SI1000072T1 - Postopek za pripravo (2-((8,9)-diokso-2,6-diazabiciklo(5.2.0)-non-1(7)- en-2-il)-etil) fosforjeve (III) kisline - Google Patents

Postopek za pripravo (2-((8,9)-diokso-2,6-diazabiciklo(5.2.0)-non-1(7)- en-2-il)-etil) fosforjeve (III) kisline

Info

Publication number
SI1000072T1
SI1000072T1 SI9830362T SI9830362T SI1000072T1 SI 1000072 T1 SI1000072 T1 SI 1000072T1 SI 9830362 T SI9830362 T SI 9830362T SI 9830362 T SI9830362 T SI 9830362T SI 1000072 T1 SI1000072 T1 SI 1000072T1
Authority
SI
Slovenia
Prior art keywords
ethyl
dioxo
ester
phosphonic acid
diazabicyclo
Prior art date
Application number
SI9830362T
Other languages
English (en)
Inventor
Andre Alfred Asselin
William Alvin Kinney
Jean Schmid
Original Assignee
Wyeth
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wyeth filed Critical Wyeth
Publication of SI1000072T1 publication Critical patent/SI1000072T1/sl

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/645Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having two nitrogen atoms as the only ring hetero atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/28Phosphorus compounds with one or more P—C bonds
    • C07F9/38Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
    • C07F9/40Esters thereof
    • C07F9/4003Esters thereof the acid moiety containing a substituent or a structure which is considered as characteristic
    • C07F9/4006Esters of acyclic acids which can have further substituents on alkyl

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
SI9830362T 1997-08-01 1998-07-31 Postopek za pripravo (2-((8,9)-diokso-2,6-diazabiciklo(5.2.0)-non-1(7)- en-2-il)-etil) fosforjeve (III) kisline SI1000072T1 (sl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US90509197A 1997-08-01 1997-08-01
EP98937292A EP1000072B1 (en) 1997-08-01 1998-07-31 Process for the preparation of [2-((8,9)- dioxo-2,6-diazabicyclo [5.2.0]-non-1(7)-en-2-yl)-ethyl] phosphonic acid
PCT/US1998/015841 WO1999006417A1 (en) 1997-08-01 1998-07-31 Process for the preparation of [2-((8,9)- dioxo-2,6-diazabicyclo [5.2.0]-non-1(7)-en-2-yl)-ethyl] phosphonic acid

Publications (1)

Publication Number Publication Date
SI1000072T1 true SI1000072T1 (sl) 2003-06-30

Family

ID=25420284

Family Applications (1)

Application Number Title Priority Date Filing Date
SI9830362T SI1000072T1 (sl) 1997-08-01 1998-07-31 Postopek za pripravo (2-((8,9)-diokso-2,6-diazabiciklo(5.2.0)-non-1(7)- en-2-il)-etil) fosforjeve (III) kisline

Country Status (19)

Country Link
EP (1) EP1000072B1 (sl)
JP (1) JP4383651B2 (sl)
KR (1) KR100606580B1 (sl)
CN (2) CN1257174C (sl)
AT (1) ATE232875T1 (sl)
AU (1) AU746119B2 (sl)
BR (1) BR9811807A (sl)
CA (1) CA2297411C (sl)
DE (1) DE69811507T2 (sl)
DK (1) DK1000072T3 (sl)
ES (1) ES2190091T3 (sl)
HK (1) HK1027814A1 (sl)
HU (1) HUP0002505A3 (sl)
IL (2) IL134082A0 (sl)
NO (1) NO325420B1 (sl)
NZ (1) NZ502509A (sl)
RU (1) RU2205834C2 (sl)
SI (1) SI1000072T1 (sl)
WO (1) WO1999006417A1 (sl)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UA78529C2 (en) 2001-10-10 2007-04-10 Wyeth Corp Derivatives of [[2-(amino-3,4-dioxo-1-cyclobutene-1-yl)amino]alkyl] acid for treating pain
DE602004029146D1 (de) 2003-04-09 2010-10-28 Wyeth Llc Derivate von 2-(8,9-dioxo-2,6-diazabicyclo(5.2.0)non-1(7)-en-2-yl)alkylphosphonsäure und deren verwendung als n-methyl-d-aspartat- (nmda-) rezeptorantagonisten
GT200400213A (es) 2003-10-22 2007-09-05 Metodos para la preparacion del acido {2-[(8,9)-dioxo-2,6-diaza-biciclo[5.2.0]-non-1(7)-en-2-il]etil} fosfonico y esteres del mismo
CA2754390A1 (en) * 2009-03-19 2010-09-23 Wyeth Llc Methods for the preparation of [2-(8,9-dioxo-2,6-diazabicyclo[5.2.0]non-1(7)-en-2-yl)ethyl]phosphonic acid and precursors thereof

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5168103A (en) * 1991-01-22 1992-12-01 American Home Products Corporation [[2-(amino-3,4-dioxo-1-cyclobuten-1-yl) amino]alkyl]-acid derivatives

Also Published As

Publication number Publication date
IL163574A (en) 2008-06-05
NO325420B1 (no) 2008-04-21
CN1257174C (zh) 2006-05-24
ES2190091T3 (es) 2003-07-16
NO20000488L (no) 2000-01-31
JP4383651B2 (ja) 2009-12-16
WO1999006417A1 (en) 1999-02-11
EP1000072A1 (en) 2000-05-17
JP2001512129A (ja) 2001-08-21
CA2297411C (en) 2008-12-02
DE69811507D1 (de) 2003-03-27
KR20010022492A (ko) 2001-03-15
IL134082A0 (en) 2001-04-30
NO20000488D0 (no) 2000-01-31
AU746119B2 (en) 2002-04-18
CN1265664A (zh) 2000-09-06
CN1526714A (zh) 2004-09-08
CA2297411A1 (en) 1999-02-11
ATE232875T1 (de) 2003-03-15
HUP0002505A3 (en) 2002-02-28
RU2205834C2 (ru) 2003-06-10
HK1027814A1 (en) 2001-01-23
KR100606580B1 (ko) 2006-08-01
DK1000072T3 (da) 2003-04-22
DE69811507T2 (de) 2003-07-24
IL163574A0 (en) 2005-12-18
NZ502509A (en) 2002-08-28
EP1000072B1 (en) 2003-02-19
CN1149218C (zh) 2004-05-12
BR9811807A (pt) 2000-08-15
HUP0002505A2 (hu) 2000-11-28
AU8603798A (en) 1999-02-22

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