RU2396251C2 - Производные альфа-аминоамидов, применимые в качестве противовоспалительных агентов - Google Patents
Производные альфа-аминоамидов, применимые в качестве противовоспалительных агентов Download PDFInfo
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- RU2396251C2 RU2396251C2 RU2006105634/04A RU2006105634A RU2396251C2 RU 2396251 C2 RU2396251 C2 RU 2396251C2 RU 2006105634/04 A RU2006105634/04 A RU 2006105634/04A RU 2006105634 A RU2006105634 A RU 2006105634A RU 2396251 C2 RU2396251 C2 RU 2396251C2
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- Prior art keywords
- inflammatory
- benzylamino
- fluorobenzyloxy
- propanamide
- inflammation
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| US49772203P | 2003-08-25 | 2003-08-25 | |
| US60/497,722 | 2003-08-25 |
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| RU2006105634A RU2006105634A (ru) | 2006-08-10 |
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| RU2006105634/04A RU2396251C2 (ru) | 2003-08-25 | 2004-04-22 | Производные альфа-аминоамидов, применимые в качестве противовоспалительных агентов |
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| PT (1) | PT1658062E (enExample) |
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| SI (1) | SI1658062T1 (enExample) |
| WO (1) | WO2005018627A1 (enExample) |
Cited By (1)
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| WO2012102645A2 (en) | 2011-01-27 | 2012-08-02 | «Garmonia», Ltd. | Peptide pharmaceutical composition, means for treatment of helicobacter pylori induced gastroduodenal diseases on the basis thereof, and a method of use thereof |
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| US20070276046A1 (en) * | 2003-08-25 | 2007-11-29 | Patricia Salvati | Alpha-Aminoamide Derivatives Useful as Anti-Inflammatory Agents |
| EP1557166A1 (en) | 2004-01-21 | 2005-07-27 | Newron Pharmaceuticals S.p.A. | Alpha-aminoamide derivatives useful in the treatment of lower urinary tract disorders |
| RS51411B (sr) * | 2004-09-10 | 2011-02-28 | Newron Pharmaceuticals S.P.A. | Upotreba (r)-(halobenziloksi) benzilamino-propanamida kao selektivnih modulatora natrijumovih i/ili kalcijumovih kanala |
| IN266803B (enExample) | 2005-12-22 | 2015-06-03 | Newron Pharm Spa | |
| KR101491541B1 (ko) | 2006-06-19 | 2015-02-09 | 뉴론 파마슈티칼즈 에스. 피. 에이. | 2-［4-(3- 및 2-플루오로벤질옥시)벤질아미노)프로판 아미드의 제조방법 |
| TR201802576T4 (tr) | 2007-06-15 | 2018-03-21 | Newron Pharm Spa | Sübsti̇tüe edi̇lmi̇ş 2-[2-(feni̇l)eti̇lami̇no]alkanami̇t türevleri̇ ve bunlarin sodyum ve/veya kalsi̇yum kanal modülatörleri̇ olarak kullanimi |
| EP3257842B1 (en) | 2007-12-11 | 2020-11-18 | Newron Pharmaceuticals S.p.A. | Therapeutic use of 2-[4-(3- or 2-fluorobenzyloxy)benzylamino]propanamides with high purity degree |
| LT2563355T (lt) | 2010-04-27 | 2016-09-26 | Newron Pharmaceuticals S.P.A. | Ralfinamido metansulfonato druskų arba jų r-enentiomerų gavimo būdas |
| DE102012108965B4 (de) | 2012-09-24 | 2014-08-14 | Exscitron Gmbh | Stromquelle mit verbesserter Dimmvorrichtung |
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| RU2164512C1 (ru) * | 1999-07-27 | 2001-03-27 | Всероссийский научный центр по безопасности биологически активных веществ | Производные аминокислот, проявляющие антиаритмическую активность |
