SE9103776D0 - NEW COMPOUNDS - Google Patents

NEW COMPOUNDS

Info

Publication number
SE9103776D0
SE9103776D0 SE9103776A SE9103776A SE9103776D0 SE 9103776 D0 SE9103776 D0 SE 9103776D0 SE 9103776 A SE9103776 A SE 9103776A SE 9103776 A SE9103776 A SE 9103776A SE 9103776 D0 SE9103776 D0 SE 9103776D0
Authority
SE
Sweden
Prior art keywords
compounds
new compounds
methyl
och3
medicine
Prior art date
Application number
SE9103776A
Other languages
Swedish (sv)
Inventor
B Holstein
Original Assignee
Astra Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astra Ab filed Critical Astra Ab
Priority to SE9103776A priority Critical patent/SE9103776D0/en
Publication of SE9103776D0 publication Critical patent/SE9103776D0/en
Priority to IS4079A priority patent/IS4079A/en
Priority to TW081109053A priority patent/TW224100B/zh
Priority to ZA928836A priority patent/ZA928836B/en
Priority to YU101692A priority patent/YU101692A/en
Priority to HR921400A priority patent/HRP921400A2/en
Priority to EP93900477A priority patent/EP0628049A1/en
Priority to AU31752/93A priority patent/AU665043B2/en
Priority to KR1019940702131A priority patent/KR940703840A/en
Priority to SK735-94A priority patent/SK73594A3/en
Priority to HU9401840A priority patent/HUT68270A/en
Priority to CZ941467A priority patent/CZ146794A3/en
Priority to JP5510832A priority patent/JPH07502503A/en
Priority to CA002124689A priority patent/CA2124689A1/en
Priority to PCT/SE1992/000844 priority patent/WO1993012124A1/en
Priority to NZ246220A priority patent/NZ246220A/en
Priority to IL104025A priority patent/IL104025A0/en
Priority to APAP/P/1992/000463A priority patent/AP397A/en
Priority to MX9207269A priority patent/MX9207269A/en
Priority to MA23036A priority patent/MA22746A1/en
Priority to TNTNSN92115A priority patent/TNSN92115A1/en
Priority to CN92114364A priority patent/CN1031827C/en
Priority to IS3960A priority patent/IS3960A/en
Priority to SI19929200402A priority patent/SI9200402A/en
Priority to NO942230A priority patent/NO942230D0/en
Priority to FI942912A priority patent/FI942912A0/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6558—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/66—Phosphorus compounds
    • A61K31/675—Phosphorus compounds having nitrogen as a ring hetero atom, e.g. pyridoxal phosphate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6558—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system
    • C07F9/65583—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system each of the hetero rings containing nitrogen as ring hetero atom

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Molecular Biology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

The novel compounds of formula (I), wherein R<1> and R<2>, which are different, are each methyl, -C(O)-CH3 or -C(O)-OCH3 and whereby one of R<1> or R<2> is always methyl; and M is a physiologically acceptable counter cation, as well as processes for the preparation of said compounds, pharmaceutical compositions containing said compounds as active ingredient, and the use of the compounds in medicine.
SE9103776A 1991-12-19 1991-12-19 NEW COMPOUNDS SE9103776D0 (en)

Priority Applications (26)

