SG47565A1 - Improved process for the synthesis of N-[3-(1H-imidazol-1-yl)phenyl-4-(substituted)-2-pyrimidinamines - Google Patents
Improved process for the synthesis of N-[3-(1H-imidazol-1-yl)phenyl-4-(substituted)-2-pyrimidinaminesInfo
- Publication number
- SG47565A1 SG47565A1 SG1996002850A SG1996002850A SG47565A1 SG 47565 A1 SG47565 A1 SG 47565A1 SG 1996002850 A SG1996002850 A SG 1996002850A SG 1996002850 A SG1996002850 A SG 1996002850A SG 47565 A1 SG47565 A1 SG 47565A1
- Authority
- SG
- Singapore
- Prior art keywords
- imidazol
- substituted
- phenyl
- pyrimidinamines
- synthesis
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Photoreceptors In Electrophotography (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Pyridine Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US07/514,455 US5064963A (en) | 1990-04-25 | 1990-04-25 | Process for the synthesis of n-(3-(1h-imidazol-1-yl)phenyl-4-(substituted)-2-pyrimidinamines |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SG47565A1 true SG47565A1 (en) | 1998-04-17 |
Family
ID=24047219
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SG1996002850A SG47565A1 (en) | 1990-04-25 | 1991-02-27 | Improved process for the synthesis of N-[3-(1H-imidazol-1-yl)phenyl-4-(substituted)-2-pyrimidinamines |
Country Status (19)
| Country | Link |
|---|---|
| US (1) | US5064963A (de) |
| EP (1) | EP0453731B1 (de) |
| JP (1) | JPH04225975A (de) |
| KR (1) | KR0168679B1 (de) |
| AT (1) | ATE170184T1 (de) |
| AU (1) | AU630849B2 (de) |
| CA (1) | CA2041031A1 (de) |
| DE (1) | DE69130029T2 (de) |
| DK (1) | DK0453731T3 (de) |
| ES (1) | ES2121757T3 (de) |
| FI (1) | FI100533B (de) |
| GR (1) | GR3027762T3 (de) |
| HU (1) | HU211774B (de) |
| IE (1) | IE911366A1 (de) |
| NO (1) | NO177567C (de) |
| NZ (1) | NZ237870A (de) |
| SG (1) | SG47565A1 (de) |
| TW (1) | TW215087B (de) |
| ZA (1) | ZA913092B (de) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5521184A (en) * | 1992-04-03 | 1996-05-28 | Ciba-Geigy Corporation | Pyrimidine derivatives and processes for the preparation thereof |
| US5516775A (en) * | 1992-08-31 | 1996-05-14 | Ciba-Geigy Corporation | Further use of pyrimidine derivatives |
| BRPI9909191B8 (pt) * | 1998-03-27 | 2021-07-06 | Janssen Pharmaceutica Nv | derivados de pirimidina inibidores do hiv, seu uso e composição farmacêutica que os compreende |
| PT1225874E (pt) | 1999-09-24 | 2006-06-30 | Janssen Pharmaceutica Nv | Composicoes antivirais. |
| CA2628474A1 (en) * | 2005-11-03 | 2007-05-10 | Sgx Pharmaceuticals, Inc. | Pyrimidinyl-thiophene kinase modulators |
| KR20090130345A (ko) * | 2007-05-04 | 2009-12-22 | 아이알엠 엘엘씨 | Ｃ-ｋｉｔ 및 ｐｄｇｆｒ 키나제 억제제로서의 화합물 및 조성물 |
| WO2013192125A1 (en) * | 2012-06-20 | 2013-12-27 | Merck Sharp & Dohme Corp. | Pyrazolyl derivatives as syk inhibitors |
| US9487504B2 (en) | 2012-06-20 | 2016-11-08 | Merck Sharp & Dohme Corp. | Imidazolyl analogs as syk inhibitors |
