SG171752A1 - Directly compressible granular microcrystalline cellulose based excipient, manufacturing process and use thereof - Google Patents
Directly compressible granular microcrystalline cellulose based excipient, manufacturing process and use thereof Download PDFInfo
- Publication number
- SG171752A1 SG171752A1 SG2011035789A SG2011035789A SG171752A1 SG 171752 A1 SG171752 A1 SG 171752A1 SG 2011035789 A SG2011035789 A SG 2011035789A SG 2011035789 A SG2011035789 A SG 2011035789A SG 171752 A1 SG171752 A1 SG 171752A1
- Authority
- SG
- Singapore
- Prior art keywords
- binder
- excipient
- microcrystalline cellulose
- slurry
- disintegrant
- Prior art date
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- 239000000546 pharmaceutical excipient Substances 0.000 title claims abstract description 215
- 229920000168 Microcrystalline cellulose Polymers 0.000 title claims abstract description 146
- 235000019813 microcrystalline cellulose Nutrition 0.000 title claims abstract description 145
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- 238000004519 manufacturing process Methods 0.000 title claims description 24
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| KR101298788B1 (ko) * | 2011-03-15 | 2013-08-22 | 보령제약 주식회사 | 안정성이 개선된 복합제제 |
| US9642807B2 (en) * | 2012-04-27 | 2017-05-09 | Japan Corn Starch Co., Ltd | Method for producing starch granules, and orally disinitegrating tablet |
| SI2968529T1 (sl) | 2013-03-14 | 2021-03-31 | Aimmune Therapeutics, Inc. | Izdelava arašidovih formulacij arašida za ustno desenzibilizacijo |
| US9492535B2 (en) | 2013-03-14 | 2016-11-15 | Aimmune Therapeutics, Inc. | Peanut formulations and uses thereof |
| WO2015187736A1 (en) * | 2014-06-02 | 2015-12-10 | Allergen Research Corporation | Placebo formulations and uses thereof |
| CN104189915B (zh) * | 2014-07-30 | 2016-08-10 | 上海新亚药业闵行有限公司 | 一种固体制剂预混剂及其制备方法 |
| CN104258411A (zh) * | 2014-09-19 | 2015-01-07 | 安徽山河药用辅料股份有限公司 | 一种硅化微晶纤维素复合辅料及其制备方法 |
| CN106265077A (zh) * | 2015-05-30 | 2017-01-04 | 天士力制药集团股份有限公司 | 一种中药浸膏雾化分散工艺及其制剂 |
| JP6650750B2 (ja) * | 2015-12-22 | 2020-02-19 | アサヒグループ食品株式会社 | 錠剤の製造方法、錠剤原料用顆粒の製造方法、及び錠剤原料用顆粒 |
| EP3836801A4 (en) | 2018-08-16 | 2022-05-18 | Société des Produits Nestlé S.A. | Peanut oral immunotherapy with maintenance dose |
| CN113891722A (zh) | 2018-12-20 | 2022-01-04 | 爱沐疗法公司 | 用于漏服剂量的花生口服免疫疗法给药计划表 |
| EP3965815A4 (en) | 2019-05-10 | 2023-05-31 | Société des Produits Nestlé S.A. | METHOD OF IMPROVING THE QUALITY OF LIFE IN A PEANUT ALLERGY PATIENT |
| EP3993646B1 (en) | 2019-07-05 | 2023-08-16 | Swedish Match North Europe AB | An oral pouched nicotine product including a filling material comprising nicotine-containing particles |
| HUE066565T2 (hu) | 2019-11-20 | 2024-08-28 | Swedish Match North Europe Ab | Orálisan alkalmazható tasakos nikotintermék, beleértve egy nikotinrészecskéket tartalmazó töltõanyagot |
| PL4018848T3 (pl) | 2020-12-22 | 2024-11-25 | Swedish Match North Europe Ab | Wyrób w saszetkach do użytku doustnego zawierający materiał pokrywający przepuszczalny dla cieczy oraz materiał wypełniający |
| CN116036291B (zh) * | 2022-08-31 | 2025-08-26 | 瑞普（天津）生物药业有限公司 | 一种具有增溶作用的组合物及其制备方法与应用 |
