SE9002206D0 - New compounds - Google Patents

New compounds

Info

Publication number
SE9002206D0
SE9002206D0 SE9002206A SE9002206A SE9002206D0 SE 9002206 D0 SE9002206 D0 SE 9002206D0 SE 9002206 A SE9002206 A SE 9002206A SE 9002206 A SE9002206 A SE 9002206A SE 9002206 D0 SE9002206 D0 SE 9002206D0
Authority
SE
Sweden
Prior art keywords
gt
lt
carbon atoms
compounds
alkyl containing
Prior art date
Application number
SE9002206A
Other languages
Swedish (sv)
Inventor
A E Braendstroem
Original Assignee
Haessle Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Haessle Ab filed Critical Haessle Ab
Priority to SE9002206A priority Critical patent/SE9002206D0/en
Publication of SE9002206D0 publication Critical patent/SE9002206D0/en
Priority claimed from DE1991631627 external-priority patent/DE69131627T2/en

Links

Abstract

The novel compounds of formula (I), wherein R<1> and R<2>, which are different, is each H, alkyl containing 1-4 carbon atoms or -C(O)-R<6>; one of R<1> or R<2> is always selected from the group -C(O)-R<6>; wherein R<6> is alkyl containing 1-4 carbon atoms or alkoxy containing 1-4 carbon atoms, R<3> is the group -CH2OCOOR<7>, wherein R<7> is alkyl containing 1-6 carbon atoms or benzyl; R<4> and R<5> are the same or different and selected from -CH3, -C2H5, (a), (b) and -CH2CH2OCH3, or R<4> and R<5> form together with the adjacent oxygen atoms attached to the pyridine ring and the carbon atoms in the pyridine ring a ring, wherein the part constituted by R<4> and R<5> is -CH2CH2CH2-, -CH2CH2- or -CH2- as well as pharmaceutical compositions containing such compounds as active ingredient, and the use of the compounds in medicine.
SE9002206A 1990-06-20 1990-06-20 New compounds SE9002206D0 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
SE9002206A SE9002206D0 (en) 1990-06-20 1990-06-20 New compounds

Applications Claiming Priority (58)