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| IL94466A (en) * | 1989-05-25 | 1995-01-24 | Erba Carlo Spa | Pharmaceutical preparations containing the history of A-amino carboxamide N-phenylalkyl are converted into such new compounds and their preparation |
| GB9726987D0 (en) * | 1997-12-22 | 1998-02-18 | Glaxo Group Ltd | Compounds |
| GB9727523D0 (en) * | 1997-12-31 | 1998-02-25 | Pharmacia & Upjohn Spa | Alpha-aminoamide derivatives useful as analgesic agents |
| SE9801494D0 (sv) * | 1998-04-28 | 1998-04-28 | Astra Pharma Prod | Novel use |
| GB9930079D0 (en) * | 1999-12-20 | 2000-02-09 | Glaxo Group Ltd | Medicaments |
| ATE357257T1 (de) * | 2000-07-27 | 2007-04-15 | Pharmacia Corp | Kombinationstherapie mit epoxy-steroidalen aldosteronantagonisten und kalziumkanalblocker zur behandlung von kongestivem herzversagen |
| CN1274306C (zh) * | 2001-09-03 | 2006-09-13 | 纽朗制药有限公司 | 包含加巴喷丁或其类似物和α－氨基酰胺的药物组合物及其止痛应用 |
| JP2005514412A (ja) * | 2001-12-27 | 2005-05-19 | オーソ−マクニール・フアーマシユーチカル・インコーポレーテツド | 中枢神経系疾患を処置するために有用なアロイルピロールヘテロアリールおよびメタノール類 |
| EP1438956A1 (en) * | 2003-01-16 | 2004-07-21 | Newron Pharmaceuticals S.p.A. | Alpha-aminoamide derivatives useful as antimigraine agents |
| CA2514574A1 (en) * | 2003-01-30 | 2004-08-12 | Dynogen Pharmaceuticals, Inc. | Use of sodium channel modulators for treating gastrointestinal tract disorders |
| AU2004207010A1 (en) * | 2003-01-30 | 2004-08-12 | Dynogen Pharmaceuticals, Inc. | Methods of treating lower urinary tract disorders using sodium channel modulators |
| AR044007A1 (es) * | 2003-04-11 | 2005-08-24 | Newron Pharmaceuticals Inc | Metodos para el tratamiento de la enfermedad de parkinson |
| US20070276046A1 (en) * | 2003-08-25 | 2007-11-29 | Patricia Salvati | Alpha-Aminoamide Derivatives Useful as Anti-Inflammatory Agents |
| EP1588704A1 (en) * | 2004-04-22 | 2005-10-26 | Newron Pharmaceuticals S.p.A. | Alpha-aminoamide derivatives useful in the treatment of restless legs syndrome and addictive disorders |
| RS51411B (sr) * | 2004-09-10 | 2011-02-28 | Newron Pharmaceuticals S.P.A. | Upotreba (r)-(halobenziloksi) benzilamino-propanamida kao selektivnih modulatora natrijumovih i/ili kalcijumovih kanala |
| IN266803B (enExample) * | 2005-12-22 | 2015-06-03 | Newron Pharm Spa | |
| EP1870097A1 (en) * | 2006-06-15 | 2007-12-26 | Newron Pharmaceuticals S.p.A. | Alpha-aminoamide derivatives useful in the treatment of cognitive disorders |
| KR101491541B1 (ko) * | 2006-06-19 | 2015-02-09 | 뉴론 파마슈티칼즈 에스. 피. 에이. | 2-［4-(3- 및 2-플루오로벤질옥시)벤질아미노)프로판 아미드의 제조방법 |
| TR201802576T4 (tr) * | 2007-06-15 | 2018-03-21 | Newron Pharm Spa | Sübsti̇tüe edi̇lmi̇ş 2-[2-(feni̇l)eti̇lami̇no]alkanami̇t türevleri̇ ve bunlarin sodyum ve/veya kalsi̇yum kanal modülatörleri̇ olarak kullanimi |
| EP3257842B1 (en) * | 2007-12-11 | 2020-11-18 | Newron Pharmaceuticals S.p.A. | Therapeutic use of 2-[4-(3- or 2-fluorobenzyloxy)benzylamino]propanamides with high purity degree |
| CN101903021B (zh) * | 2007-12-19 | 2012-11-14 | 纽朗制药有限公司 | 用于治疗精神病的α-氨基酰胺衍生物 |
-
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- 2004-04-22 US US10/569,403 patent/US20070276046A1/en not_active Abandoned
- 2004-04-22 AT AT04728870T patent/ATE457724T1/de active
