NO942230L - Substituted benzimidazoles, processes for their preparation and their use - Google Patents
Substituted benzimidazoles, processes for their preparation and their useInfo
- Publication number
- NO942230L NO942230L NO942230A NO942230A NO942230L NO 942230 L NO942230 L NO 942230L NO 942230 A NO942230 A NO 942230A NO 942230 A NO942230 A NO 942230A NO 942230 L NO942230 L NO 942230L
- Authority
- NO
- Norway
- Prior art keywords
- compounds
- processes
- preparation
- substituted benzimidazoles
- och
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic System
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/6558—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/66—Phosphorus compounds
- A61K31/675—Phosphorus compounds having nitrogen as a ring hetero atom, e.g. pyridoxal phosphate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic System
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/6558—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system
- C07F9/65583—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system each of the hetero rings containing nitrogen as ring hetero atom
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Molecular Biology (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Biochemistry (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
Nye forbindelser av formelen: OCH, OM hvor R1 og R2, som er forskjellige, hver er metyl, -C(0)-CH3 eller -C(0)-OCH3 og hvorved en av R1 eller R2 alltid er metyl; og M er et fysiologisk akseptabelt motion, samt fremgangsmåter for fremstilling av disse forbindelsene, farmasøytiske preparater inneholdene forbindelsene som aktiv bestanddel og anvendelse av forbindelsene innen medisinen.New compounds of the formula: OCH, OM wherein R 1 and R 2 which are different are each methyl, -C (O) -CH 3 or -C (O) -OCH 3 and wherein one of R 1 or R 2 is always methyl; and M is a physiologically acceptable exercise, as well as methods for preparing these compounds, pharmaceutical compositions containing the compounds as active ingredient and the use of the compounds in medicine.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| SE9103776A SE9103776D0 (en) | 1991-12-19 | 1991-12-19 | NEW COMPOUNDS |
| PCT/SE1992/000844 WO1993012124A1 (en) | 1991-12-19 | 1992-12-08 | Substituted benzimidazoles, process for their preparation as well as their use |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| NO942230D0 NO942230D0 (en) | 1994-06-14 |
| NO942230L true NO942230L (en) | 1994-06-14 |
Family
ID=20384667
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO942230A NO942230L (en) | 1991-12-19 | 1994-06-14 | Substituted benzimidazoles, processes for their preparation and their use |
Country Status (25)
| Country | Link |
|---|---|
| EP (1) | EP0628049A1 (en) |
| JP (1) | JPH07502503A (en) |
| KR (1) | KR940703840A (en) |
| CN (1) | CN1031827C (en) |
| AP (1) | AP397A (en) |
| AU (1) | AU665043B2 (en) |
| CA (1) | CA2124689A1 (en) |
| CZ (1) | CZ146794A3 (en) |
| FI (1) | FI942912A (en) |
| HR (1) | HRP921400A2 (en) |
| HU (1) | HUT68270A (en) |
| IL (1) | IL104025A0 (en) |
| IS (2) | IS4079A (en) |
| MA (1) | MA22746A1 (en) |
| MX (1) | MX9207269A (en) |
| NO (1) | NO942230L (en) |
| NZ (1) | NZ246220A (en) |
| SE (1) | SE9103776D0 (en) |
| SI (1) | SI9200402A (en) |
| SK (1) | SK73594A3 (en) |
| TN (1) | TNSN92115A1 (en) |
| TW (1) | TW224100B (en) |
| WO (1) | WO1993012124A1 (en) |
| YU (1) | YU101692A (en) |
| ZA (1) | ZA928836B (en) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE19645974C1 (en) * | 1996-11-07 | 1998-08-13 | Andreas Johannes Kesel | (Z) -5 - [[3-Hydroxy-2-methyl-5 - [(phosphonooxy) methyl] -4-pyridinyl] methylene] -2-thioxo-4-thiazolidinone, process for its preparation and use |
| WO1999033846A2 (en) * | 1997-12-31 | 1999-07-08 | The University Of Kansas | Water soluble prodrugs of secondary and tertiary amine containing drugs and methods of making thereof |
| ATE467637T1 (en) | 2005-07-28 | 2010-05-15 | Intervet Int Bv | NEW BENZIMIDAZOLE(THIO)CARBAMATES WITH ANTIPARASITIC EFFECT AND THEIR SYNTHESIS |
| TWI385169B (en) | 2005-10-31 | 2013-02-11 | Eisai R&D Man Co Ltd | Heterocyclic substituted pyridine derivatives and antifungal agent containing same |
