SG11201502893WA - Bruton's tyrosine kinase inhibitors - Google Patents

Bruton's tyrosine kinase inhibitors

Info

Publication number
SG11201502893WA
SG11201502893WA SG11201502893WA SG11201502893WA SG11201502893WA SG 11201502893W A SG11201502893W A SG 11201502893WA SG 11201502893W A SG11201502893W A SG 11201502893WA SG 11201502893W A SG11201502893W A SG 11201502893WA SG 11201502893W A SG11201502893W A SG 11201502893WA
Authority
SG
Singapore
Prior art keywords
bruton
tyrosine kinase
kinase inhibitors
inhibitors
tyrosine
Prior art date
Application number
SG11201502893WA
Other languages
English (en)
Inventor
John Robert Springer
Balekudru Devadas
Danny James Garland
Margaret Lanahan Grapperhaus
Seungil Han
Susan Landis Hockerman
Robert Owen Hughes
Eddine Saiah
Mark Edward Schnute
Shaun Raj Selness
Daniel Patrick Walker
Zhao-Kui Wan
Li Xing
Christoph Wolfgang Zapf
Michelle Ann Schmidt
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=49596360&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SG11201502893W(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer filed Critical Pfizer
Publication of SG11201502893WA publication Critical patent/SG11201502893WA/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
SG11201502893WA 2012-11-02 2013-11-01 Bruton's tyrosine kinase inhibitors SG11201502893WA (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201261721920P 2012-11-02 2012-11-02
US201361772028P 2013-03-04 2013-03-04
PCT/IB2013/059846 WO2014068527A1 (en) 2012-11-02 2013-11-01 Bruton's tyrosine kinase inhibitors

Publications (1)

Publication Number Publication Date
SG11201502893WA true SG11201502893WA (en) 2015-05-28

Family

ID=49596360

Family Applications (1)

Application Number Title Priority Date Filing Date
SG11201502893WA SG11201502893WA (en) 2012-11-02 2013-11-01 Bruton's tyrosine kinase inhibitors

Country Status (27)

Country Link
US (4) US20150291554A1 (ru)
EP (1) EP2914586B1 (ru)
JP (1) JP6178861B2 (ru)
KR (1) KR101668574B1 (ru)
CN (1) CN105008344B (ru)
AP (1) AP2015008381A0 (ru)
AU (1) AU2013340345B2 (ru)
BR (1) BR112015009624A2 (ru)
CA (1) CA2888960C (ru)
CL (1) CL2015001168A1 (ru)
CO (1) CO7350624A2 (ru)
CR (1) CR20150228A (ru)
DO (1) DOP2015000100A (ru)
EA (1) EA201500393A1 (ru)
ES (1) ES2625944T3 (ru)
GE (1) GEP201606597B (ru)
HK (1) HK1211293A1 (ru)
IL (1) IL238571A0 (ru)
MD (1) MD20150035A2 (ru)
MX (1) MX2015005422A (ru)
NI (1) NI201500059A (ru)
PE (1) PE20151070A1 (ru)
PH (1) PH12015500940A1 (ru)
SG (1) SG11201502893WA (ru)
TN (1) TN2015000168A1 (ru)
TW (1) TWI518080B (ru)
WO (1) WO2014068527A1 (ru)

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JP6953445B2 (ja) * 2016-05-16 2021-10-27 スーチョウ、シノベント、ファーマスーティカルズ、カンパニー、リミテッドＳｕｚｈｏｕ Ｓｉｎｏｖｅｎｔ Ｐｈａｒｍａｃｅｕｔｉｃａｌｓ Ｃｏ．， Ｌｔｄ． Ｂｔｋ阻害剤としての５−アミノピラゾールカルボキサミド誘導体およびその製造方法および医薬組成物
KR102391693B1 (ko) 2016-06-29 2022-04-29 프린시피아 바이오파마, 인코퍼레이티드 2-[3-[4-아미노-3-(2-플루오로-4-페녹시-페닐)피라졸로[3,4-d]피리미딘-1-일]피페리딘-1-카르보닐]-4-메틸-4-[4-(옥세탄-3-일)피페라진-1-일]펜트-2-엔니트릴의 변형 방출 제제
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CN108530436B (zh) * 2018-05-17 2020-12-29 黄传满 一种吡唑类化合物及其制备方法和应用
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Also Published As

Publication number Publication date
WO2014068527A1 (en) 2014-05-08
KR20150075114A (ko) 2015-07-02
IL238571A0 (en) 2015-06-30
CO7350624A2 (es) 2015-08-10
US20150291554A1 (en) 2015-10-15
DOP2015000100A (es) 2015-12-31
ES2625944T3 (es) 2017-07-21
EA201500393A1 (ru) 2016-05-31
BR112015009624A2 (pt) 2017-11-14
US10815213B2 (en) 2020-10-27
JP2015535277A (ja) 2015-12-10
AU2013340345A1 (en) 2015-04-30
US20190202798A1 (en) 2019-07-04
TWI518080B (zh) 2016-01-21
CR20150228A (es) 2015-09-14
TN2015000168A1 (fr) 2016-10-03
CN105008344A (zh) 2015-10-28
US20210002251A1 (en) 2021-01-07
EP2914586B1 (en) 2017-04-05
HK1211293A1 (en) 2016-05-20
MX2015005422A (es) 2015-08-05
AU2013340345B2 (en) 2016-10-27
AP2015008381A0 (en) 2015-04-30
EP2914586A1 (en) 2015-09-09
CL2015001168A1 (es) 2015-07-10
JP6178861B2 (ja) 2017-08-09
PE20151070A1 (es) 2015-08-01
PH12015500940A1 (en) 2015-06-29
GEP201606597B (en) 2017-01-10
US20170283393A1 (en) 2017-10-05
US10266513B2 (en) 2019-04-23
TW201431851A (zh) 2014-08-16
MD20150035A2 (ru) 2015-10-31
KR101668574B1 (ko) 2016-10-24
NI201500059A (es) 2015-06-05
CN105008344B (zh) 2017-07-25
CA2888960A1 (en) 2014-05-08
CA2888960C (en) 2017-08-15

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