SE9301057L - Beredning med kontrollerad frisättning - Google Patents

Beredning med kontrollerad frisättning

Info

Publication number
SE9301057L
SE9301057L SE9301057A SE9301057A SE9301057L SE 9301057 L SE9301057 L SE 9301057L SE 9301057 A SE9301057 A SE 9301057A SE 9301057 A SE9301057 A SE 9301057A SE 9301057 L SE9301057 L SE 9301057L
Authority
SE
Sweden
Prior art keywords
morphine
controlled release
preparations
manufacture
serum concentration
Prior art date
Application number
SE9301057A
Other languages
English (en)
Swedish (sv)
Other versions
SE9301057D0 (sv
Inventor
Birgitta Olsson
Maritta Anneli Pesonen
Gert Ragnarsson
Original Assignee
Pharmacia Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=20389415&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SE9301057(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pharmacia Ab filed Critical Pharmacia Ab
Priority to SE9301057A priority Critical patent/SE9301057L/xx
Publication of SE9301057D0 publication Critical patent/SE9301057D0/xx
Priority to US08/213,518 priority patent/US5614218A/en
Priority to EP94912116A priority patent/EP0642335B2/en
Priority to CZ942986A priority patent/CZ284924B6/cs
Priority to DE69423028T priority patent/DE69423028T3/de
Priority to CN94190160A priority patent/CN1104891C/zh
Priority to DK94912116T priority patent/DK0642335T4/da
Priority to RU94046147A priority patent/RU2136283C1/ru
Priority to PCT/SE1994/000264 priority patent/WO1994022431A1/en
Priority to KR1019940704397A priority patent/KR100316206B1/ko
Priority to AT94912116T priority patent/ATE189771T1/de
Priority to SK1437-94A priority patent/SK280362B6/sk
Priority to AU64393/94A priority patent/AU680891C/en
Priority to ES94912116T priority patent/ES2144516T5/es
Priority to PT94912116T priority patent/PT642335E/pt
Priority to HU9403437A priority patent/HU227344B1/hu
Priority to PL94306421A priority patent/PL175326B1/pl
Priority to JP52197694A priority patent/JP4107678B2/ja
Priority to CA002135639A priority patent/CA2135639C/en
Priority to NZ263632A priority patent/NZ263632A/en
Publication of SE9301057L publication Critical patent/SE9301057L/xx
Priority to EE9400376A priority patent/EE03147B1/xx
Priority to NO944565A priority patent/NO310015B1/no
Priority to FI945621A priority patent/FI113743B/fi
Priority to LVP-94-228A priority patent/LV10684B/xx
Priority to US08/844,556 priority patent/US5952005A/en
Priority to GR20000401009T priority patent/GR3033325T3/el

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005Wall or coating material
    • A61K9/5021Organic macromolecular compounds
    • A61K9/5036Polysaccharides, e.g. gums, alginate; Cyclodextrin
    • A61K9/5042Cellulose; Cellulose derivatives, e.g. phthalate or acetate succinate esters of hydroxypropyl methylcellulose
    • A61K9/5047Cellulose ethers containing no ester groups, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/485Morphinan derivatives, e.g. morphine, codeine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Emergency Medicine (AREA)
  • Neurosurgery (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Iron Core Of Rotating Electric Machines (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
SE9301057A 1993-03-30 1993-03-30 Beredning med kontrollerad frisättning SE9301057L (sv)

Priority Applications (26)

