SG148023A1 - New benzothiazine and benzothiadiazine compounds, a process for their preparation and pharmaceutical compositions containing them - Google Patents

New benzothiazine and benzothiadiazine compounds, a process for their preparation and pharmaceutical compositions containing them

Info

Publication number
SG148023A1
SG148023A1 SG200404677-7A SG2004046777A SG148023A1 SG 148023 A1 SG148023 A1 SG 148023A1 SG 2004046777 A SG2004046777 A SG 2004046777A SG 148023 A1 SG148023 A1 SG 148023A1
Authority
SG
Singapore
Prior art keywords
preparation
represents hydrogen
pharmaceutical compositions
compositions containing
alkyl
Prior art date
Application number
SG200404677-7A
Other languages
English (en)
Inventor
Patrice Desos
Alex Cordi
Pierre Lestage
Original Assignee
Servier Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Servier Lab filed Critical Servier Lab
Publication of SG148023A1 publication Critical patent/SG148023A1/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
SG200404677-7A 2003-06-13 2004-06-07 New benzothiazine and benzothiadiazine compounds, a process for their preparation and pharmaceutical compositions containing them SG148023A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0307118A FR2856065B1 (fr) 2003-06-13 2003-06-13 Nouveaux derives de benzothiazine et benzothiadiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent.

Publications (1)

Publication Number Publication Date
SG148023A1 true SG148023A1 (en) 2008-12-31

Family

ID=33186482

Family Applications (1)

Application Number Title Priority Date Filing Date
SG200404677-7A SG148023A1 (en) 2003-06-13 2004-06-07 New benzothiazine and benzothiadiazine compounds, a process for their preparation and pharmaceutical compositions containing them

Country Status (28)

Country Link
US (2) US7253162B2 (es)
EP (1) EP1486503B1 (es)
JP (1) JP2005002114A (es)
KR (1) KR100586683B1 (es)
CN (1) CN1277823C (es)
AR (1) AR044672A1 (es)
AT (1) ATE344265T1 (es)
AU (1) AU2004202586A1 (es)
BR (1) BRPI0401956A (es)
CA (1) CA2470263A1 (es)
CY (1) CY1105939T1 (es)
DE (1) DE602004002990T2 (es)
DK (1) DK1486503T3 (es)
EA (1) EA008797B1 (es)
EG (1) EG24207A (es)
ES (1) ES2276249T3 (es)
FR (1) FR2856065B1 (es)
GE (1) GEP20063815B (es)
HK (1) HK1071750A1 (es)
HR (1) HRP20070030T3 (es)
MA (1) MA27092A1 (es)
MX (1) MXPA04005580A (es)
NO (1) NO20042422L (es)
NZ (1) NZ533472A (es)
PL (1) PL1486503T3 (es)
PT (1) PT1486503E (es)
SG (1) SG148023A1 (es)
SI (1) SI1486503T1 (es)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2879201B1 (fr) * 2004-12-10 2007-02-16 Servier Lab Nouveaux derives de benzothiazine et benzothiadiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
US7939528B2 (en) 2005-10-13 2011-05-10 Glaxosmithkline Llc Heterocycle compounds
JP2010502706A (ja) * 2006-09-07 2010-01-28 ミレニアム・ファーマシューティカルズ・インコーポレイテッド キナーゼ阻害活性を有するフェネチルアミド誘導体
GB0821166D0 (en) * 2008-11-19 2008-12-24 Glaxo Group Ltd Compounds
FR2955106B1 (fr) * 2010-01-08 2011-12-23 Servier Lab Nouveaux derives de benzothiadiazines cyclopropylees, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
EP2813508B1 (en) * 2012-02-08 2018-01-31 Takeda Pharmaceutical Company Limited Heterocyclic compound and use thereof
WO2019130229A1 (en) * 2017-12-28 2019-07-04 Mylan Laboratories Ltd Methods and intermediates for preparing rucaparib

Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5536719A (en) * 1994-07-12 1996-07-16 Adir Et Compagnie Benzothiadiazine compound
US20020161222A1 (en) * 2001-04-18 2002-10-31 Elsa Foucher Process for the synthesis of (3aS)-5,5-dioxo-2,3,3a,4-tetrahydro-1H-pyrrolo[2,1-c][1,2,4] benzothiadiazine
WO2003053979A1 (fr) * 2001-12-21 2003-07-03 Les Laboratoires Servier Nouveaux derives de benzothiazine et benzothiadiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1377693A (fr) * 1962-12-06 1964-11-06 Geigy Ag J R Nouveaux composés dibenzo [1.2] thiaziniques et produits pesticides qui en contiennent
ZA991301B (en) * 1998-02-18 1999-09-13 Neurosearch As Glutamate receptor modulators.
FR2833950B1 (fr) * 2001-12-21 2005-12-16 Servier Lab Nouveaux derives de benzothiazine et de benzothiadiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent

Patent Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5536719A (en) * 1994-07-12 1996-07-16 Adir Et Compagnie Benzothiadiazine compound
US20020161222A1 (en) * 2001-04-18 2002-10-31 Elsa Foucher Process for the synthesis of (3aS)-5,5-dioxo-2,3,3a,4-tetrahydro-1H-pyrrolo[2,1-c][1,2,4] benzothiadiazine
WO2003053979A1 (fr) * 2001-12-21 2003-07-03 Les Laboratoires Servier Nouveaux derives de benzothiazine et benzothiadiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
US20050124606A1 (en) * 2001-12-21 2005-06-09 Alex Cordi Novel benzothiazine and benzothiadiazine derivatives method for preparing same and pharmaceutical compositions containing same

Also Published As

Publication number Publication date
KR100586683B1 (ko) 2006-06-08
PT1486503E (pt) 2007-01-31
EA200400666A2 (ru) 2004-12-30
PL1486503T3 (pl) 2006-12-29
EG24207A (en) 2008-10-21
AU2004202586A1 (en) 2005-01-06
BRPI0401956A (pt) 2005-06-28
EP1486503A1 (fr) 2004-12-15
AR044672A1 (es) 2005-09-21
EA008797B1 (ru) 2007-08-31
US20070249594A1 (en) 2007-10-25
US20040254161A1 (en) 2004-12-16
JP2005002114A (ja) 2005-01-06
EA200400666A3 (ru) 2005-10-27
ATE344265T1 (de) 2006-11-15
FR2856065B1 (fr) 2005-08-19
DK1486503T3 (da) 2007-02-26
CY1105939T1 (el) 2011-04-06
CN1572791A (zh) 2005-02-02
GEP20063815B (en) 2006-05-10
NO20042422L (no) 2004-12-14
ES2276249T3 (es) 2007-06-16
FR2856065A1 (fr) 2004-12-17
MA27092A1 (fr) 2004-12-20
US7423034B2 (en) 2008-09-09
DE602004002990T2 (de) 2007-07-05
KR20040107410A (ko) 2004-12-20
SI1486503T1 (sl) 2007-02-28
EP1486503B1 (fr) 2006-11-02
CA2470263A1 (fr) 2004-12-13
CN1277823C (zh) 2006-10-04
MXPA04005580A (es) 2005-03-23
US7253162B2 (en) 2007-08-07
HRP20070030T3 (en) 2007-08-31
HK1071750A1 (en) 2005-07-29
NZ533472A (en) 2005-09-30
DE602004002990D1 (de) 2006-12-14

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