RU2501550C2 - Сублингвальная спреевая композиция, содержащая дигидроартемизинин - Google Patents
Сублингвальная спреевая композиция, содержащая дигидроартемизинин Download PDFInfo
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- RU2501550C2 RU2501550C2 RU2011139637/15A RU2011139637A RU2501550C2 RU 2501550 C2 RU2501550 C2 RU 2501550C2 RU 2011139637/15 A RU2011139637/15 A RU 2011139637/15A RU 2011139637 A RU2011139637 A RU 2011139637A RU 2501550 C2 RU2501550 C2 RU 2501550C2
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
- A61K47/14—Esters of carboxylic acids, e.g. fatty acid monoglycerides, medium-chain triglycerides, parabens or PEG fatty acid esters
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0043—Nose
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/10—Dispersions; Emulsions
- A61K9/12—Aerosols; Foams
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/14—Ectoparasiticides, e.g. scabicides
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
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- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Epidemiology (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Dispersion Chemistry (AREA)
- Tropical Medicine & Parasitology (AREA)
- Engineering & Computer Science (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Nutrition Science (AREA)
- Physiology (AREA)
- Otolaryngology (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines Containing Plant Substances (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB0906971.7 | 2009-04-23 | ||
| PCT/GB2009/050415 WO2010122275A1 (en) | 2009-04-23 | 2009-04-23 | Pharmaceutical preparation |
| GBPCT/GB2009/050415 | 2009-04-23 | ||
| GB0906971.7A GB2469791B (en) | 2009-04-23 | 2009-04-23 | Transmucosal formulation of compounds providing dihydroartemesinin for use in the treatment of neoplastic disease |
| PCT/GB2010/050672 WO2010122356A1 (en) | 2009-04-23 | 2010-04-23 | Sublingual spray formulation comprising dihydroartemesinin |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| RU2011139637A RU2011139637A (ru) | 2013-05-27 |
| RU2501550C2 true RU2501550C2 (ru) | 2013-12-20 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| RU2011139637/15A RU2501550C2 (ru) | 2009-04-23 | 2010-04-23 | Сублингвальная спреевая композиция, содержащая дигидроартемизинин |
Country Status (23)
| Country | Link |
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| US (4) | US20120157518A1 (enExample) |
| EP (1) | EP2424523B1 (enExample) |
| JP (1) | JP5795760B2 (enExample) |
| CN (1) | CN102395362B (enExample) |
| AU (1) | AU2010240654C1 (enExample) |
| BR (1) | BRPI1014887A8 (enExample) |
| CA (1) | CA2756925A1 (enExample) |
| DK (1) | DK2424523T3 (enExample) |
| ES (1) | ES2390046T3 (enExample) |
| HR (1) | HRP20120711T1 (enExample) |
| IL (1) | IL215453A (enExample) |
| ME (1) | ME02008B (enExample) |
| MX (1) | MX2011010961A (enExample) |
| MY (1) | MY155646A (enExample) |
| NZ (1) | NZ595469A (enExample) |
| PL (1) | PL2424523T3 (enExample) |
| PT (1) | PT2424523E (enExample) |
| RS (1) | RS52430B (enExample) |
| RU (1) | RU2501550C2 (enExample) |
| SG (1) | SG175162A1 (enExample) |
| SI (1) | SI2424523T1 (enExample) |
| WO (1) | WO2010122356A1 (enExample) |
| ZA (1) | ZA201107088B (enExample) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB0720967D0 (en) * | 2007-10-25 | 2007-12-05 | Protophama Ltd | Anti-material pharmaceutical composition |
| CA2756879A1 (en) * | 2009-04-23 | 2010-10-28 | Londonpharma Ltd. | Sublingual pharmaceutical composition comprising a neutral oil |
| CA2898113C (en) * | 2013-01-14 | 2022-05-31 | Health Clinics Limited | Combination cancer therapeutics and uses thereof |
| US20170326102A1 (en) | 2014-11-27 | 2017-11-16 | Cipla Limited | Pharmaceutical Composition Comprising an Artemisinin Derivative for Nasal or Pulmonary Delivery |
| JP2020033304A (ja) * | 2018-08-30 | 2020-03-05 | 医療法人ふじいやさか | 薬剤又はサプリメント、組成物、及び水素供給器の使用 |
Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20040092583A1 (en) * | 2001-01-02 | 2004-05-13 | Elizabeth Shanahan-Prendergast | Treatment for inhibiting neoplastic lesions |
| RU2236413C2 (ru) * | 1998-07-14 | 2004-09-20 | Байер Акциенгезельшафт | Производные артемизинина, способ их получения, фармацевтическая композиция на их основе и способ лечения |