Application Number Priority Date Filing Date Title
SE9103776A SE9103776D0 (en) 1991-12-19 1991-12-19 NEW COMPOUNDS
IS4079A IS4079A (en) 1991-12-19 1992-10-06 Intermediates for the production of substituted benzimidazoles
TW081109053A TW224100B (en) 1991-12-19 1992-11-11
ZA928836A ZA928836B (en) 1991-12-19 1992-11-16 Substituted benzimidazoles, process for their preparation as well as their use.
YU101692A YU101692A (en) 1991-12-19 1992-11-25 SUBSTITUTED BENZIMIDAZOLES AND THE PROCEDURE FOR THEIR MANAGEMENT
HR921400A HRP921400A2 (en) 1991-12-19 1992-12-07 Substituted benzimidazoles, process for their preparation as well as their use
IL104025A IL104025A0 (en) 1991-12-19 1992-12-08 Substituted benzimidazoles,process for their preparation as well as their use
JP5510832A JPH07502503A (en) 1991-12-19 1992-12-08 Substituted benzimidazoles, their production methods and their uses
NZ246220A NZ246220A (en) 1991-12-19 1992-12-08 Substituted benzimidazol-1-yl methyl esters of phosphoric acid, medicaments and precursors
KR1019940702131A KR940703840A (en) 1991-12-19 1992-12-08 Substituted benzimidazoles, preparation methods and uses thereof (SUBSTITUTED BENZIMIDAZOLES, PROCESS FOR THEIR PREPARATION AS WELL AS THEIR USE)
SK735-94A SK73594A3 (en) 1991-12-19 1992-12-08 Substituted benzimidazoles, process for their production as well as their use
HU9401840A HUT68270A (en) 1991-12-19 1992-12-08 Substituted benzimidazoles, process for their preparation as well as their use
CZ941467A CZ146794A3 (en) 1991-12-19 1992-12-08 Substituted benzimidazoles, process of their preparation and their use
EP93900477A EP0628049A1 (en) 1991-12-19 1992-12-08 Substituted benzimidazoles, process for their preparation as well as their use
CA002124689A CA2124689A1 (en) 1991-12-19 1992-12-08 Substituted benzimidazoles, process for their preparation as well as their use
PCT/SE1992/000844 WO1993012124A1 (en) 1991-12-19 1992-12-08 Substituted benzimidazoles, process for their preparation as well as their use
AU31752/93A AU665043B2 (en) 1991-12-19 1992-12-08 Substituted benzimidazoles, process for their preparation as well as their use
APAP/P/1992/000463A AP397A (en) 1991-12-19 1992-12-14 Substituted benzimidazoles, process for their preparation as well as their use.
MX9207269A MX9207269A (en) 1991-12-19 1992-12-15 SUBSTITUTED BENZMIDAZOLES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM.
MA23036A MA22746A1 (en) 1991-12-19 1992-12-16 SUBSTITUTES OF BENZIMIDAZOLES, PROCESS FOR THEIR PREPARATION AND THEIR USE
TNTNSN92115A TNSN92115A1 (en) 1991-12-19 1992-12-18 BENZIMIDAZOLES SUBSTITUTES, PROCESS FOR THEIR PREPARATION AND THEIR USE
CN92114364A CN1031827C (en) 1991-12-19 1992-12-18 Substituted benzimidazoles, process for their preparation as well as their use
IS3960A IS3960A (en) 1991-12-19 1992-12-18 Method of producing substituted benzimidazole sols
SI19929200402A SI9200402A (en) 1991-12-19 1992-12-18 Substituted benzimidazoles, process for their preparation and their use
NO942230A NO942230D0 (en) 1991-12-19 1994-06-14 Substituted benzimidazoles, processes for their preparation and their use
FI942912A FI942912A0 (en) 1991-12-19 1994-06-17 Substituted benzimidazoles, a process for their preparation and their use

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
SE9103776A SE9103776D0 (en) 1991-12-19 1991-12-19 NEW COMPOUNDS

Publications (1)

Publication Number Publication Date
SE9103776D0 true SE9103776D0 (en) 1991-12-19

Family

ID=20384667

Family Applications (1)

Application Number Title Priority Date Filing Date
SE9103776A SE9103776D0 (en) 1991-12-19 1991-12-19 NEW COMPOUNDS

Country Status (25)

