CY1105939T1 - Παραγωγα βενζοθειαζινης και βενζοθεαδιαζινης, μεθοδος παρασκευης αυτων και φαρμακευτικες συνθεσεις οι οποιες τα πepιεχουν - Google Patents
Παραγωγα βενζοθειαζινης και βενζοθεαδιαζινης, μεθοδος παρασκευης αυτων και φαρμακευτικες συνθεσεις οι οποιες τα πepιεχουνInfo
- Publication number
- CY1105939T1 CY1105939T1 CY20071100074T CY071100074T CY1105939T1 CY 1105939 T1 CY1105939 T1 CY 1105939T1 CY 20071100074 T CY20071100074 T CY 20071100074T CY 071100074 T CY071100074 T CY 071100074T CY 1105939 T1 CY1105939 T1 CY 1105939T1
- Authority
- CY
- Cyprus
- Prior art keywords
- benzotheadiazine
- benzothiazine
- derivatives
- preparation
- pharmaceutical compositions
- Prior art date
Links
- UJVBZCCNLAAMOV-UHFFFAOYSA-N 2h-1,2-benzothiazine Chemical compound C1=CC=C2C=CNSC2=C1 UJVBZCCNLAAMOV-UHFFFAOYSA-N 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Psychology (AREA)
- Hospice & Palliative Care (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Abstract
Ενώσεις του τύπου (1):
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0307118A FR2856065B1 (fr) | 2003-06-13 | 2003-06-13 | Nouveaux derives de benzothiazine et benzothiadiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent. |
Publications (1)
Publication Number | Publication Date |
---|---|
CY1105939T1 true CY1105939T1 (el) | 2011-04-06 |
Family
ID=33186482
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CY20071100074T CY1105939T1 (el) | 2003-06-13 | 2007-01-16 | Παραγωγα βενζοθειαζινης και βενζοθεαδιαζινης, μεθοδος παρασκευης αυτων και φαρμακευτικες συνθεσεις οι οποιες τα πepιεχουν |
Country Status (28)
Country | Link |
---|---|
US (2) | US7253162B2 (el) |
EP (1) | EP1486503B1 (el) |
JP (1) | JP2005002114A (el) |
KR (1) | KR100586683B1 (el) |
CN (1) | CN1277823C (el) |
AR (1) | AR044672A1 (el) |
AT (1) | ATE344265T1 (el) |
AU (1) | AU2004202586A1 (el) |
BR (1) | BRPI0401956A (el) |
CA (1) | CA2470263A1 (el) |
CY (1) | CY1105939T1 (el) |
DE (1) | DE602004002990T2 (el) |
DK (1) | DK1486503T3 (el) |
EA (1) | EA008797B1 (el) |
EG (1) | EG24207A (el) |
ES (1) | ES2276249T3 (el) |
FR (1) | FR2856065B1 (el) |
GE (1) | GEP20063815B (el) |
HK (1) | HK1071750A1 (el) |
HR (1) | HRP20070030T3 (el) |
MA (1) | MA27092A1 (el) |
MX (1) | MXPA04005580A (el) |
NO (1) | NO20042422L (el) |
NZ (1) | NZ533472A (el) |
PL (1) | PL1486503T3 (el) |
PT (1) | PT1486503E (el) |
SG (1) | SG148023A1 (el) |
SI (1) | SI1486503T1 (el) |
Families Citing this family (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2879201B1 (fr) * | 2004-12-10 | 2007-02-16 | Servier Lab | Nouveaux derives de benzothiazine et benzothiadiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
US7939528B2 (en) | 2005-10-13 | 2011-05-10 | Glaxosmithkline Llc | Heterocycle compounds |
JP2010502706A (ja) * | 2006-09-07 | 2010-01-28 | ミレニアム・ファーマシューティカルズ・インコーポレイテッド | キナーゼ阻害活性を有するフェネチルアミド誘導体 |
GB0821166D0 (en) * | 2008-11-19 | 2008-12-24 | Glaxo Group Ltd | Compounds |
FR2955106B1 (fr) * | 2010-01-08 | 2011-12-23 | Servier Lab | Nouveaux derives de benzothiadiazines cyclopropylees, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
