SG10202000590SA - Antimitotic amides for the treatment of cancer and proliferative disorders - Google Patents

Antimitotic amides for the treatment of cancer and proliferative disorders

Info

Publication number
SG10202000590SA
SG10202000590SA SG10202000590SA SG10202000590SA SG10202000590SA SG 10202000590S A SG10202000590S A SG 10202000590SA SG 10202000590S A SG10202000590S A SG 10202000590SA SG 10202000590S A SG10202000590S A SG 10202000590SA SG 10202000590S A SG10202000590S A SG 10202000590SA
Authority
SG
Singapore
Prior art keywords
antimitotic
amides
cancer
treatment
proliferative disorders
Prior art date
Application number
SG10202000590SA
Other languages
English (en)
Inventor
Adam Siddiqui-Jain
Original Assignee
Frost Biologic Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Frost Biologic Inc filed Critical Frost Biologic Inc
Publication of SG10202000590SA publication Critical patent/SG10202000590SA/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
    • A61K31/41781,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4409Non condensed pyridines; Hydrogenated derivatives thereof only substituted in position 4, e.g. isoniazid, iproniazid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/444Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/14Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2121/00Preparations for use in therapy

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
SG10202000590SA 2014-02-21 2015-02-20 Antimitotic amides for the treatment of cancer and proliferative disorders SG10202000590SA (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201461942956P 2014-02-21 2014-02-21

Publications (1)

Publication Number Publication Date
SG10202000590SA true SG10202000590SA (en) 2020-03-30

Family

ID=52684675

Family Applications (2)

Application Number Title Priority Date Filing Date
SG10202000590SA SG10202000590SA (en) 2014-02-21 2015-02-20 Antimitotic amides for the treatment of cancer and proliferative disorders
SG11201606869TA SG11201606869TA (en) 2014-02-21 2015-02-20 Antimitotic amides for the treatment of cancer and proliferative disorders

Family Applications After (1)

Application Number Title Priority Date Filing Date
SG11201606869TA SG11201606869TA (en) 2014-02-21 2015-02-20 Antimitotic amides for the treatment of cancer and proliferative disorders

Country Status (15)

Country Link
US (5) US10016398B2 (enExample)
EP (1) EP3107909B1 (enExample)
JP (1) JP6506313B2 (enExample)
KR (1) KR102420508B1 (enExample)
CN (2) CN114634483B (enExample)
AU (1) AU2015218775C1 (enExample)
BR (1) BR112016019161B1 (enExample)
CA (1) CA2940237C (enExample)
ES (1) ES2893374T3 (enExample)
IL (1) IL247293B (enExample)
MX (1) MX390530B (enExample)
RU (1) RU2713179C2 (enExample)
SG (2) SG10202000590SA (enExample)
WO (1) WO2015127284A2 (enExample)
ZA (1) ZA201606471B (enExample)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6420622B1 (en) 1997-08-01 2002-07-16 3M Innovative Properties Company Medical article having fluid control film
WO2015127284A2 (en) * 2014-02-21 2015-08-27 Frost Biologic, Inc. Antimitotic amides for the treatment of cancer and proliferative disorders
CN106727583A (zh) * 2016-12-12 2017-05-31 范旭升 一种治疗舒张性心衰的药物组合物
US11377436B2 (en) * 2017-07-12 2022-07-05 The Brigham And Women's Hospital, Inc. EAAT2 enhancing molecules
US11760701B2 (en) 2018-02-27 2023-09-19 The Research Foundation For The State University Of New Yrok Difluoromethoxylation and trifluoromethoxylation compositions and methods for synthesizing same
KR20250173438A (ko) * 2024-05-30 2025-12-10 삼진제약주식회사 Nr2f6 억제제 및 이의 용도