| PL2037914T3 (en) | 2006-06-14 | 2014-04-30 | Intervet Int Bv | A suspension comprising benzimidazole carbamate and a polysorbate |
| TW200841879A (en) | 2007-04-27 | 2008-11-01 | Eisai R&D Man Co Ltd | Pyridine derivatives substituted by heterocyclic ring and phosphonoamino group, and anti-fungal agent containing same |
| US8513287B2 (en) * | 2007-12-27 | 2013-08-20 | Eisai R&D Management Co., Ltd. | Heterocyclic ring and phosphonoxymethyl group substituted pyridine derivatives and antifungal agent containing same |
| US8188119B2 (en) | 2008-10-24 | 2012-05-29 | Eisai R&D Management Co., Ltd | Pyridine derivatives substituted with heterocyclic ring and γ-glutamylamino group, and antifungal agents containing same |
| MX365051B (en) | 2014-11-26 | 2019-05-09 | Univ Mexico Nac Autonoma | Novel hydrosoluble compounds derived from benzimidazole used in treating fasciolosis. |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NZ222495A (en) * | 1986-11-21 | 1991-04-26 | Haessle Ab | Benzimidazole derivatives and pharmaceutical compositions |
| SE8801907D0 (en) * | 1988-05-20 | 1988-05-20 | Haessle Ab | NOVEL PHARMACOLOGICAL COMPOUNDS |
| SE9002206D0 (en) * | 1990-06-20 | 1990-06-20 | Haessle Ab | NEW COMPOUNDS |
| WO1991019712A1 (en) * | 1990-06-20 | 1991-12-26 | Aktiebolaget Astra | Dialkoxy-pyridinyl-benzimidazole derivatives, process for their preparation and their pharmaceutical use |
-
1991
- 1991-12-19 SE SE9103776A patent/SE9103776D0/en unknown
-
1992
- 1992-10-06 IS IS4079A patent/IS4079A/en unknown
- 1992-11-11 TW TW081109053A patent/TW224100B/zh active
- 1992-11-16 ZA ZA928836A patent/ZA928836B/en unknown
- 1992-11-25 YU YU101692A patent/YU101692A/en unknown
- 1992-12-07 HR HR921400A patent/HRP921400A2/en not_active Application Discontinuation
- 1992-12-08 KR KR1019940702131A patent/KR940703840A/en not_active Application Discontinuation
- 1992-12-08 JP JP5510832A patent/JPH07502503A/en active Pending
- 1992-12-08 CA CA002124689A patent/CA2124689A1/en not_active Abandoned
- 1992-12-08 NZ NZ246220A patent/NZ246220A/en unknown
- 1992-12-08 IL IL104025A patent/IL104025A0/en unknown
- 1992-12-08 WO PCT/SE1992/000844 patent/WO1993012124A1/en not_active Application Discontinuation
- 1992-12-08 EP EP93900477A patent/EP0628049A1/en not_active Withdrawn
- 1992-12-08 SK SK735-94A patent/SK73594A3/en unknown
- 1992-12-08 AU AU31752/93A patent/AU665043B2/en not_active Ceased
- 1992-12-08 CZ CZ941467A patent/CZ146794A3/en unknown
- 1992-12-08 HU HU9401840A patent/HUT68270A/en unknown
- 1992-12-14 AP APAP/P/1992/000463A patent/AP397A/en active
- 1992-12-15 MX MX9207269A patent/MX9207269A/en unknown
- 1992-12-16 MA MA23036A patent/MA22746A1/en unknown
- 1992-12-18 TN TNTNSN92115A patent/TNSN92115A1/en unknown
- 1992-12-18 CN CN92114364A patent/CN1031827C/en not_active Expired - Fee Related
- 1992-12-18 SI SI19929200402A patent/SI9200402A/en unknown
- 1992-12-18 IS IS3960A patent/IS3960A/en unknown
-
1994
- 1994-06-14 NO NO942230A patent/NO942230L/en unknown
- 1994-06-17 FI FI942912A patent/FI942912A/en not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| MA22746A1 (en) | 1993-07-01 |
| AU3175293A (en) | 1993-07-19 |
| TW224100B (en) | 1994-05-21 |
| CN1073446A (en) | 1993-06-23 |
| FI942912A0 (en) | 1994-06-17 |
| NO942230D0 (en) | 1994-06-14 |
| AP397A (en) | 1995-08-14 |
| ZA928836B (en) | 1993-07-05 |
| HUT68270A (en) | 1995-06-28 |
| YU101692A (en) | 1995-10-03 |
| HU9401840D0 (en) | 1994-09-28 |
| AU665043B2 (en) | 1995-12-14 |
| MX9207269A (en) | 1993-06-01 |
| IS4079A (en) | 1993-06-20 |
| TNSN92115A1 (en) | 1993-06-08 |
| CA2124689A1 (en) | 1993-06-24 |
| KR940703840A (en) | 1994-12-12 |
| SE9103776D0 (en) | 1991-12-19 |
| NZ246220A (en) | 1996-02-27 |
| HRP921400A2 (en) | 1994-08-31 |
| SI9200402A (en) | 1993-06-30 |
| EP0628049A1 (en) | 1994-12-14 |
| CN1031827C (en) | 1996-05-22 |
| SK73594A3 (en) | 1995-02-08 |
| FI942912A (en) | 1994-06-17 |
| AP9200463A0 (en) | 1993-01-31 |
| JPH07502503A (en) | 1995-03-16 |
| CZ146794A3 (en) | 1996-02-14 |
| IL104025A0 (en) | 1993-05-13 |
| IS3960A (en) | 1993-06-20 |
| WO1993012124A1 (en) | 1993-06-24 |
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