| US20060084675A1 (en) * | 2004-10-18 | 2006-04-20 | Thomas Efferth | Combined treatment with artesunate and an epidermal growth factor receptor kinase inhibitor |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20030082107A1 (en) * | 1997-10-01 | 2003-05-01 | Dugger Harry A. | Buccal, polar and non-polar spray or capsule containing drugs for treating an infectious disease or cancer |
| CH692321A5 (de) * | 1997-11-03 | 2002-05-15 | Mepha Ag | Pharmazeutisch wirksame Zusammensetzung, welche eine gegen Malariaparasiten wirksame Substanz enthält. |
| US20060257463A1 (en) * | 2002-05-31 | 2006-11-16 | University Of Mississippi | Transmucosal delivery of cannabinoids |
| JP2005529938A (ja) * | 2002-06-06 | 2005-10-06 | ユニバーシティ オブ ワシントン | 癌の発症を予防または遅延するためのアルテミシニン様化合物を使用する方法 |
| WO2004075921A1 (en) * | 2003-02-26 | 2004-09-10 | Vrije Universiteit Brussel | Inclusion complex of artemisinin or derivates thereof with cyclodextrins |
| US20060233895A1 (en) * | 2005-04-15 | 2006-10-19 | Brown Paul R | Herbal remedy for treating Lyme disease |
| ATE544444T1 (de) * | 2005-10-11 | 2012-02-15 | Yissum Res Dev Co | Zusammensetzungen für die nasale abgabe |
| CN100418524C (zh) * | 2005-10-26 | 2008-09-17 | 重庆医药工业研究院有限责任公司 | 一种稳定的青蒿素及青蒿素衍生物的药物组合物 |
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2010
- 2010-04-23 DK DK10715337.1T patent/DK2424523T3/da active
- 2010-04-23 SI SI201030076T patent/SI2424523T1/sl unknown
- 2010-04-23 CN CN201080017965.1A patent/CN102395362B/zh not_active Expired - Fee Related
- 2010-04-23 EP EP10715337A patent/EP2424523B1/en active Active
- 2010-04-23 ES ES10715337T patent/ES2390046T3/es active Active
- 2010-04-23 RS RS20120393A patent/RS52430B/sr unknown
- 2010-04-23 MX MX2011010961A patent/MX2011010961A/es active IP Right Grant
- 2010-04-23 MY MYPI2011005080A patent/MY155646A/en unknown
- 2010-04-23 SG SG2011073954A patent/SG175162A1/en unknown
- 2010-04-23 PL PL10715337T patent/PL2424523T3/pl unknown
- 2010-04-23 US US13/265,518 patent/US20120157518A1/en not_active Abandoned
- 2010-04-23 HR HRP20120711AT patent/HRP20120711T1/hr unknown
- 2010-04-23 AU AU2010240654A patent/AU2010240654C1/en not_active Ceased
- 2010-04-23 WO PCT/GB2010/050672 patent/WO2010122356A1/en not_active Ceased
- 2010-04-23 RU RU2011139637/15A patent/RU2501550C2/ru active
- 2010-04-23 JP JP2012506584A patent/JP5795760B2/ja not_active Expired - Fee Related
- 2010-04-23 BR BRPI1014887A patent/BRPI1014887A8/pt not_active Application Discontinuation
- 2010-04-23 PT PT10715337T patent/PT2424523E/pt unknown
- 2010-04-23 CA CA2756925A patent/CA2756925A1/en not_active Abandoned
- 2010-04-23 NZ NZ595469A patent/NZ595469A/xx not_active IP Right Cessation
- 2010-04-23 ME MEP-2012-393A patent/ME02008B/me unknown
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2011
- 2011-09-28 ZA ZA2011/07088A patent/ZA201107088B/en unknown
- 2011-10-02 IL IL215453A patent/IL215453A/en active IP Right Grant
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2015
- 2015-07-30 US US14/813,424 patent/US20160022629A1/en not_active Abandoned
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2017
- 2017-09-06 US US15/697,240 patent/US20170368023A1/en not_active Abandoned
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2018
- 2018-10-18 US US16/164,610 patent/US20190142737A1/en not_active Abandoned
Patent Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2236413C2 (ru) * | 1998-07-14 | 2004-09-20 | Байер Акциенгезельшафт | Производные артемизинина, способ их получения, фармацевтическая композиция на их основе и способ лечения |
| US20040092583A1 (en) * | 2001-01-02 | 2004-05-13 | Elizabeth Shanahan-Prendergast | Treatment for inhibiting neoplastic lesions |
| US20060084675A1 (en) * | 2004-10-18 | 2006-04-20 | Thomas Efferth | Combined treatment with artesunate and an epidermal growth factor receptor kinase inhibitor |
Non-Patent Citations (1)
| Title |
|---|
| Nakase I et. all. "Anticancer properties of artemisinin derivatives and their targeted delivery by transferrin conjugation.", Int J Pharm. 2008 Apr 16; 354(1-2):28-33. Epub 2007 Sep 6., найдено в PubMed PMID: 17942255, реферат. Buommino E et. all. "Artemisinin reduces human melanoma cell migration by down-regulating alpha V beta 3 integrin and reducing metalloproteinase 2 production", Invest New Drugs. 2009 Oct; 27(5):412-8. doi: 10.1007/s10637-008-9188-2. Epub 2008 Oct 28. найдено в PubMed PMID: 18956140, реферат. * |
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