CY1105939T1 - Παραγωγα βενζοθειαζινης και βενζοθεαδιαζινης, μεθοδος παρασκευης αυτων και φαρμακευτικες συνθεσεις οι οποιες τα πepιεχουν - Google Patents

Παραγωγα βενζοθειαζινης και βενζοθεαδιαζινης, μεθοδος παρασκευης αυτων και φαρμακευτικες συνθεσεις οι οποιες τα πepιεχουν

Info

Publication number
CY1105939T1
CY1105939T1 CY20071100074T CY071100074T CY1105939T1 CY 1105939 T1 CY1105939 T1 CY 1105939T1 CY 20071100074 T CY20071100074 T CY 20071100074T CY 071100074 T CY071100074 T CY 071100074T CY 1105939 T1 CY1105939 T1 CY 1105939T1
Authority
CY
Cyprus
Prior art keywords
benzotheadiazine
benzothiazine
derivatives
preparation
pharmaceutical compositions
Prior art date
Application number
CY20071100074T
Other languages
English (en)
Inventor
Patrice Desos
Alex Cordi
Pierre Lestage
Original Assignee
Les Laboratoires Servier
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Les Laboratoires Servier filed Critical Les Laboratoires Servier
Publication of CY1105939T1 publication Critical patent/CY1105939T1/el

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Psychology (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

Abstract

Ενώσεις του τύπου (1):
CY20071100074T 2003-06-13 2007-01-16 Παραγωγα βενζοθειαζινης και βενζοθεαδιαζινης, μεθοδος παρασκευης αυτων και φαρμακευτικες συνθεσεις οι οποιες τα πepιεχουν CY1105939T1 (el)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0307118A FR2856065B1 (fr) 2003-06-13 2003-06-13 Nouveaux derives de benzothiazine et benzothiadiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent.

Publications (1)

Publication Number Publication Date
CY1105939T1 true CY1105939T1 (el) 2011-04-06

Family

ID=33186482

Family Applications (1)

Application Number Title Priority Date Filing Date
CY20071100074T CY1105939T1 (el) 2003-06-13 2007-01-16 Παραγωγα βενζοθειαζινης και βενζοθεαδιαζινης, μεθοδος παρασκευης αυτων και φαρμακευτικες συνθεσεις οι οποιες τα πepιεχουν

Country Status (28)

Country Link
US (2) US7253162B2 (el)
EP (1) EP1486503B1 (el)
JP (1) JP2005002114A (el)
KR (1) KR100586683B1 (el)
CN (1) CN1277823C (el)
AR (1) AR044672A1 (el)
AT (1) ATE344265T1 (el)
AU (1) AU2004202586A1 (el)
BR (1) BRPI0401956A (el)
CA (1) CA2470263A1 (el)
CY (1) CY1105939T1 (el)
DE (1) DE602004002990T2 (el)
DK (1) DK1486503T3 (el)
EA (1) EA008797B1 (el)
EG (1) EG24207A (el)
ES (1) ES2276249T3 (el)
FR (1) FR2856065B1 (el)
GE (1) GEP20063815B (el)
HK (1) HK1071750A1 (el)
HR (1) HRP20070030T3 (el)
MA (1) MA27092A1 (el)
MX (1) MXPA04005580A (el)
NO (1) NO20042422L (el)
NZ (1) NZ533472A (el)
PL (1) PL1486503T3 (el)
PT (1) PT1486503E (el)
SG (1) SG148023A1 (el)
SI (1) SI1486503T1 (el)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2879201B1 (fr) * 2004-12-10 2007-02-16 Servier Lab Nouveaux derives de benzothiazine et benzothiadiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
US7939528B2 (en) 2005-10-13 2011-05-10 Glaxosmithkline Llc Heterocycle compounds
JP2010502706A (ja) * 2006-09-07 2010-01-28 ミレニアム・ファーマシューティカルズ・インコーポレイテッド キナーゼ阻害活性を有するフェネチルアミド誘導体
GB0821166D0 (en) * 2008-11-19 2008-12-24 Glaxo Group Ltd Compounds
FR2955106B1 (fr) * 2010-01-08 2011-12-23 Servier Lab Nouveaux derives de benzothiadiazines cyclopropylees, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
JP6134654B2 (ja) * 2012-02-08 2017-05-24 武田薬品工業株式会社 複素環化合物およびその用途
WO2019130229A1 (en) * 2017-12-28 2019-07-04 Mylan Laboratories Ltd Methods and intermediates for preparing rucaparib

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1377693A (fr) * 1962-12-06 1964-11-06 Geigy Ag J R Nouveaux composés dibenzo [1.2] thiaziniques et produits pesticides qui en contiennent
FR2722502B1 (fr) * 1994-07-12 1996-08-23 Adir Nouveau derive de benzothiadiazine, son procede depreparation et les compositions pharmaceutiques qui le contiennent
HUP0101280A3 (en) * 1998-02-18 2003-02-28 Neurosearch As Positive ampa receptor modulator compounds and their use
FR2823753B1 (fr) * 2001-04-18 2004-07-16 Servier Lab Nouveau procede de synthese de la (3as)-5,5-dioxo-2,3,3a, 4-tetrahydro-1h-pyrrolo [2,1-c] [1,2,4] benzothiadiazine
FR2833950B1 (fr) * 2001-12-21 2005-12-16 Servier Lab Nouveaux derives de benzothiazine et de benzothiadiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
FR2833956B1 (fr) * 2001-12-21 2004-01-30 Servier Lab Nouveaux derives de benzothiazine et de benzothiadiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent

Also Published As

Publication number Publication date
US7253162B2 (en) 2007-08-07
PT1486503E (pt) 2007-01-31
AU2004202586A1 (en) 2005-01-06
NZ533472A (en) 2005-09-30
PL1486503T3 (pl) 2006-12-29
ATE344265T1 (de) 2006-11-15
NO20042422L (no) 2004-12-14
EA200400666A2 (ru) 2004-12-30
EP1486503B1 (fr) 2006-11-02
CN1277823C (zh) 2006-10-04
CN1572791A (zh) 2005-02-02
SG148023A1 (en) 2008-12-31
MXPA04005580A (es) 2005-03-23
CA2470263A1 (fr) 2004-12-13
DK1486503T3 (da) 2007-02-26
ES2276249T3 (es) 2007-06-16
EG24207A (en) 2008-10-21
EA008797B1 (ru) 2007-08-31
GEP20063815B (en) 2006-05-10
EP1486503A1 (fr) 2004-12-15
FR2856065A1 (fr) 2004-12-17
KR20040107410A (ko) 2004-12-20
FR2856065B1 (fr) 2005-08-19
DE602004002990T2 (de) 2007-07-05
BRPI0401956A (pt) 2005-06-28
MA27092A1 (fr) 2004-12-20
SI1486503T1 (sl) 2007-02-28
US20070249594A1 (en) 2007-10-25
AR044672A1 (es) 2005-09-21
HRP20070030T3 (en) 2007-08-31
US20040254161A1 (en) 2004-12-16
US7423034B2 (en) 2008-09-09
DE602004002990D1 (de) 2006-12-14
HK1071750A1 (en) 2005-07-29
KR100586683B1 (ko) 2006-06-08
EA200400666A3 (ru) 2005-10-27
JP2005002114A (ja) 2005-01-06

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