JP6134654B2 (ja) * | 2012-02-08 | 2017-05-24 | 武田薬品工業株式会社 | 複素環化合物およびその用途 |
WO2019130229A1 (en) * | 2017-12-28 | 2019-07-04 | Mylan Laboratories Ltd | Methods and intermediates for preparing rucaparib |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR1377693A (fr) * | 1962-12-06 | 1964-11-06 | Geigy Ag J R | Nouveaux composés dibenzo [1.2] thiaziniques et produits pesticides qui en contiennent |
FR2722502B1 (fr) * | 1994-07-12 | 1996-08-23 | Adir | Nouveau derive de benzothiadiazine, son procede depreparation et les compositions pharmaceutiques qui le contiennent |
HUP0101280A3 (en) * | 1998-02-18 | 2003-02-28 | Neurosearch As | Positive ampa receptor modulator compounds and their use |
FR2823753B1 (fr) * | 2001-04-18 | 2004-07-16 | Servier Lab | Nouveau procede de synthese de la (3as)-5,5-dioxo-2,3,3a, 4-tetrahydro-1h-pyrrolo [2,1-c] [1,2,4] benzothiadiazine |
FR2833950B1 (fr) * | 2001-12-21 | 2005-12-16 | Servier Lab | Nouveaux derives de benzothiazine et de benzothiadiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
FR2833956B1 (fr) * | 2001-12-21 | 2004-01-30 | Servier Lab | Nouveaux derives de benzothiazine et de benzothiadiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
-
2003
- 2003-06-13 FR FR0307118A patent/FR2856065B1/fr not_active Expired - Fee Related
-
2004
- 2004-06-04 MA MA27721A patent/MA27092A1/fr unknown
- 2004-06-07 SG SG200404677-7A patent/SG148023A1/en unknown
- 2004-06-09 MX MXPA04005580A patent/MXPA04005580A/es active IP Right Grant
- 2004-06-09 AT AT04291435T patent/ATE344265T1/de not_active IP Right Cessation
- 2004-06-09 SI SI200430111T patent/SI1486503T1/sl unknown
- 2004-06-09 EP EP04291435A patent/EP1486503B1/fr active Active
- 2004-06-09 ES ES04291435T patent/ES2276249T3/es active Active
- 2004-06-09 PT PT04291435T patent/PT1486503E/pt unknown
- 2004-06-09 DK DK04291435T patent/DK1486503T3/da active
- 2004-06-09 PL PL04291435T patent/PL1486503T3/pl unknown
- 2004-06-09 DE DE602004002990T patent/DE602004002990T2/de not_active Expired - Fee Related
- 2004-06-10 NO NO20042422A patent/NO20042422L/no not_active Application Discontinuation
- 2004-06-10 US US10/865,184 patent/US7253162B2/en not_active Expired - Fee Related
- 2004-06-10 EG EG2004060261A patent/EG24207A/xx active
- 2004-06-11 AU AU2004202586A patent/AU2004202586A1/en not_active Abandoned
- 2004-06-11 CA CA002470263A patent/CA2470263A1/fr not_active Abandoned
- 2004-06-11 EA EA200400666A patent/EA008797B1/ru not_active IP Right Cessation
- 2004-06-11 KR KR1020040042991A patent/KR100586683B1/ko not_active IP Right Cessation
- 2004-06-11 AR ARP040102023A patent/AR044672A1/es unknown
- 2004-06-11 NZ NZ533472A patent/NZ533472A/en unknown
- 2004-06-11 GE GE5557A patent/GEP20063815B/en unknown
- 2004-06-14 CN CNB2004100482744A patent/CN1277823C/zh not_active Expired - Fee Related
- 2004-06-14 JP JP2004175278A patent/JP2005002114A/ja active Pending
- 2004-06-14 BR BR0401956-3A patent/BRPI0401956A/pt not_active IP Right Cessation