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| DE3505433A1 (de) * | 1985-02-16 | 1986-08-21 | Basf Ag, 6700 Ludwigshafen | Direkttablettierhilfsmittel |
| CA2126441C (en) * | 1991-12-30 | 1999-12-21 | David F. Erkoboni | Microcrystalline cellulose spheronization composition |
| US5686107A (en) * | 1995-01-30 | 1997-11-11 | Fmc Corporation | Chewable pharmaceutical tablets |
| DE19628617A1 (de) * | 1996-07-16 | 1998-01-22 | Basf Ag | Direkttablettierhilfsmittel |
| ES2301223T3 (es) * | 1999-07-19 | 2008-06-16 | Fit Gmbh | Producto polisacaridico coprocesado con carboximetilcelulosa insoluble. |
| AU2002211018B2 (en) * | 2000-11-06 | 2004-08-05 | Asahi Kasei Kabushiki Kaisha | Cellulosic particle for pharmaceutical preparation |
| US20040213839A1 (en) * | 2001-02-05 | 2004-10-28 | Andrew Favara | Methods and compositions for reducing the taste of pharmaceutically active agents |
| NZ556465A (en) * | 2005-02-03 | 2010-10-29 | Nycomed Pharma As | Fast wet-massing method for the preparation of calcium-containing compositions |
| WO2008020990A1 (en) * | 2006-08-09 | 2008-02-21 | Mallinckrodt Baker, Inc. | New direct compressible excipient blend |
| US8932629B2 (en) * | 2006-10-27 | 2015-01-13 | Fmc Corporation | Co-processed microcrystalline cellulose and sugar alcohol as an excipient for tablet formulations |
| NZ584521A (en) * | 2007-10-10 | 2011-03-31 | Avantor Performance Mat Inc | Directly compressible high functionality granular microcrystalline cellulose based excipient, manufacturing process and use thereof |
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2009
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- 2009-11-16 US US12/998,659 patent/US20110288146A1/en not_active Abandoned
- 2009-11-16 JP JP2011537526A patent/JP2012509329A/ja active Pending
- 2009-11-16 CN CN2009801461591A patent/CN102215825A/zh active Pending
- 2009-11-16 BR BRPI0921507A patent/BRPI0921507A2/pt not_active IP Right Cessation
- 2009-11-16 EP EP09752702A patent/EP2376067A2/en not_active Ceased
- 2009-11-16 CA CA2744142A patent/CA2744142A1/en not_active Abandoned
- 2009-11-16 SG SG2011035789A patent/SG171752A1/en unknown
- 2009-11-16 MX MX2011005168A patent/MX2011005168A/es not_active Application Discontinuation
- 2009-11-16 KR KR1020117013939A patent/KR20110089180A/ko not_active Ceased
- 2009-11-16 AU AU2009316812A patent/AU2009316812A1/en not_active Abandoned
- 2009-11-19 TW TW098139345A patent/TW201023897A/zh unknown
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2011
- 2011-05-17 IL IL212955A patent/IL212955A0/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| MX2011005168A (es) | 2011-05-30 |
| US20110288146A1 (en) | 2011-11-24 |
| CA2744142A1 (en) | 2010-05-27 |
| KR20110089180A (ko) | 2011-08-04 |
| WO2010059534A3 (en) | 2011-01-20 |
| EP2376067A2 (en) | 2011-10-19 |
| WO2010059534A2 (en) | 2010-05-27 |
| TW201023897A (en) | 2010-07-01 |
| IL212955A0 (en) | 2011-07-31 |
| JP2012509329A (ja) | 2012-04-19 |
| AU2009316812A1 (en) | 2011-07-07 |
| CN102215825A (zh) | 2011-10-12 |
| BRPI0921507A2 (pt) | 2016-01-19 |
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