NZ582445A - OXADIAZOLE DERIVATIVES AND THEIR USE AS mGluR POTENTIATORS - 842 - Google Patents

OXADIAZOLE DERIVATIVES AND THEIR USE AS mGluR POTENTIATORS - 842

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Publication number
NZ582445A
NZ582445A NZ582445A NZ58244508A NZ582445A NZ 582445 A NZ582445 A NZ 582445A NZ 582445 A NZ582445 A NZ 582445A NZ 58244508 A NZ58244508 A NZ 58244508A NZ 582445 A NZ582445 A NZ 582445A
Authority
NZ
New Zealand
Prior art keywords
compound according
pharmaceutically acceptable
methyl
chloro
solvate
Prior art date
Application number
NZ582445A
Other languages
English (en)
Inventor
James Folmer
Joshua Clayton
Ian Egle
James Empfield
Methvin Isaac
Fupeng Ma
Abdelmalik Slassi
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=40093925&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NZ582445(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of NZ582445A publication Critical patent/NZ582445A/en

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    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
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    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08—Bridged systems

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  • Health & Medical Sciences (AREA)
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  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Addiction (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Diabetes (AREA)
  • Urology & Nephrology (AREA)
  • Psychology (AREA)
  • Cardiology (AREA)
  • Vascular Medicine (AREA)
  • Rheumatology (AREA)
  • Hospice & Palliative Care (AREA)
  • Ophthalmology & Optometry (AREA)
  • Anesthesiology (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Epidemiology (AREA)
NZ582445A 2007-06-07 2008-06-05 OXADIAZOLE DERIVATIVES AND THEIR USE AS mGluR POTENTIATORS - 842 NZ582445A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US94255307P 2007-06-07 2007-06-07
PCT/SE2008/050666 WO2008150233A1 (en) 2007-06-07 2008-06-05 Oxadiazole derivatives and their use as metabotropic glutamate receptor potentiators - 842

Publications (1)

Publication Number Publication Date
NZ582445A true NZ582445A (en) 2012-03-30

Family

ID=40093925

Family Applications (1)

Application Number Title Priority Date Filing Date
NZ582445A NZ582445A (en) 2007-06-07 2008-06-05 OXADIAZOLE DERIVATIVES AND THEIR USE AS mGluR POTENTIATORS - 842

Country Status (33)

Country Link
US (2) US8377940B2 (enExample)
EP (2) EP2167502B3 (enExample)
JP (2) JP5416696B2 (enExample)
KR (2) KR20100017640A (enExample)
CN (2) CN101679403B (enExample)
AR (1) AR066882A1 (enExample)
AU (1) AU2008260717B2 (enExample)
BR (1) BRPI0812889A2 (enExample)
CA (1) CA2690856C (enExample)
CL (1) CL2008001667A1 (enExample)
CO (1) CO6251287A2 (enExample)
CY (2) CY1113422T1 (enExample)
DK (2) DK2444399T3 (enExample)
EC (1) ECSP109856A (enExample)
ES (2) ES2393425T7 (enExample)
HR (2) HRP20120909T4 (enExample)
IL (1) IL202158A (enExample)
ME (1) ME01488B (enExample)
MX (1) MX2009013078A (enExample)
MY (1) MY158066A (enExample)
NZ (1) NZ582445A (enExample)
PE (1) PE20090328A1 (enExample)
PL (2) PL2167502T6 (enExample)
PT (2) PT2444399E (enExample)
RS (2) RS53845B1 (enExample)
RU (2) RU2470931C2 (enExample)
SA (1) SA08290344B1 (enExample)
SI (2) SI2444399T1 (enExample)
TW (1) TWI417100B (enExample)
UA (1) UA99129C2 (enExample)
UY (1) UY31124A1 (enExample)
WO (1) WO2008150233A1 (enExample)
ZA (1) ZA200908285B (enExample)

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