Country Link
EP (1) EP0628049A1 (en)
JP (1) JPH07502503A (en)
KR (1) KR940703840A (en)
CN (1) CN1031827C (en)
AP (1) AP397A (en)
AU (1) AU665043B2 (en)
CA (1) CA2124689A1 (en)
CZ (1) CZ146794A3 (en)
FI (1) FI942912A0 (en)
HR (1) HRP921400A2 (en)
HU (1) HUT68270A (en)
IL (1) IL104025A0 (en)
IS (2) IS4079A (en)
MA (1) MA22746A1 (en)
MX (1) MX9207269A (en)
NO (1) NO942230D0 (en)
NZ (1) NZ246220A (en)
SE (1) SE9103776D0 (en)
SI (1) SI9200402A (en)
SK (1) SK73594A3 (en)
TN (1) TNSN92115A1 (en)
TW (1) TW224100B (en)
WO (1) WO1993012124A1 (en)
YU (1) YU101692A (en)
ZA (1) ZA928836B (en)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19645974C1 (en) * 1996-11-07 1998-08-13 Andreas Johannes Kesel (Z) -5 - [[3-Hydroxy-2-methyl-5 - [(phosphonooxy) methyl] -4-pyridinyl] methylene] -2-thioxo-4-thiazolidinone, process for its preparation and use
US5985856A (en) * 1997-12-31 1999-11-16 University Of Kansas Water soluble prodrugs of secondary and tertiary amine containing drugs and methods of making thereof
PL1913009T3 (en) 2005-07-28 2010-10-29 Intervet Int Bv Novel benzimidazole (thio) carbamates with antiparasitic activity and the synthesis thereof
TWI385169B (en) 2005-10-31 2013-02-11 Eisai R&D Man Co Ltd Heterocyclic substituted pyridine derivatives and antifungal agent containing same
EP2037914B1 (en) 2006-06-14 2013-10-23 Intervet International BV A suspension comprising benzimidazole carbamate and a polysorbate
TW200841879A (en) 2007-04-27 2008-11-01 Eisai R&D Man Co Ltd Pyridine derivatives substituted by heterocyclic ring and phosphonoamino group, and anti-fungal agent containing same
US8513287B2 (en) * 2007-12-27 2013-08-20 Eisai R&D Management Co., Ltd. Heterocyclic ring and phosphonoxymethyl group substituted pyridine derivatives and antifungal agent containing same
US8188119B2 (en) 2008-10-24 2012-05-29 Eisai R&D Management Co., Ltd Pyridine derivatives substituted with heterocyclic ring and γ-glutamylamino group, and antifungal agents containing same
MX365051B (en) 2014-11-26 2019-05-09 Univ Mexico Nac Autonoma Novel hydrosoluble compounds derived from benzimidazole used in treating fasciolosis.

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ222495A (en) * 1986-11-21 1991-04-26 Haessle Ab Benzimidazole derivatives and pharmaceutical compositions
SE8801907D0 (en) * 1988-05-20 1988-05-20 Haessle Ab NOVEL PHARMACOLOGICAL COMPOUNDS
CA2083606C (en) * 1990-06-20 2001-08-21 Arne Elof Brandstrom Dialkoxy-pyridinyl-benzimidazole derivatives, process for their preparation and their pharmaceutical use
SE9002206D0 (en) * 1990-06-20 1990-06-20 Haessle Ab NEW COMPOUNDS

Also Published As

Publication number Publication date
IS4079A (en) 1993-06-20
AP397A (en) 1995-08-14
ZA928836B (en) 1993-07-05
NZ246220A (en) 1996-02-27
AU665043B2 (en) 1995-12-14
IL104025A0 (en) 1993-05-13
YU101692A (en) 1995-10-03
CZ146794A3 (en) 1996-02-14
FI942912A (en) 1994-06-17
AU3175293A (en) 1993-07-19
IS3960A (en) 1993-06-20
SI9200402A (en) 1993-06-30
SK73594A3 (en) 1995-02-08
HRP921400A2 (en) 1994-08-31
EP0628049A1 (en) 1994-12-14
WO1993012124A1 (en) 1993-06-24
TW224100B (en) 1994-05-21
HUT68270A (en) 1995-06-28
KR940703840A (en) 1994-12-12
MA22746A1 (en) 1993-07-01
AP9200463A0 (en) 1993-01-31
NO942230L (en) 1994-06-14
FI942912A0 (en) 1994-06-17
TNSN92115A1 (en) 1993-06-08
CN1073446A (en) 1993-06-23
JPH07502503A (en) 1995-03-16
CN1031827C (en) 1996-05-22
MX9207269A (en) 1993-06-01
HU9401840D0 (en) 1994-09-28
CA2124689A1 (en) 1993-06-24
NO942230D0 (en) 1994-06-14

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