- 2004-04-22 CA CA2536764A patent/CA2536764C/en not_active Expired - Lifetime
- 2004-04-22 EP EP04728870A patent/EP1658062B1/en not_active Expired - Lifetime
- 2004-04-22 IL IL173886A patent/IL173886A/en active IP Right Grant
- 2004-04-22 SI SI200431379T patent/SI1658062T1/sl unknown
- 2004-04-22 RU RU2006105634/04A patent/RU2396251C2/ru active
- 2004-04-22 JP JP2006524432A patent/JP5042625B2/ja not_active Expired - Lifetime
- 2004-04-22 KR KR1020067003725A patent/KR101233711B1/ko not_active Expired - Lifetime
- 2004-04-22 NZ NZ545502A patent/NZ545502A/en not_active IP Right Cessation
- 2004-04-22 DE DE602004025586T patent/DE602004025586D1/de not_active Expired - Lifetime
- 2004-04-22 PL PL04728870T patent/PL1658062T3/pl unknown
- 2004-04-22 CN CNA2004800242753A patent/CN1842328A/zh active Pending
- 2004-04-22 BR BRPI0413982-8A patent/BRPI0413982A/pt not_active Application Discontinuation
- 2004-04-22 WO PCT/IB2004/001574 patent/WO2005018627A1/en not_active Ceased
- 2004-04-22 ES ES04728870T patent/ES2339021T3/es not_active Expired - Lifetime
- 2004-04-22 PT PT04728870T patent/PT1658062E/pt unknown
- 2004-04-22 AU AU2004266494A patent/AU2004266494B2/en not_active Expired
- 2004-04-22 DK DK04728870.9T patent/DK1658062T3/da active
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2006
- 2006-02-23 NO NO20060896A patent/NO335245B1/no unknown
-
2009
- 2009-08-20 US US12/544,456 patent/US20100016440A1/en not_active Abandoned
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2010
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| RU2164512C1 (ru) * | 1999-07-27 | 2001-03-27 | Всероссийский научный центр по безопасности биологически активных веществ | Производные аминокислот, проявляющие антиаритмическую активность |
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Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2012102645A2 (en) | 2011-01-27 | 2012-08-02 | «Garmonia», Ltd. | Peptide pharmaceutical composition, means for treatment of helicobacter pylori induced gastroduodenal diseases on the basis thereof, and a method of use thereof |
Also Published As
| Publication number | Publication date |
|---|---|
| US20100016440A1 (en) | 2010-01-21 |
| DK1658062T3 (da) | 2010-05-31 |
| IL173886A0 (en) | 2006-07-05 |
| NO335245B1 (no) | 2014-10-27 |
| KR20060128825A (ko) | 2006-12-14 |
| EP1658062B1 (en) | 2010-02-17 |
| SI1658062T1 (sl) | 2010-05-31 |
| IL173886A (en) | 2012-09-24 |
| CY1109992T1 (el) | 2014-09-10 |
| PL1658062T3 (pl) | 2010-07-30 |
| RU2006105634A (ru) | 2006-08-10 |
| CA2536764C (en) | 2013-09-17 |
| KR101233711B1 (ko) | 2013-02-18 |
| CN1842328A (zh) | 2006-10-04 |
| US20070276046A1 (en) | 2007-11-29 |
| NZ545502A (en) | 2010-04-30 |
| WO2005018627A8 (en) | 2005-09-01 |
| EP1658062A1 (en) | 2006-05-24 |
| DE602004025586D1 (de) | 2010-04-01 |
| ES2339021T3 (es) | 2010-05-14 |
| WO2005018627A1 (en) | 2005-03-03 |
| NO20060896L (no) | 2006-03-09 |
| JP5042625B2 (ja) | 2012-10-03 |
| AU2004266494A1 (en) | 2005-03-03 |
| PT1658062E (pt) | 2010-03-31 |
| AU2004266494B2 (en) | 2010-04-08 |
| ATE457724T1 (de) | 2010-03-15 |
| BRPI0413982A (pt) | 2006-11-07 |
| CA2536764A1 (en) | 2005-03-03 |
| JP2007503424A (ja) | 2007-02-22 |
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