EA200400667A2 - Новые соединения бензотиазина и бензотиадиазина, способ их получения и фармацевтические композиции, которые их содержат - Google Patents

Новые соединения бензотиазина и бензотиадиазина, способ их получения и фармацевтические композиции, которые их содержат

Info

Publication number
EA200400667A2
EA200400667A2 EA200400667A EA200400667A EA200400667A2 EA 200400667 A2 EA200400667 A2 EA 200400667A2 EA 200400667 A EA200400667 A EA 200400667A EA 200400667 A EA200400667 A EA 200400667A EA 200400667 A2 EA200400667 A2 EA 200400667A2
Authority
EA
Eurasian Patent Office
Prior art keywords
processes
preparation
pharmaceutical compositions
compositions containing
benzothiadiazine compounds
Prior art date
Application number
EA200400667A
Other languages
English (en)
Other versions
EA009522B1 (ru
EA200400667A3 (ru
Inventor
Патрик Десо
Алекс Корди
Пьер Лестаж
Original Assignee
Ле Лаборатуар Сервье
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ле Лаборатуар Сервье filed Critical Ле Лаборатуар Сервье
Publication of EA200400667A2 publication Critical patent/EA200400667A2/ru
Publication of EA200400667A3 publication Critical patent/EA200400667A3/ru
Publication of EA009522B1 publication Critical patent/EA009522B1/ru

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Abstract

Соединения формулы (I)в которой Rпредставляет собой гетероцикл,Rпредставляет собой водород, галоген или гидроксильную группу,A представляет собой CRRили NR,Rпредставляет собой водород, алкил или циклоалкил,Rпредставляет собой водород или алкил,илиA представляет собой азот и вместе со смежной -CHR- образует кольцогде m представляет собой 1, 2 или 3,Rпредставляет собой водород или галоген,их изомеры, а также их аддитивные соли. Лекарственные средства.
EA200400667A 2003-06-13 2004-06-11 Новые соединения бензотиазина и бензотиадиазина, способ их получения и фармацевтические композиции, которые их содержат EA009522B1 (ru)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0307117A FR2856064B1 (fr) 2003-06-13 2003-06-13 Nouveaux derives de benzothiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent.

Publications (3)

Publication Number Publication Date
EA200400667A2 true EA200400667A2 (ru) 2004-12-30
EA200400667A3 EA200400667A3 (ru) 2005-08-25
EA009522B1 EA009522B1 (ru) 2008-02-28

Family

ID=33186481

Family Applications (1)

Application Number Title Priority Date Filing Date
EA200400667A EA009522B1 (ru) 2003-06-13 2004-06-11 Новые соединения бензотиазина и бензотиадиазина, способ их получения и фармацевтические композиции, которые их содержат

Country Status (19)

Country Link
US (1) US7253163B2 (ru)
EP (1) EP1486502A1 (ru)
JP (1) JP2005002113A (ru)
KR (1) KR100645142B1 (ru)
CN (1) CN1274678C (ru)
AR (1) AR044671A1 (ru)
AU (1) AU2004202585A1 (ru)
BR (1) BRPI0401949A (ru)
CA (1) CA2470065A1 (ru)
EA (1) EA009522B1 (ru)
FR (1) FR2856064B1 (ru)
GE (1) GEP20063873B (ru)
HK (1) HK1071751A1 (ru)
MA (1) MA27091A1 (ru)
MX (1) MXPA04005579A (ru)
NO (1) NO20042396L (ru)
NZ (1) NZ533473A (ru)
SG (1) SG139548A1 (ru)
UA (1) UA82183C2 (ru)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2865474B1 (fr) * 2004-01-26 2008-06-13 Servier Lab Nouveaux derives de benzothiazines fluorees, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
FR2879201B1 (fr) * 2004-12-10 2007-02-16 Servier Lab Nouveaux derives de benzothiazine et benzothiadiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
KR100674861B1 (ko) * 2005-08-17 2007-01-29 삼성전기주식회사 무선랜 ａｄ-ｈｏｃ 모드에서의 채널 자동 설정 방법
FR2964969B1 (fr) * 2010-09-16 2012-08-24 Servier Lab Nouveaux derives dihydrobenzoxathiazepines, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
WO2013118845A1 (ja) * 2012-02-08 2013-08-15 武田薬品工業株式会社 複素環化合物およびその用途

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1377693A (fr) * 1962-12-06 1964-11-06 Geigy Ag J R Nouveaux composés dibenzo [1.2] thiaziniques et produits pesticides qui en contiennent
FR2722502B1 (fr) * 1994-07-12 1996-08-23 Adir Nouveau derive de benzothiadiazine, son procede depreparation et les compositions pharmaceutiques qui le contiennent
GB9604926D0 (en) * 1996-03-08 1996-05-08 Sandoz Ltd Organic compounds
RU2214405C2 (ru) * 1998-02-18 2003-10-20 НьюроСёрч А/С Новые соединения и их применение в качестве положительных модуляторов амра-рецепторов
FR2812291B1 (fr) * 2000-07-28 2002-12-13 Adir Nouveaux derives de benzothiadiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
CA2458388A1 (en) * 2001-10-10 2003-04-17 Neurosearch A/S Novel benzothiazine derivatives, their preparation and use
FR2833956B1 (fr) * 2001-12-21 2004-01-30 Servier Lab Nouveaux derives de benzothiazine et de benzothiadiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
FR2833950B1 (fr) * 2001-12-21 2005-12-16 Servier Lab Nouveaux derives de benzothiazine et de benzothiadiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent

Also Published As

Publication number Publication date
GEP20063873B (en) 2006-07-10
CN1572790A (zh) 2005-02-02
EA009522B1 (ru) 2008-02-28
EA200400667A3 (ru) 2005-08-25
CN1274678C (zh) 2006-09-13
BRPI0401949A (pt) 2005-06-07
FR2856064A1 (fr) 2004-12-17
FR2856064B1 (fr) 2005-08-19
KR20040107411A (ko) 2004-12-20
KR100645142B1 (ko) 2006-11-10
HK1071751A1 (en) 2005-07-29
US20040254371A1 (en) 2004-12-16
MXPA04005579A (es) 2005-03-23
JP2005002113A (ja) 2005-01-06
NZ533473A (en) 2005-09-30
NO20042396L (no) 2004-12-14
AU2004202585A1 (en) 2005-01-06
SG139548A1 (en) 2008-02-29
US7253163B2 (en) 2007-08-07
UA82183C2 (ru) 2008-03-25
AR044671A1 (es) 2005-09-21
CA2470065A1 (fr) 2004-12-13
EP1486502A1 (fr) 2004-12-15
MA27091A1 (fr) 2004-12-20

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EA200400666A2 (ru) Новые соединения бензотиазина и бензотиадиазина, способ их получения и фармацевтические композиции, которые их содержат
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Legal Events

Date Code Title Description
MM4A Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s)

Designated state(s): AM AZ BY KZ KG MD TJ TM RU