| CN110330447B (zh) * | 2019-07-16 | 2022-04-15 | 北京赛升药业股份有限公司 | 一种甲磺酸萘莫司他中间体的制备方法及其应用 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU5319479A (en) * | 1978-12-22 | 1980-06-26 | Ici Australia Limited | Pyrimidinyl amino phenoxy carboxylate derivatives |
| EP0164204A1 (de) * | 1984-05-12 | 1985-12-11 | FISONS plc | Pharmazeutisch nützliche Pyrimidine |
| US4788195A (en) * | 1986-01-13 | 1988-11-29 | American Cyanamid Company | 4,5,6-substituted-N-(substituted-phenyl)-2-pyrimidinamines |
-
1990
- 1990-04-25 US US07/514,455 patent/US5064963A/en not_active Expired - Fee Related
-
1991
- 1991-02-27 DE DE69130029T patent/DE69130029T2/de not_active Expired - Fee Related
- 1991-02-27 ES ES91102859T patent/ES2121757T3/es not_active Expired - Lifetime
- 1991-02-27 EP EP91102859A patent/EP0453731B1/de not_active Expired - Lifetime
- 1991-02-27 AT AT91102859T patent/ATE170184T1/de active
- 1991-02-27 DK DK91102859T patent/DK0453731T3/da active
- 1991-02-27 SG SG1996002850A patent/SG47565A1/en unknown
- 1991-03-22 TW TW080102248A patent/TW215087B/zh active
- 1991-04-18 NZ NZ237870A patent/NZ237870A/xx unknown
- 1991-04-23 JP JP3117918A patent/JPH04225975A/ja active Pending
- 1991-04-23 CA CA002041031A patent/CA2041031A1/en not_active Abandoned
- 1991-04-24 FI FI911983A patent/FI100533B/fi active
- 1991-04-24 NO NO911632A patent/NO177567C/no unknown
- 1991-04-24 HU HU911373A patent/HU211774B/hu not_active IP Right Cessation
- 1991-04-24 ZA ZA913092A patent/ZA913092B/xx unknown
- 1991-04-24 IE IE136691A patent/IE911366A1/en unknown
- 1991-04-24 KR KR1019910006612A patent/KR0168679B1/ko not_active IP Right Cessation
- 1991-04-24 AU AU75905/91A patent/AU630849B2/en not_active Ceased
-
1998
- 1998-08-27 GR GR980401941T patent/GR3027762T3/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| EP0453731B1 (de) | 1998-08-26 |
| DK0453731T3 (da) | 1999-02-15 |
| HU211774B (en) | 1995-12-28 |
| NO177567C (no) | 1995-10-11 |
| NO911632D0 (no) | 1991-04-24 |
| CA2041031A1 (en) | 1991-10-26 |
| ES2121757T3 (es) | 1998-12-16 |
| JPH04225975A (ja) | 1992-08-14 |
| FI911983A0 (fi) | 1991-04-24 |
| KR910018375A (ko) | 1991-11-30 |
| GR3027762T3 (en) | 1998-11-30 |
| FI911983A (fi) | 1991-10-26 |
| EP0453731A3 (en) | 1992-09-02 |
| FI100533B (fi) | 1997-12-31 |
| EP0453731A2 (de) | 1991-10-30 |
| NO911632L (no) | 1991-10-28 |
| ZA913092B (en) | 1992-02-26 |
| DE69130029T2 (de) | 1999-02-18 |
| KR0168679B1 (ko) | 1999-01-15 |
| IE911366A1 (en) | 1991-11-06 |
| US5064963A (en) | 1991-11-12 |
| DE69130029D1 (de) | 1998-10-01 |
| HUT57719A (en) | 1991-12-30 |
| AU630849B2 (en) | 1992-11-05 |
| NZ237870A (en) | 1993-05-26 |
| HU911373D0 (en) | 1991-10-28 |
| ATE170184T1 (de) | 1998-09-15 |
| TW215087B (de) | 1993-10-21 |
| AU7590591A (en) | 1991-11-07 |
| NO177567B (no) | 1995-07-03 |
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