Application Number Priority Date Filing Date Title
SE9301057A SE9301057L (sv) 1993-03-30 1993-03-30 Beredning med kontrollerad frisättning
US08/213,518 US5614218A (en) 1993-03-30 1994-03-16 Controlled release preparation
CA002135639A CA2135639C (en) 1993-03-30 1994-03-24 Controlled release preparation containing a salt of morphine
NZ263632A NZ263632A (en) 1993-03-30 1994-03-24 Oral sustained release morphine composition having a barrier coating comprising at least one water insoluble compound
SK1437-94A SK280362B6 (sk) 1993-03-30 1994-03-24 Orálny farmaceutický prostriedok obsahujúci terape
HU9403437A HU227344B1 (en) 1993-03-30 1994-03-24 Oral pharmaceutical preparation containing a salt of morphine and process for producing them
DE69423028T DE69423028T3 (de) 1993-03-30 1994-03-24 Zubereitung mit kontrollierter freisetzung, die ein morphinsalz enthält
CN94190160A CN1104891C (zh) 1993-03-30 1994-03-24 缓释制剂
DK94912116T DK0642335T4 (da) 1993-03-30 1994-03-24 Morphinsaltholdigt præparat med styret frigivelse
RU94046147A RU2136283C1 (ru) 1993-03-30 1994-03-24 Препарат с контролируемым высвобождением лекарства и способ его получения, способ лечения
PCT/SE1994/000264 WO1994022431A1 (en) 1993-03-30 1994-03-24 Controlled release preparation containing a salt of morphine
KR1019940704397A KR100316206B1 (ko) 1993-03-30 1994-03-24 모르핀의염을함유하는방출조절식제제
AT94912116T ATE189771T1 (de) 1993-03-30 1994-03-24 Zubereitung mit kontrollierter freisetzung, die ein morphinsalz enthält
EP94912116A EP0642335B2 (en) 1993-03-30 1994-03-24 Controlled release preparation containing a salt of morphine
AU64393/94A AU680891C (en) 1993-03-30 1994-03-24 Controlled release preparation containing a salt of morphine
ES94912116T ES2144516T5 (es) 1993-03-30 1994-03-24 Preparacion con liberacion controlada que contiene una sal de morfina.
PT94912116T PT642335E (pt) 1993-03-30 1994-03-24 Preparacao de um sal de morfina de libertacao controlada
CZ942986A CZ284924B6 (cs) 1993-03-30 1994-03-24 Prostředek s řízeným uvolňováním, který obsahuje morfinovou sůl
PL94306421A PL175326B1 (pl) 1993-03-30 1994-03-24 Preparat doustny wielojednostkowy o kontrolowanym uwalnianiu zawierający morfinę i sposób wytwarzania preparatu doustnego wielojednostkowego o kontrolowanym uwalnianiu zawierającego morfinę
JP52197694A JP4107678B2 (ja) 1993-03-30 1994-03-24 制御放出製剤
EE9400376A EE03147B1 (et) 1993-03-30 1994-11-16 Kontrollitud vabanemisega preparaat ja selle valmistamismeetodid
FI945621A FI113743B (fi) 1993-03-30 1994-11-29 Menetelmä säädetysti vapauttavan valmisteen valmistamiseksi
NO944565A NO310015B1 (no) 1993-03-30 1994-11-29 Preparat med regulert frigjörelse som inneholder et morfinsalt, fremgangsmåte for fremstilling derav, samt anvendelse av preparatet for fremstilling av et medikament
LVP-94-228A LV10684B (en) 1993-03-30 1994-11-30 Controlled release preparation containing a salt of morphine
US08/844,556 US5952005A (en) 1993-03-30 1997-04-21 Controlled release preparation for administering morphine
GR20000401009T GR3033325T3 (en) 1993-03-30 2000-04-26 Controlled release preparation containing a salt of morphine.

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
SE9301057A SE9301057L (sv) 1993-03-30 1993-03-30 Beredning med kontrollerad frisättning

Publications (2)

Publication Number Publication Date
SE9301057D0 SE9301057D0 (sv) 1993-03-30
SE9301057L true SE9301057L (sv) 1994-10-01

Family

ID=20389415

Family Applications (1)

Application Number Title Priority Date Filing Date
SE9301057A SE9301057L (sv) 1993-03-30 1993-03-30 Beredning med kontrollerad frisättning

Country Status (25)

Country Link
US (1) US5614218A (fi)
EP (1) EP0642335B2 (fi)
JP (1) JP4107678B2 (fi)
KR (1) KR100316206B1 (fi)
CN (1) CN1104891C (fi)
AT (1) ATE189771T1 (fi)
AU (1) AU680891C (fi)
CA (1) CA2135639C (fi)
CZ (1) CZ284924B6 (fi)
DE (1) DE69423028T3 (fi)
DK (1) DK0642335T4 (fi)
EE (1) EE03147B1 (fi)
ES (1) ES2144516T5 (fi)
FI (1) FI113743B (fi)
GR (1) GR3033325T3 (fi)
HU (1) HU227344B1 (fi)
LV (1) LV10684B (fi)
NO (1) NO310015B1 (fi)
NZ (1) NZ263632A (fi)
PL (1) PL175326B1 (fi)
PT (1) PT642335E (fi)
RU (1) RU2136283C1 (fi)
SE (1) SE9301057L (fi)
SK (1) SK280362B6 (fi)
WO (1) WO1994022431A1 (fi)