Application Number Priority Date Filing Date Title
SE9002206A SE9002206D0 (en) 1990-06-20 1990-06-20 New compounds
ZA914296A ZA9104296B (en) 1990-06-20 1991-06-05 Dialkoxy-pyridinyl-benzimidazole derivatives,process for their preparation and their pharmaceutical use
ZA914297A ZA9104297B (en) 1990-06-20 1991-06-05 Substituted benzimidazoles,process for their preparation and their pharmaceutical use
DE1991631627 DE69131627T2 (en) 1990-06-20 1991-06-11 Dialkoxypyridinylbenzimidazolderivate, methods of making and their pharmaceutical use
PL29729591A PL165898B1 (en) 1990-06-20 1991-06-11 Method of obtaining novel derivatives of dialkoxy pyridinyl benzimidazole
HU924034A HUT62882A (en) 1990-06-20 1991-06-11 Process for producing dialkoxy pyridylmethyl sulfinyl benzimidazole derivatives and pharmaceutical compositions comprising same
JP3511436A JP3049367B2 (en) 1990-06-20 1991-06-11 Dialkoxy - pyridinyl - benzimidazole derivatives, their preparation and medicaments containing it
AT91911618T AT184602T (en) 1990-06-20 1991-06-11 Dialkoxypyridinylbenzimidazolderivate, methods of making and their pharmaceutical use
ES91911618T ES2140391T3 (en) 1990-06-20 1991-06-11 Derivatives dialkoxy-pyridinyl benzimidazole process for their preparation and their pharmaceutical use.
PCT/SE1991/000415 WO1991019711A1 (en) 1990-06-20 1991-06-11 Substituted benzimidazoles, process for their preparation and their pharmaceutical use
EP19910911659 EP0535081A1 (en) 1990-06-20 1991-06-11 Substituted benzimidazoles, process for their preparation and their pharmaceutical use
JP51143591A JPH05507713A (en) 1990-06-20 1991-06-11
EP19910911618 EP0593463B1 (en) 1990-06-20 1991-06-11 Dialkoxy-pyridinyl-benzimidazole derivatives, process for their preparation and their pharmaceutical use
PL29729491A PL166209B1 (en) 1990-06-20 1991-06-11 Method of obtaining novel derivatives of benzimidazole
HU924033A HUT62881A (en) 1990-06-20 1991-06-11 Process for producing substituted benzimidazoles and pharmaceutical compositions comprising same
PCT/SE1991/000416 WO1991019712A1 (en) 1990-06-20 1991-06-11 Dialkoxy-pyridinyl-benzimidazole derivatives, process for their preparation and their pharmaceutical use
CA 2083714 CA2083714A1 (en) 1990-06-20 1991-06-11 Substituted benzimidazoles, process for their preparation and their pharmaceutical use
RO9201543A RO110497B1 (en) 1990-06-20 1991-06-11 Benzimidazole dialcoxipyridynil derivates, preparation process therefor and intermediaries for the process making therefor
CA 2083606 CA2083606C (en) 1990-06-20 1991-06-11 Dialkoxy-pyridinyl-benzimidazole derivatives, process for their preparation and their pharmaceutical use
DE1991631627 DE69131627D1 (en) 1990-06-20 1991-06-11 Dialkoxypyridinylbenzimidazolderivate, methods of making and their pharmaceutical use
RO9201581A RO110493B1 (en) 1990-06-20 1991-06-11 Benzimidazole derivates and preparation processes therefor
AU80097/91A AU649453B2 (en) 1990-06-20 1991-06-11 Substituted benzimidazoles, process for their preparation and their pharmaceutical use
AU80617/91A AU649456B2 (en) 1990-06-20 1991-06-11 Dialkoxy-pyridinyl-benzimidazole derivatives, process for their preparation and their pharmaceutical use
YU104091A YU104091A (en) 1990-06-20 1991-06-12 Dialkoxy-pyridinyl-benzimidazole derivatives of one method for the preparation thereof
YU104191A YU104191A (en) 1990-06-20 1991-06-12 Substituted benzimidazoles and procedure for their preparation
IL9847291A IL98472A (en) 1990-06-20 1991-06-12 Dialkoxy-pyridinyl-benzimidazole derivatives process for their preparation and their pharmaceutical use
IL9847091A IL98470D0 (en) 1990-06-20 1991-06-12 Substituted benzimidazoles,process for their preparation and their pharmaceutical use
TW80104582A TW216418B (en) 1990-06-20 1991-06-12
NZ23854591A NZ238545A (en) 1990-06-20 1991-06-14 Dialkoxy-pyridinyl-benzimidazole derivatives; preparation and pharmaceutical compositions thereof
IE202591A IE912025A1 (en) 1990-06-20 1991-06-14 Substituted benzimidazoles, process for their preparation¹and their pharmaceutical use
NZ23854691A NZ238546A (en) 1990-06-20 1991-06-14 Pyridinyl-substituted benzimidazoles and pharmaceutical compositions
IE202691A IE912026A1 (en) 1990-06-20 1991-06-14 Dialkoxy-pyridinyl-benzimidazole derivatives, process for¹their preparation and their pharmaceutical use
MA22462A MA22199A1 (en) 1990-06-20 1991-06-18 Substituted benzimidazole, the processes for their preparation and their use
MA22461A MA22198A1 (en) 1990-06-20 1991-06-18 Derivatives dialkoxy-pyridinyl-benzimidazole, the processes for their preparation and their use
EG38491A EG19752A (en) 1990-06-20 1991-06-18 Dialkoxy-pyridinyl-benzimidazole derivatives process for their preparation and their pharmaceutical use
AP9100286A AP253A (en) 1990-06-20 1991-06-19 Dialkoxy-pyridinyl-benzimidazole derivatives process for their preparation and thei phamaceutical use.
TNSN91049 TNSN91049A1 (en) 1990-06-20 1991-06-19 Substituted benzimidazoles, processes for their preparation, and their pharmaceutical use
PT9803591A PT98035A (en) 1990-06-20 1991-06-19 Substituted benzimidazoes and pharmaceutical compositions that contain them
TNSN91050 TNSN91050A1 (en) 1990-06-20 1991-06-19 Derivatives dialkoxy-pyridinyl-benzimidazole, processes for their preparation, and their pharmaceutical use
PT9803691A PT98036A (en) 1990-06-20 1991-06-19 Method for preparing new di-alcoxy-pyridinyl-benzimidazole derivatives and pharmaceutical compositions containing them
AP9100285A AP215A (en) 1990-06-20 1991-06-19 Substituted benzimidazoles, process for their preparation and their pharmaceutical use.
US07/718,188 US5430042A (en) 1990-06-20 1991-06-20 Dialkoxy-pyridinyl-benzimidazole derivatives, process for their preparation and their pharmaceutical use
CN 91105024 CN1058212A (en) 1990-06-20 1991-06-20 Substituted benzimidazoles, process for their preparation and their pharmaceutical use
CS911894A CZ279772B6 (en) 1990-06-20 1991-06-20 Substituted benzimidazoles, process of their preparation and pharmaceutical preparation containing thereof as well as their use in the preparation of a medicament
IS3720A IS3720A7 (en) 1990-06-20 1991-06-20 Derivatives step, the dialkoxy-pyridinyl-benzimidazole, aðferðvið features and pharmacological use
CS911893A CZ279434B6 (en) 1990-06-20 1991-06-20 Dialkoxypiridylbenzimidazole derivatives, process of their preparation pharmaceutical preparation in which they are comprised and use of the dialkoxypyridylbenzimidazole derivatives in the preparation of a medicament
CN 91105025 CN1058213A (en) 1990-06-20 1991-06-20 Dialkoxy-pyridinyl-benzimidazole derivatives, process for their preparation and their pharmaceutical use
IS3721A IS3721A7 (en) 1990-06-20 1991-06-20 Conv Deleted benzimidazole, the method of their shape and pharmacological use
OA60306A OA9682A (en) 1990-06-20 1992-11-27 Substituted benzimidazoles process for their preparation and their pharmaceutical use
OA60307A OA9683A (en) 1990-06-20 1992-11-27 Dialkoxy-pyridinyl-benzimidazole derivatives process for their preparation and their pharmaceutical use
NO924650A NO924650D0 (en) 1990-06-20 1992-12-02 Dialkoxy-pyridinyl-benzimidazole derivatives, process for their preparation and their use farmasoeytiske
NO92924775A NO924775L (en) 1990-06-20 1992-12-10 Substituted benzimidazoles, process for their preparation and their use farmasoeytiske
FI925766A FI925766A0 (en) 1990-06-20 1992-12-18 And substituted bensimidazoler, foerfarande Foer deras framstaellning Science deras of pharmaceutical anvaendning
FI925767A FI925767A0 (en) 1990-06-20 1992-12-18 Dialkoxi-pyridinyl-bensimidazolderivater, foerfaranden Foer deras framstaellning Science deras of pharmaceutical anvaendning
LV930820A LV10269B (en) 1990-06-20 1993-06-30 Dialkoxy-pyridinyl-benzimidazole derivatives, process for their preparation and their pharmaceutical use
LV931045A LV10953A (en) 1990-06-20 1993-08-27 Substituted benzimidazoles for use in the manufacture of a pharmaceutical composition
LTIP1713A LT3977B (en) 1990-06-20 1993-12-30 Dialkoxy-pyridinyl-benzimidazole derivatives, process for their preparation and their pharmaceutical use
LTIP1712A LT3952B (en) 1990-06-20 1993-12-30 Substituted benzimidazoles, process for their preparation and their pharmaceutical use

