SE437517B - 3-(1-pyrazolyl)-pyridazinderivat - Google Patents

3-(1-pyrazolyl)-pyridazinderivat

Info

Publication number
SE437517B
SE437517B SE7806576A SE7806576A SE437517B SE 437517 B SE437517 B SE 437517B SE 7806576 A SE7806576 A SE 7806576A SE 7806576 A SE7806576 A SE 7806576A SE 437517 B SE437517 B SE 437517B
Authority
SE
Sweden
Prior art keywords
group
amino
pyrazolyl
cyano
acid
Prior art date
Application number
SE7806576A
Other languages
English (en)
Swedish (sv)
Other versions
SE7806576L (sv
Inventor
G Szilagyi
E Kasztreiner
L Tardos
E Kosa
L Jaszlits
G Cseh
A Divald
P Tolnay
S Elek
I Elekes
I Polgari
Original Assignee
Richter Gedeon Vegyeszet
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Richter Gedeon Vegyeszet filed Critical Richter Gedeon Vegyeszet
Publication of SE7806576L publication Critical patent/SE7806576L/xx
Publication of SE437517B publication Critical patent/SE437517B/sv

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
SE7806576A 1977-06-13 1978-06-05 3-(1-pyrazolyl)-pyridazinderivat SE437517B (sv)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
HU77GO1373A HU175471B (hu) 1977-06-13 1977-06-13 Sposob poluchenija novykh proizvodnykh 3-skobka-1-pirazolil-skobka zakryta-piridazina

Publications (2)

Publication Number Publication Date
SE7806576L SE7806576L (sv) 1978-12-14
SE437517B true SE437517B (sv) 1985-03-04

Family

ID=10996834

Family Applications (1)

Application Number Title Priority Date Filing Date
SE7806576A SE437517B (sv) 1977-06-13 1978-06-05 3-(1-pyrazolyl)-pyridazinderivat

Country Status (25)

Country Link
US (1) US4251658A (cs)
JP (1) JPS5416487A (cs)
AT (1) AT357548B (cs)
AU (1) AU521394B2 (cs)
BE (1) BE867967A (cs)
BG (1) BG28709A3 (cs)
CA (1) CA1095912A (cs)
CH (1) CH638202A5 (cs)
CS (1) CS204029B2 (cs)
DD (1) DD140043A5 (cs)
DE (1) DE2825906A1 (cs)
DK (1) DK263078A (cs)
ES (1) ES470750A1 (cs)
FI (1) FI64156C (cs)
FR (1) FR2394542A1 (cs)
GB (1) GB1603958A (cs)
HU (1) HU175471B (cs)
IL (1) IL54816A (cs)
IT (1) IT1098216B (cs)
NL (1) NL7806380A (cs)
NO (1) NO149210C (cs)
PL (1) PL111252B1 (cs)
SE (1) SE437517B (cs)
SU (2) SU797577A3 (cs)
YU (1) YU140078A (cs)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU176100B (en) * 1977-10-25 1980-12-28 Gyogyszerkutato Intezet Process for preparing new 3-/1-pyrazolyl/-pyridazine derivatives
DE2935359A1 (de) * 1979-09-01 1981-03-26 Basf Ag, 67063 Ludwigshafen 6-imidazolyl-3-hydrazino-pyridazine
DE3130251A1 (de) * 1981-07-31 1983-02-17 A. Nattermann & Cie GmbH, 5000 Köln 6-(4-((omega)-(1-imidazolyl)-alkyl)-phenyl)-3-oxo -2,3,4,5-tetrahydro-pyridazine und deren saeureadditionssalze, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische praeparate
US4353905A (en) * 1981-09-17 1982-10-12 Warner-Lambert Company Substituted 4,5-dihydro-6-[4-(1H-imidazol-1-yl)phenyl]-3(2H)-pyridazinones and 6-[4-(1H-imidazol-1-yl)phenyl]-3(2H)-pyridazinones
US4590194A (en) * 1981-10-05 1986-05-20 Sterling Drug Inc. 3-[methyl or dimethyl)amino]-6-(pyridinyl)pyridazines and their cardiotonic use
US4503056A (en) * 1982-03-02 1985-03-05 Abbott Laboratories 1-(Pyridazinyl)pyrazoline derivatives
DE3825867A1 (de) * 1988-03-04 1989-09-14 Bayer Ag Heterocyclisch substituierte sulfonylaminoazole und ihre verwendung als herbizide
US5536701A (en) * 1994-10-11 1996-07-16 Monsanto Company 3-pyrazolyloxypyridazines, herbicidal compositions and uses thereof
FR2847160A1 (fr) * 2002-11-20 2004-05-21 Oreal Composition capillaire contenant un compose pyrasol-carboxamide, son utilisation pour stimuler la pousse des cheveux et/ou freiner leur chute
WO2004047776A1 (fr) * 2002-11-20 2004-06-10 L'oreal Utilisation d’un compose pyrazolcarboxamide pour stimuler la pousse des fibres keratiniques et/ou freiner leur chute
RU2442775C2 (ru) * 2005-07-04 2012-02-20 Хай Пойнт Фармасьютикалс, ЛЛС Антагонисты гистаминовых н3-рецепторов
MX2007015675A (es) * 2005-07-04 2008-02-20 Novo Nordisk As Antagonistas del receptor de histamina h3.
CA2653062A1 (en) * 2006-05-23 2007-11-29 Transtech Pharma, Inc. 6- (4-cyclopropylpiperazin-1-yl) -2 ' -methyl- [3, 4 ' ] -bipyridine and its use as a medicament
BRPI0711370A2 (pt) * 2006-05-29 2011-11-01 High Point Pharmaceuticals Llc 3-(1,3-benzodioxol-5-il)-6-(4-ciclopropilpiperazin-1-il)pi ridazina e seus sais e solvatos e seu uso como antagonista receptor h3 de histamina
EP2014656A3 (en) * 2007-06-11 2011-08-24 High Point Pharmaceuticals, LLC New heteocyclic h3 antagonists
AR081331A1 (es) 2010-04-23 2012-08-08 Cytokinetics Inc Amino- pirimidinas composiciones de las mismas y metodos para el uso de los mismos
AR081626A1 (es) * 2010-04-23 2012-10-10 Cytokinetics Inc Compuestos amino-piridazinicos, composiciones farmaceuticas que los contienen y uso de los mismos para tratar trastornos musculares cardiacos y esqueleticos
WO2011133920A1 (en) 2010-04-23 2011-10-27 Cytokinetics, Inc. Certain amino-pyridines and amino-triazines, compositions thereof, and methods for their use

