Date Filing Date
SI200831385T SI2444399T1 (sl) 2007-06-07 2008-06-05 Derivati oksadizola in njihova uporaba kot potenciator metabotropskega receptorja glutamata -842

Country Status (33)

Country Link
US (2) US8377940B2 (enExample)
EP (2) EP2167502B3 (enExample)
JP (2) JP5416696B2 (enExample)
KR (2) KR20150116907A (enExample)
CN (2) CN102977086B (enExample)
AR (1) AR066882A1 (enExample)
AU (1) AU2008260717B2 (enExample)
BR (1) BRPI0812889A2 (enExample)
CA (1) CA2690856C (enExample)
CL (1) CL2008001667A1 (enExample)
CO (1) CO6251287A2 (enExample)
CY (2) CY1113422T1 (enExample)
DK (2) DK2444399T3 (enExample)
EC (1) ECSP109856A (enExample)
ES (2) ES2531443T3 (enExample)
HR (2) HRP20120909T4 (enExample)
IL (1) IL202158A (enExample)
ME (1) ME01488B (enExample)
MX (1) MX2009013078A (enExample)
MY (1) MY158066A (enExample)
NZ (1) NZ582445A (enExample)
PE (1) PE20090328A1 (enExample)
PL (2) PL2444399T3 (enExample)
PT (2) PT2444399E (enExample)
RS (2) RS52526B2 (enExample)
RU (2) RU2470931C2 (enExample)
SA (1) SA08290344B1 (enExample)
SI (2) SI2167502T1 (enExample)
TW (1) TWI417100B (enExample)
UA (1) UA99129C2 (enExample)
UY (1) UY31124A1 (enExample)
WO (1) WO2008150233A1 (enExample)
ZA (1) ZA200908285B (enExample)

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US20130203995A1 (en) * 2010-01-07 2013-08-08 Astrazeneca Ab Process for Making a Metabotropic Glutamate Receptor Positive Allosteric Modulator - 874
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