SG11202001925WA - Substituted imidazoquinolines - Google Patents
Substituted imidazoquinolinesInfo
- Publication number
- SG11202001925WA SG11202001925WA SG11202001925WA SG11202001925WA SG11202001925WA SG 11202001925W A SG11202001925W A SG 11202001925WA SG 11202001925W A SG11202001925W A SG 11202001925WA SG 11202001925W A SG11202001925W A SG 11202001925WA SG 11202001925W A SG11202001925W A SG 11202001925WA
- Authority
- SG
- Singapore
- Prior art keywords
- substituted imidazoquinolines
- imidazoquinolines
- substituted
- Prior art date
Links
- RHKWIGHJGOEUSM-UHFFFAOYSA-N 3h-imidazo[4,5-h]quinoline Chemical class C1=CN=C2C(N=CN3)=C3C=CC2=C1 RHKWIGHJGOEUSM-UHFFFAOYSA-N 0.000 title 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/4738—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems
- A61K31/4745—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems condensed with ring systems having nitrogen as a ring hetero atom, e.g. phenantrolines
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/4738—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
PCT/EP2017/072352 WO2019048036A1 (en) | 2017-09-06 | 2017-09-06 | SUBSTITUTED IMIDAZOQUINOLINES |
PCT/EP2018/073470 WO2019048350A1 (en) | 2017-09-06 | 2018-08-31 | SUBSTITUTED IMIDAZOQUINOLINES |
Publications (1)
Publication Number | Publication Date |
---|---|
SG11202001925WA true SG11202001925WA (en) | 2020-04-29 |
Family
ID=59914433
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SG11202001925WA SG11202001925WA (en) | 2017-09-06 | 2018-08-31 | Substituted imidazoquinolines |
Country Status (14)
Country | Link |
---|---|
US (2) | US11267813B2 (ru) |
EP (1) | EP3679038B1 (ru) |
JP (1) | JP7241738B2 (ru) |
KR (1) | KR20200050963A (ru) |
CN (1) | CN111094287A (ru) |
AU (1) | AU2018327414B2 (ru) |
BR (1) | BR112020004504A2 (ru) |
CA (1) | CA3074166A1 (ru) |
IL (1) | IL273002B2 (ru) |
MX (1) | MX2020002367A (ru) |
RU (1) | RU2768629C2 (ru) |
SG (1) | SG11202001925WA (ru) |
WO (2) | WO2019048036A1 (ru) |
ZA (2) | ZA202001266B (ru) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2019048036A1 (en) * | 2017-09-06 | 2019-03-14 | Biontech Ag | SUBSTITUTED IMIDAZOQUINOLINES |
PT3679025T (pt) * | 2017-09-06 | 2022-06-01 | BioNTech SE | Imidazoquinolinas substituídas como agonistas de tlr7 |
CU24679B1 (es) * | 2019-03-07 | 2023-09-07 | BioNTech SE | Proceso para la preparación de una imidazoquinolina sustituida |
BR112022008039A2 (pt) * | 2019-10-29 | 2022-07-12 | Prime Reach Trading Ltd | Compostos de 4-amino-imidazoquinolina e usos relacionados |
WO2023083439A1 (en) * | 2021-11-09 | 2023-05-19 | BioNTech SE | Tlr7 agonist and combinations for cancer treatment |
Family Cites Families (16)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS585623B2 (ja) | 1976-07-12 | 1983-02-01 | 日本電信電話株式会社 | ファクシミリ通信方式 |
US6451810B1 (en) | 1999-06-10 | 2002-09-17 | 3M Innovative Properties Company | Amide substituted imidazoquinolines |
US6756382B2 (en) | 1999-06-10 | 2004-06-29 | 3M Innovative Properties Company | Amide substituted imidazoquinolines |
US6573273B1 (en) | 1999-06-10 | 2003-06-03 | 3M Innovative Properties Company | Urea substituted imidazoquinolines |
US6677349B1 (en) | 2001-12-21 | 2004-01-13 | 3M Innovative Properties Company | Sulfonamide and sulfamide substituted imidazoquinolines |
AU2003223467B2 (en) | 2002-04-08 | 2007-10-04 | Merck Sharp & Dohme Corp. | Inhibitors of Akt activity |
