SG149880A1 - Novel inhibitors of chymase - Google Patents

Novel inhibitors of chymase

Info

Publication number
SG149880A1
SG149880A1 SG200900530-7A SG2009005307A SG149880A1 SG 149880 A1 SG149880 A1 SG 149880A1 SG 2009005307 A SG2009005307 A SG 2009005307A SG 149880 A1 SG149880 A1 SG 149880A1
Authority
SG
Singapore
Prior art keywords
chymase
novel inhibitors
methods
intermediates
derivatives
Prior art date
Application number
SG200900530-7A
Other languages
English (en)
Inventor
Michael J Hawkins
Michael N Greco
Eugene Powell
Bruce E Maryanoff
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of SG149880A1 publication Critical patent/SG149880A1/en

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    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6561—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings
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    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/28—Phosphorus compounds with one or more P—C bonds
    • C07F9/30—Phosphinic acids [R2P(=O)(OH)]; Thiophosphinic acids ; [R2P(=X1)(X2H) (X1, X2 are each independently O, S or Se)]
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SG200900530-7A 2004-01-23 2005-01-18 Novel inhibitors of chymase SG149880A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US53866304P 2004-01-23 2004-01-23

Publications (1)

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SG149880A1 true SG149880A1 (en) 2009-02-27

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SG200900530-7A SG149880A1 (en) 2004-01-23 2005-01-18 Novel inhibitors of chymase

Country Status (24)

Country Link
US (2) US7459444B2 (ko)
EP (1) EP1716160B1 (ko)
JP (1) JP5022711B2 (ko)
KR (1) KR101182143B1 (ko)
CN (2) CN1934120B (ko)
AR (1) AR047448A1 (ko)
AT (1) ATE493421T1 (ko)
AU (1) AU2005207856B2 (ko)
BR (1) BRPI0507052A (ko)
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JP2010506928A (ja) * 2006-10-18 2010-03-04 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ チマーゼの新インヒビター
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JP5587914B2 (ja) 2009-01-30 2014-09-10 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング キマーゼ阻害剤として有用なアザキナゾリンジオン
JP5690286B2 (ja) * 2009-03-04 2015-03-25 イデニク プハルマセウティカルス，インコーポレイテッド ホスホチオフェン及びホスホチアゾールｈｃｖポリメラーゼ阻害剤
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CN108383875B (zh) * 2018-03-22 2020-04-28 昆明学院 一种银催化的3-膦酰甲基吲哚啉及制备方法

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KR20060129401A (ko) 2006-12-15
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IL177037A0 (en) 2006-12-10
AU2005207856A1 (en) 2005-08-11
ECSP066721A (es) 2006-10-31
CA2554205C (en) 2013-08-27
US20050176769A1 (en) 2005-08-11
NZ548684A (en) 2009-04-30
US7459444B2 (en) 2008-12-02
EP1716160B1 (en) 2010-12-29
EA200601358A1 (ru) 2007-02-27
NO20063647L (no) 2006-10-19
WO2005073214A3 (en) 2005-10-20
BRPI0507052A (pt) 2007-06-12
TW200539881A (en) 2005-12-16
JP5022711B2 (ja) 2012-09-12
ZA200607024B (en) 2010-02-24
HK1148753A1 (en) 2011-09-16
ATE493421T1 (de) 2011-01-15
CN101863923A (zh) 2010-10-20
CN1934120A (zh) 2007-03-21
CR8563A (es) 2009-01-14
EA011745B1 (ru) 2009-06-30
KR101182143B1 (ko) 2012-09-13
CN1934120B (zh) 2010-05-26
AR047448A1 (es) 2006-01-18
WO2005073214A2 (en) 2005-08-11
DE602005025600D1 (de) 2011-02-10
IL177037A (en) 2013-05-30
MXPA06008375A (es) 2007-03-21
US20090036409A1 (en) 2009-02-05
JP2007518807A (ja) 2007-07-12
ES2357013T3 (es) 2011-04-15
CA2554205A1 (en) 2005-08-11
EP1716160A2 (en) 2006-11-02

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