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1595920B2 (de) * 1964-11-04 1978-08-10 Merck Patent Gmbh, 6100 Darmstadt 4-(co-Piperazinoalkyl)-pyrazole, ihre Salze und Verfahren zu ihrer Herstellung
JPS5831347B2 (ja) * 1975-09-05 1983-07-05 中外製薬株式会社 ピラゾリルピリダジンユウドウタイノ セイホウ

Also Published As

Publication number Publication date
BG28709A3 (bg) 1980-06-16
NO149210B (no) 1983-11-28
JPS569506B2 (cs) 1981-03-02
DK263078A (da) 1978-12-14
CH638202A5 (de) 1983-09-15
DE2825906A1 (de) 1979-01-18
GB1603958A (en) 1981-12-02
HU175471B (hu) 1980-08-28
CS204029B2 (en) 1981-03-31
NO782043L (no) 1978-12-14
ATA414478A (de) 1979-12-15
FI64156C (fi) 1983-10-10
NO149210C (no) 1984-03-07
IT1098216B (it) 1985-09-07
ES470750A1 (es) 1979-01-16
IL54816A0 (en) 1978-07-31
CA1095912A (en) 1981-02-17
BE867967A (fr) 1978-12-11
FR2394542B1 (cs) 1980-12-05
PL111252B1 (en) 1980-08-30
US4251658A (en) 1981-02-17
SU797577A3 (ru) 1981-01-15
IT7824490A0 (it) 1978-06-13
YU140078A (en) 1983-01-21
FI781856A7 (fi) 1978-12-14
SU860703A1 (ru) 1981-08-30
SE7806576L (sv) 1978-12-14
AU521394B2 (en) 1982-04-01
AT357548B (de) 1980-07-10
IL54816A (en) 1981-09-13
FR2394542A1 (fr) 1979-01-12
PL207570A1 (pl) 1979-05-21
AU3683678A (en) 1979-12-06
FI64156B (fi) 1983-06-30
JPS5416487A (en) 1979-02-07
DD140043A5 (de) 1980-02-06
NL7806380A (nl) 1978-12-15

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