Publications (1)

Publication Number Publication Date
SE9002206D0 true SE9002206D0 (en) 1990-06-20

Family

ID=20379831

Family Applications (1)

Application Number Title Priority Date Filing Date
SE9002206A SE9002206D0 (en) 1990-06-20 1990-06-20 New compounds

Country Status (26)

Country Link
EP (1) EP0535081A1 (en)
JP (1) JPH05507713A (en)
CN (1) CN1058212A (en)
AP (1) AP215A (en)
AU (1) AU649453B2 (en)
CA (1) CA2083714A1 (en)
CZ (1) CZ279772B6 (en)
FI (1) FI925766A0 (en)
HU (1) HUT62881A (en)
IE (1) IE912025A1 (en)
IL (1) IL98470D0 (en)
IS (1) IS3721A7 (en)
LT (2) LT3952B (en)
LV (1) LV10953A (en)
MA (1) MA22199A1 (en)
NO (1) NO924775L (en)
NZ (1) NZ238546A (en)
OA (1) OA9682A (en)
PT (1) PT98035A (en)
RO (1) RO110493B1 (en)
SE (1) SE9002206D0 (en)
TN (1) TNSN91049A1 (en)
TW (1) TW216418B (en)
WO (1) WO1991019711A1 (en)
YU (1) YU104191A (en)
ZA (2) ZA9104297B (en)