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US5266331A (en) * 1991-11-27 1993-11-30 Euroceltique, S.A. Controlled release oxycodone compositions
US5958459A (en) * 1991-12-24 1999-09-28 Purdue Pharma L.P. Opioid formulations having extended controlled released
US5968551A (en) 1991-12-24 1999-10-19 Purdue Pharma L.P. Orally administrable opioid formulations having extended duration of effect
AU735113C (en) * 1991-12-24 2007-06-14 Mundipharma Medical Gmbh Opioid formulations for treating pain
US5478577A (en) * 1993-11-23 1995-12-26 Euroceltique, S.A. Method of treating pain by administering 24 hour oral opioid formulations exhibiting rapid rate of initial rise of plasma drug level
US5472712A (en) * 1991-12-24 1995-12-05 Euroceltique, S.A. Controlled-release formulations coated with aqueous dispersions of ethylcellulose
US20080075781A1 (en) * 1992-11-25 2008-03-27 Purdue Pharma Lp Controlled release oxycodone compositions
IL109460A (en) * 1993-05-10 1998-03-10 Euro Celtique Sa Controlled release formulation comprising tramadol
US20070275062A1 (en) * 1993-06-18 2007-11-29 Benjamin Oshlack Controlled release oxycodone compositions
IL110014A (en) * 1993-07-01 1999-11-30 Euro Celtique Sa Solid controlled-release oral dosage forms of opioid analgesics
US7740881B1 (en) 1993-07-01 2010-06-22 Purdue Pharma Lp Method of treating humans with opioid formulations having extended controlled release
IL109944A (en) 1993-07-01 1998-12-06 Euro Celtique Sa Continuous release dosage form containing morphine and a method of preparing such sustained release unit dosage forms
US5879705A (en) * 1993-07-27 1999-03-09 Euro-Celtique S.A. Sustained release compositions of morphine and a method of preparing pharmaceutical compositions
US5891471A (en) * 1993-11-23 1999-04-06 Euro-Celtique, S.A. Pharmaceutical multiparticulates
US20020006438A1 (en) * 1998-09-25 2002-01-17 Benjamin Oshlack Sustained release hydromorphone formulations exhibiting bimodal characteristics
GB9519363D0 (en) 1995-09-22 1995-11-22 Euro Celtique Sa Pharmaceutical formulation
DE19607395C2 (de) * 1996-02-28 2002-11-21 Lohmann Therapie Syst Lts Salze aus einem kationischen narkotischen Analgetikum mit einem anionischen nichtnarkotischen Analgetikum, Verfahren zu deren Herstellung und die diese Salze enthaltenden pharmazeutischen Präparate
US6245351B1 (en) 1996-03-07 2001-06-12 Takeda Chemical Industries, Ltd. Controlled-release composition
US5891474A (en) 1997-01-29 1999-04-06 Poli Industria Chimica, S.P.A. Time-specific controlled release dosage formulations and method of preparing same
US6066339A (en) * 1997-10-17 2000-05-23 Elan Corporation, Plc Oral morphine multiparticulate formulation
US6806294B2 (en) 1998-10-15 2004-10-19 Euro-Celtique S.A. Opioid analgesic
FR2794646B1 (fr) 1999-06-09 2001-09-21 Ethypharm Lab Prod Ethiques Microgranules de sulfate de morphine, procede de preparation et composition les contenant
EP2295043A1 (en) * 1999-10-29 2011-03-16 Euro-Celtique S.A. Controlled release hydrocodone formulations
US10179130B2 (en) 1999-10-29 2019-01-15 Purdue Pharma L.P. Controlled release hydrocodone formulations
EP2932964A1 (en) 2000-10-30 2015-10-21 Euro-Celtique S.A. Controlled release hydrocodone formulations
UA81224C2 (uk) * 2001-05-02 2007-12-25 Euro Celtic S A Дозована форма оксикодону та її застосування
US20110104214A1 (en) 2004-04-15 2011-05-05 Purdue Pharma L.P. Once-a-day oxycodone formulations
US20030070584A1 (en) * 2001-05-15 2003-04-17 Cynthia Gulian Dip coating compositions containing cellulose ethers
AU4061702A (en) * 2001-05-15 2003-04-03 Mcneil-Ppc, Inc. Dip coating compositions containing starch or dextrin
US20030072731A1 (en) * 2001-05-15 2003-04-17 Cynthia Gulian Dip coating compositions containing starch or dextrin
WO2003024429A1 (en) 2001-09-21 2003-03-27 Egalet A/S Polymer release system
US20040253310A1 (en) 2001-09-21 2004-12-16 Gina Fischer Morphine polymer release system
US8309118B2 (en) * 2001-09-28 2012-11-13 Mcneil-Ppc, Inc. Film forming compositions containing sucralose
CA2479350A1 (en) * 2002-03-15 2003-09-25 Cypress Bioscience, Inc. Ne and 5-ht reuptake inhibitors for treating visceral pain syndromes
US7429619B2 (en) * 2002-08-02 2008-09-30 Mcneil Consumer Healthcare Polyacrylic film forming compositions
CA2498798A1 (en) * 2002-09-20 2004-04-01 Alpharma, Inc. Sustained-release opioid formulations and methods of use
CA2499550C (en) * 2002-09-20 2013-10-15 Alpharma, Inc. Sequestering subunit and related compositions and methods
US20040138200A1 (en) * 2002-10-04 2004-07-15 Michael Hawley Pharmaceutical compositions for treatment of Parkinson's disease
US20060003004A1 (en) * 2002-10-25 2006-01-05 Collegium Pharmaceutical, Inc. Pulsatile release compositions of milnacipran
US20040132826A1 (en) * 2002-10-25 2004-07-08 Collegium Pharmaceutical, Inc. Modified release compositions of milnacipran
US20040228830A1 (en) * 2003-01-28 2004-11-18 Collegium Pharmaceutical, Inc. Multiparticulate compositions of milnacipran for oral administration
ATE495732T1 (de) 2003-03-26 2011-02-15 Egalet As Morphin-system mit kontrollierter freisetzung
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CA2524300C (en) * 2003-08-08 2008-10-28 Biovail Laboratories International Srl Modified-release tablet of bupropion hydrochloride
EP1810678A1 (de) 2006-01-19 2007-07-25 Holger Lars Hermann Verwendung einer Kombination von Morphin und Naloxon zur Drogensubstitution
US20070190141A1 (en) * 2006-02-16 2007-08-16 Aaron Dely Extended release opiate composition
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WO2009023672A2 (en) 2007-08-13 2009-02-19 Abuse Deterrent Pharmaceutical Llc Abuse resistant drugs, method of use and method of making
GB2462022B (en) * 2008-06-16 2011-05-25 Biovascular Inc Controlled release compositions of agents that reduce circulating levels of platelets and methods thereof
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US9707184B2 (en) 2014-07-17 2017-07-18 Pharmaceutical Manufacturing Research Services, Inc. Immediate release abuse deterrent liquid fill dosage form
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US5478577A (en) 1993-11-23 1995-12-26 Euroceltique, S.A. Method of treating pain by administering 24 hour oral opioid formulations exhibiting rapid rate of initial rise of plasma drug level
US5273760A (en) 1991-12-24 1993-12-28 Euroceltigue, S.A. Stabilized controlled release substrate having a coating derived from an aqueous dispersion of hydrophobic polymer
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Also Published As