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* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0001930D0 (en) * 2000-01-27 2000-03-22 Novartis Ag Organic compounds
JP2003535860A (ja) * 2000-06-05 2003-12-02 ドン・ア・ファーム・カンパニー・リミテッド 新規なオキサゾリジノン誘導体及びその製造方法
US6995162B2 (en) * 2001-01-12 2006-02-07 Amgen Inc. Substituted alkylamine derivatives and methods of use
GB0209715D0 (en) * 2002-04-27 2002-06-05 Astrazeneca Ab Chemical compounds
EP1763348A1 (en) * 2004-06-30 2007-03-21 Novartis AG Method for increasing the susceptibility of peptide deformylase inhibitors by using efflux pump inhibitors
JPWO2007018319A1 (ja) * 2005-08-11 2009-02-19 武田薬品工業株式会社 ピリジルフェノール化合物およびその用途
JP5430944B2 (ja) * 2006-01-31 2014-03-05 シンタ ファーマシューティカルズ コーポレーション 炎症および免疫関連用途のためのピリジルフェニル化合物
WO2008059042A1 (en) 2006-11-17 2008-05-22 Smithkline Beecham Corporation 2-carboxy thiophene derivatives as anti viral agents
CA2683624A1 (en) * 2007-04-12 2008-10-23 F. Hoffmann-La Roche Ag Pharmaceutical compounds
US20110118281A9 (en) * 2008-10-01 2011-05-19 Gary Bohnert Compounds for inflammation and immune-related uses
WO2010100475A1 (en) * 2009-03-02 2010-09-10 Astrazeneca Ab Hydroxamic acid derivatives as gram-negative antibacterial agents
NZ598758A (en) * 2009-09-11 2013-12-20 Amgen Inc N-4 (-((3-(2-amino-4 pyrimidinyl)-2-pyridinyl)oxy)phenyl)-4-(4-methyl-2-thienyl)-1-phthalazinamine for use in the treatment of antimitotic agent resistant cancer
WO2011139489A2 (en) 2010-04-27 2011-11-10 Calcimedica Inc. Compounds that modulate intracellular calcium
US20130063385A1 (en) * 2010-05-14 2013-03-14 Sharp Kabushiki Kaisha Portable information terminal and method for controlling same
TWI541243B (zh) * 2010-09-10 2016-07-11 拜耳知識產權公司 經取代咪唑并嗒
CN103380117A (zh) * 2011-01-21 2013-10-30 Abbvie公司 激酶的吡啶酰胺抑制剂
CN103402985A (zh) * 2011-02-10 2013-11-20 先正达参股股份有限公司 杀微生物的吡唑衍生物
CN103702665B (zh) * 2011-05-03 2016-08-17 幸讬制药公司 用于炎症和免疫相关用途的化合物
WO2013063385A1 (en) * 2011-10-28 2013-05-02 Synta Pharmaceuticals Corp. Compounds for inflammation and immune-related uses
WO2015127284A2 (en) * 2014-02-21 2015-08-27 Frost Biologic, Inc. Antimitotic amides for the treatment of cancer and proliferative disorders

Also Published As

Publication number Publication date
JP2017506267A (ja) 2017-03-02
RU2713179C2 (ru) 2020-02-04
WO2015127284A2 (en) 2015-08-27
US10016398B2 (en) 2018-07-10
US20170172984A1 (en) 2017-06-22
EP3107909B1 (en) 2021-07-14
MX2016010877A (es) 2017-05-04
US10772872B2 (en) 2020-09-15
CA2940237A1 (en) 2015-08-27
ZA201606471B (en) 2025-06-25
WO2015127284A3 (en) 2015-10-15
US20260034101A1 (en) 2026-02-05
US12383533B2 (en) 2025-08-12
IL247293B (en) 2021-01-31
IL247293A0 (en) 2016-09-29
US11129813B2 (en) 2021-09-28
BR112016019161A2 (enExample) 2017-08-15
AU2015218775B2 (en) 2019-06-20
KR102420508B1 (ko) 2022-07-13
RU2016135555A3 (enExample) 2018-10-05
MX390530B (es) 2025-03-20
RU2016135555A (ru) 2018-03-28
CN114634483A (zh) 2022-06-17
JP6506313B2 (ja) 2019-04-24
US20200397758A1 (en) 2020-12-24
CN106068263A (zh) 2016-11-02
SG11201606869TA (en) 2016-09-29
US20220008395A1 (en) 2022-01-13
US20180325871A1 (en) 2018-11-15
ES2893374T3 (es) 2022-02-08
KR20160116009A (ko) 2016-10-06
CA2940237C (en) 2023-03-07
AU2015218775A1 (en) 2016-08-25
CN114634483B (zh) 2024-08-13
BR112016019161B1 (pt) 2022-12-20
EP3107909A2 (en) 2016-12-28
AU2015218775C1 (en) 2020-01-16

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