US8778963B2 (en) | 2003-11-25 | 2014-07-15 | 3M Innovative Properties Company | Hydroxylamine and oxime substituted imidazoquinolines, imidazopyridines, and imidazonaphthyridines |
AU2005283085B2 (en) * | 2004-06-18 | 2012-06-21 | 3M Innovative Properties Company | Substituted imidazoquinolines, imidazopyridines, and imidazonaphthyridines |
WO2007056112A2 (en) * | 2005-11-04 | 2007-05-18 | Coley Pharmaceutical Group, Inc. | Hydroxy and alkoxy substituted 1h-imidazoquinolines and methods |
JP2010519309A (ja) * | 2007-02-20 | 2010-06-03 | ノバルティス アーゲー | 脂質キナーゼおよびmTORのデュアル阻害剤としてのイミダゾキノリン |
DK2155743T3 (da) * | 2007-05-08 | 2012-11-05 | Astrazeneca Ab | Imidazoquinoliner med immunmodulerende egenskaber |
SI2276486T1 (sl) | 2008-03-24 | 2014-01-31 | 4Sc Discovery Gmbh | Novi substituirani imidazokinolini |
EP2419429B1 (en) | 2009-04-16 | 2014-03-26 | Centro Nacional de Investigaciones Oncológicas (CNIO) | Imidazopyrazines as inhibitors of protein kinases |
CN103012398B (zh) | 2011-09-19 | 2015-10-14 | 上海恒瑞医药有限公司 | 咪唑并喹啉类衍生物及其可药用盐、其制备方法及其在医药上的应用 |
PT3679025T (pt) | 2017-09-06 | 2022-06-01 | BioNTech SE | Imidazoquinolinas substituídas como agonistas de tlr7 |
WO2019048036A1 (en) * | 2017-09-06 | 2019-03-14 | Biontech Ag | SUBSTITUTED IMIDAZOQUINOLINES |
-
2017
- 2017-09-06 WO PCT/EP2017/072352 patent/WO2019048036A1/en active Application Filing
-
2018
- 2018-08-31 WO PCT/EP2018/073470 patent/WO2019048350A1/en unknown
- 2018-08-31 MX MX2020002367A patent/MX2020002367A/es unknown
- 2018-08-31 BR BR112020004504-7A patent/BR112020004504A2/pt unknown
- 2018-08-31 EP EP18759137.5A patent/EP3679038B1/en active Active
- 2018-08-31 AU AU2018327414A patent/AU2018327414B2/en active Active
- 2018-08-31 RU RU2020112229A patent/RU2768629C2/ru active
- 2018-08-31 CA CA3074166A patent/CA3074166A1/en active Pending
- 2018-08-31 SG SG11202001925WA patent/SG11202001925WA/en unknown
- 2018-08-31 KR KR1020207006119A patent/KR20200050963A/ko not_active Application Discontinuation
- 2018-08-31 JP JP2020513734A patent/JP7241738B2/ja active Active
- 2018-08-31 CN CN201880057628.1A patent/CN111094287A/zh active Pending
- 2018-08-31 US US16/644,076 patent/US11267813B2/en active Active
-
2020
- 2020-02-27 ZA ZA2020/01266A patent/ZA202001266B/en unknown
- 2020-03-01 IL IL273002A patent/IL273002B2/en unknown
-
2021
- 2021-02-26 ZA ZA2021/01322A patent/ZA202101322B/en unknown
-
2022
- 2022-02-01 US US17/590,550 patent/US20220227756A1/en active Pending
Also Published As
Publication number | Publication date |
---|---|
EP3679038A1 (en) | 2020-07-15 |
KR20200050963A (ko) | 2020-05-12 |
ZA202001266B (en) | 2021-08-25 |
US20220227756A1 (en) | 2022-07-21 |
WO2019048036A1 (en) | 2019-03-14 |
BR112020004504A2 (pt) | 2020-09-15 |
RU2020112229A3 (ru) | 2021-10-06 |
US20200317663A1 (en) | 2020-10-08 |
CN111094287A (zh) | 2020-05-01 |
JP2020532570A (ja) | 2020-11-12 |
WO2019048350A1 (en) | 2019-03-14 |
MX2020002367A (es) | 2020-07-20 |
IL273002B1 (en) | 2023-04-01 |
AU2018327414B2 (en) | 2024-02-15 |
IL273002B2 (en) | 2023-08-01 |
RU2768629C2 (ru) | 2022-03-24 |
JP7241738B2 (ja) | 2023-03-17 |
RU2020112229A (ru) | 2021-10-06 |
US11267813B2 (en) | 2022-03-08 |
EP3679038B1 (en) | 2024-04-03 |
AU2018327414A1 (en) | 2020-03-19 |
CA3074166A1 (en) | 2019-03-14 |
ZA202101322B (en) | 2022-09-28 |
IL273002A (en) | 2020-04-30 |
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