Publication number Publication date
PL175326B1 (pl) 1998-12-31
DE69423028T2 (de) 2001-01-18
KR100316206B1 (ko) 2002-11-09
PT642335E (pt) 2000-08-31
CZ298694A3 (en) 1995-05-17
FI945621A (fi) 1994-11-29
EP0642335A1 (en) 1995-03-15
NZ263632A (en) 1997-06-24
AU6439394A (en) 1994-10-24
CA2135639A1 (en) 1994-10-13
ES2144516T5 (es) 2005-07-01
NO944565D0 (no) 1994-11-29
EP0642335B2 (en) 2005-01-19
SK143794A3 (en) 1995-06-07
CN1104891C (zh) 2003-04-09
HU227344B1 (en) 2011-04-28
US5614218A (en) 1997-03-25
LV10684B (en) 1996-02-20
SE9301057D0 (sv) 1993-03-30
DK0642335T3 (da) 2000-07-24
NO944565L (no) 1994-11-29
ATE189771T1 (de) 2000-03-15
CN1106608A (zh) 1995-08-09
PL306421A1 (en) 1995-04-03
AU680891B2 (en) 1997-08-14
ES2144516T3 (es) 2000-06-16
LV10684A (lv) 1995-06-20
JP4107678B2 (ja) 2008-06-25
CZ284924B6 (cs) 1999-04-14
SK280362B6 (sk) 1999-12-10
DE69423028T3 (de) 2006-07-20
DK0642335T4 (da) 2005-05-23
JPH08501319A (ja) 1996-02-13
RU2136283C1 (ru) 1999-09-10
RU94046147A (ru) 1996-11-10
AU680891C (en) 2002-01-03
FI945621A0 (fi) 1994-11-29
CA2135639C (en) 2006-02-07
NO310015B1 (no) 2001-05-07
FI113743B (fi) 2004-06-15
HUT71417A (en) 1995-11-28
EP0642335B1 (en) 2000-02-16
HU9403437D0 (en) 1995-02-28
DE69423028D1 (de) 2000-03-23
EE03147B1 (et) 1999-02-15
WO1994022431A1 (en) 1994-10-13
GR3033325T3 (en) 2000-09-29

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