-
2005
- 2005-05-30 HK HK05104495A patent/HK1071750A1/xx not_active IP Right Cessation
-
2007
- 2007-01-16 CY CY20071100074T patent/CY1105939T1/el unknown
- 2007-02-01 HR HR20070030T patent/HRP20070030T3/xx unknown
- 2007-06-27 US US11/823,439 patent/US7423034B2/en not_active Expired - Fee Related
Also Published As
Similar Documents
Publication | Publication Date | Title |
---|---|---|
CY1108754T1 (el) | Νεα παραγωγα θειοφαινογλυκοσιδης, μεθοδος για την παρασκευη τους, φαρμακα περιεχοντα αυτες τις ενωσεις και η χρηση τους | |
ATE296826T1 (de) | Pyrazolo(1,5)pyridinderivate | |
CY1110034T1 (el) | Παραγωγα 1,2,4,5-τετραϋδρο-3h-βενζαζεπινων, μεθοδος παρασκευης αυτων και οι φαρμακευτικες συνθεσεις που τα περιεχουν | |
CY1116372T1 (el) | Φαρμακευτικα σκευασματα που περιεχουν μεθυλναλτρεξονη | |
CY1109227T1 (el) | Παραγωγα της 5-φαινυλο-4-μεθυλο-θειαζολ-2-υλ-αμινης ως αναστολεις των ενζυμων κινασης της φωσφατιδυλινοσιτολης 3 (p13) για την θεραπεια των φλεγμονωδων ασθενειων των αεραγωγων | |
CY1106383T1 (el) | Νεες διφαινζυλαζητιδινονες, η διαδικασια για την παραγωγη τους, τα φαρμακευτικα παρασκευασματα που πepιεχουν τις ενωσεις τους καθως και η χρηση τους για την αντιμετωπιση των διαταραχων μεταβολισμου λιπιδιων | |
CY1108522T1 (el) | Μεθοδος συνθεσης της περινδοπριλης και των φαρμακευτικως αποδεκτων αλατων της | |
CY1105617T1 (el) | Νεα αρωματικα παραγωγα των φθορογλυκοσιδων, φαρμακα περιεχοντα αυτες τις ενωσεις και η χρηση τους | |
CY1107301T1 (el) | Ιμιδαζο και θειαζολοπυριδινες ως αναστολεις κινασης jak3 | |
JO2353B1 (en) | New derivatives of mixed-ring fluoroglycosides and drugs containing these compounds and their use | |
CY1113011T1 (el) | Νεα κρυσταλλικη μορφη v της αγομελατινης, μεθοδος παρασκευης αυτης και φαρμακευτικες συνθεσεις που περιεχουν αυτην | |
NO20054787L (no) | Indenderivater som farmasotiske midler | |
CY1108529T1 (el) | Νεα αζαδικυκλικα παραγωγα, μεθοδος παρασκευης τους και φαρμακευτικες συνθεσεις που τα περιεχουν | |
CY1105939T1 (el) | Παραγωγα βενζοθειαζινης και βενζοθεαδιαζινης, μεθοδος παρασκευης αυτων και φαρμακευτικες συνθεσεις οι οποιες τα πepιεχουν | |
CY1112960T1 (el) | Παραγωγα ουριας, μεθοδοι για την παρασκευη τους και χρησεις αυτων | |
IL173810A0 (en) | Imidazopyridine derivatives and pharmaceutical compositions containing the same | |
SE0302192D0 (sv) | Novel compounds | |
CY1106544T1 (el) | Μεθοδος συνθεσεως υπερινδοπριλης και τα φαρμακευτικως αποδεκτα αλατα αυτης | |
CY1107028T1 (el) | Παραγωγα ινδανυλ-πιπεραζινων μεθοδος παρασκευης αυτων και οι φαρμακευτικες συνθεσεις που τα περιεχουν | |
ATE300541T1 (de) | Pyrazolopyridinderivate | |
NO20040881L (no) | Orale antidiabetes midler. | |
SE0302139D0 (sv) | Novel compounds | |
CR10974A (es) | Inhibidores de carboxipeptidasa b plasmatica (divisional) | |
NO20043016L (no) | 6-aminomorfinan-derivater, fremgangsmate for fremstilling og anvendelse derav | |
CY1106376T1 (el) | Δικυκλικα παραγωγα των αμινο-πυραζινονων, μεθοδος παρασκευης τους και οι φαρμακευτικες συνθεσεις που τα πepιεχουν |