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SE9002043D0 (en) * 1990-06-07 1990-06-07 Astra Ab Improved method for synthesis
SE9103776D0 (en) * 1991-12-19 1991-12-19 Astra Ab New compounds
IS4232A (en) * 1993-12-06 1995-06-07 Astra Aktiebolag Súbstitúerað benzimidazole, methods of production and pharmaceutical use
SE9500422D0 (en) * 1995-02-06 1995-02-06 Astra Ab New Oral Pharmaceutical Dosage Forms
SE9500478D0 (en) * 1995-02-09 1995-02-09 Astra Ab New pharmaceutical formulation and process
SE9600070D0 (en) 1996-01-08 1996-01-08 Astra Ab New Oral Pharmaceutical Dosage Forms
JP2003523386A (en) 2000-02-24 2003-08-05 コプラン・リサーチ・ラボラトリーズ・リミテッド Orally administrable acid stable anti-ulcer benzimidazole derivatives
SE0101379D0 (en) 2001-04-18 2001-04-18 Diabact Ab The composition that inhibits gastric acid secretion
US8206741B2 (en) 2001-06-01 2012-06-26 Pozen Inc. Pharmaceutical compositions for the coordinated delivery of NSAIDs
CA2480826C (en) 2002-04-09 2012-02-07 Flamel Technologies Oral pharmaceutical formulation in the form of microcapsule aqueous suspension allowing modified release of active ingredient(s)
SE0203065D0 (en) 2002-10-16 2002-10-16 Diabact Ab Gastric acid secretion inhibiting composition
US8541026B2 (en) 2004-09-24 2013-09-24 Abbvie Inc. Sustained release formulations of opioid and nonopioid analgesics
EP1708684A2 (en) 2003-09-26 2006-10-11 Alza Corporation Drug coating providing high drug loading and methods for providing the same
TW200606163A (en) 2004-04-22 2006-02-16 Eisai Co Ltd Imidazopyridine compound
US20070015782A1 (en) * 2005-04-15 2007-01-18 Eisai Co., Ltd. Benzimidazole compound
US9040564B2 (en) 2005-04-28 2015-05-26 Eisai R&D Management Co., Ltd. Stabilized composition
US7803817B2 (en) 2005-05-11 2010-09-28 Vecta, Ltd. Composition and methods for inhibiting gastric acid secretion
US7981908B2 (en) 2005-05-11 2011-07-19 Vecta, Ltd. Compositions and methods for inhibiting gastric acid secretion
WO2007122686A1 (en) 2006-04-14 2007-11-01 Eisai R & D Management Co., Ltd. Benzimidazole compounds
US9233092B2 (en) 2006-07-25 2016-01-12 Vecta, Ltd. Compositions and methods for inhibiting gastric acid secretion using derivatives of small dicarboxylic acids in combination with PPI
WO2008047681A1 (en) * 2006-10-13 2008-04-24 Eisai R & D Management Co., Ltd. Benzimidazole compound having gastric acid secretion inhibitory activity
US9220698B2 (en) 2008-09-09 2015-12-29 Pozen Inc. Method for delivering a pharmaceutical composition to patient in need thereof
KR20120030106A (en) 2009-06-25 2012-03-27 아스트라제네카 아베 Method for treating a patient at risk for developing an nsaid-associated ulcer
WO2011080502A2 (en) 2009-12-29 2011-07-07 Orexo Ab New pharmaceutical dosage form for the treatment of gastric acid-related disorders
WO2011080500A2 (en) 2009-12-29 2011-07-07 Orexo Ab New pharmaceutical dosage form for the treatment of gastric acid-related disorders
WO2011080501A2 (en) 2009-12-29 2011-07-07 Orexo Ab New pharmaceutical dosage form for the treatment of gastric acid-related disorders
EP2601947A1 (en) 2011-12-05 2013-06-12 Abo Bakr Mohammed Ali Al-Mehdar Fixed-dose combination for treatment of helicobacter pylori associated diseases
CN104519888A (en) 2011-12-28 2015-04-15 波曾公司 Improved compositions and methods for delivery of omeprazole plus acetylsalicylic acid

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Also Published As

Publication number Publication date
ZA9104296B (en) 1992-03-25
ZA9104297B (en) 1992-03-25
JPH05507713A (en) 1993-11-04
HU9204033D0 (en) 1993-03-29
RO110493B1 (en) 1996-01-30
CA2083714A1 (en) 1991-12-21
FI925766A0 (en) 1992-12-18
CN1058212A (en) 1992-01-29
MA22199A1 (en) 1992-04-01
LTIP1712A (en) 1995-08-25
OA9682A (en) 1993-05-15
CS189491A3 (en) 1992-04-15
FI925766A (en) 1992-12-18
NO924775L (en) 1992-12-10
NO924775D0 (en) 1992-12-10
IE912025A1 (en) 1992-01-01
AU649453B2 (en) 1994-05-26
AP215A (en) 1992-09-02
YU104191A (en) 1994-01-20
LV10953A (en) 1995-12-20
NZ238546A (en) 1994-03-25
FI925766D0 (en)
PT98035A (en) 1992-03-31
LTIP1713A (en) 1995-08-25
EP0535081A1 (en) 1993-04-07
LT3952B (en) 1996-05-27
CZ279772B6 (en) 1995-06-14
IL98470D0 (en) 1992-07-15
LT3977B (en) 1996-06-25
TNSN91049A1 (en) 1992-10-25
AP9100285A0 (en) 1991-07-31
AU8009791A (en) 1992-01-07
TW216418B (en) 1993-11-21
HUT62881A (en) 1993-06-28
WO1991019711A1 (en) 1991-12-26
IS3721A7 (en) 1991-12-21

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