RU2376297C2 - Производные изотиомочевины и способ их получения, их применение и фармацевтическая композиция - Google Patents
Производные изотиомочевины и способ их получения, их применение и фармацевтическая композиция Download PDFInfo
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- RU2376297C2 RU2376297C2 RU2006134019/04A RU2006134019A RU2376297C2 RU 2376297 C2 RU2376297 C2 RU 2376297C2 RU 2006134019/04 A RU2006134019/04 A RU 2006134019/04A RU 2006134019 A RU2006134019 A RU 2006134019A RU 2376297 C2 RU2376297 C2 RU 2376297C2
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- isothiourea
- dihydroimidazo
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| GB0404434.3 | 2004-02-27 | ||
| GBGB0404434.3A GB0404434D0 (en) | 2004-02-27 | 2004-02-27 | Organic compounds |
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| RU2006134019A RU2006134019A (ru) | 2008-04-10 |
| RU2376297C2 true RU2376297C2 (ru) | 2009-12-20 |
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| EP (1) | EP1720845A1 (https=) |
| JP (1) | JP2007523941A (https=) |
| KR (1) | KR20060124722A (https=) |
| CN (1) | CN1922158A (https=) |
| AU (1) | AU2005219531B2 (https=) |
| CA (1) | CA2556386A1 (https=) |
| GB (1) | GB0404434D0 (https=) |
| RU (1) | RU2376297C2 (https=) |
| WO (1) | WO2005085219A1 (https=) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2503450C1 (ru) * | 2012-04-19 | 2014-01-10 | Федеральное Государственное Бюджетное Учреждение "Медицинский Радиологический Научный Центр" Министерства Здравоохранения и Социального Развития Российской Федерации (ФГБУ МРНЦ Минздравсоцразвития России) | Противоопухолевое средство |
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| WO2007058322A1 (ja) | 2005-11-18 | 2007-05-24 | Ono Pharmaceutical Co., Ltd. | 塩基性基を含有する化合物およびその用途 |
| WO2009005675A1 (en) | 2007-06-28 | 2009-01-08 | Abbott Laboratories | Novel triazolopyridazines |
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| US20100305210A1 (en) * | 2007-11-06 | 2010-12-02 | Barkan-Farma S.R.L. | S-alkylisothiouronium derivatives for treating abnormal uterine bleeding disorders |
| CN102088856B (zh) | 2008-07-09 | 2015-11-25 | 巴斯夫欧洲公司 | 包含异*唑啉化合物的杀虫活性混合物i |
| US8921328B2 (en) | 2010-09-14 | 2014-12-30 | Glycomimetics, Inc. | E-selectin antagonists |
| WO2012061662A1 (en) * | 2010-11-03 | 2012-05-10 | Glycomimetics, Inc. | Glycomimetic-peptidomimetic inhibitors of e-selectins and cxcr4 chemokine receptors |
| PT2794626T (pt) | 2011-12-22 | 2018-01-12 | Glycomimetics Inc | Compostos de antagonistas de e-selectina |
| CA2891514C (en) | 2012-12-07 | 2020-08-25 | Glycomimetics, Inc. | Compounds, compositions and methods using e-selectin antagonists for mobilization of hematopoietic cells |
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| WO2017151708A1 (en) | 2016-03-02 | 2017-09-08 | Glycomimetics, Inc. | Methods for the treatment and/or prevention of cardiovescular disease by inhibition of e-selectin |
| EP3497131B1 (en) | 2016-08-08 | 2022-03-09 | GlycoMimetics, Inc. | Combination of t-cell checkpoint inhibitors with inhibitors of e-selectin or cxcr4, or with heterobifunctional inhibitors of both e-selectin and cxcr4. |
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| CA3054605A1 (en) | 2017-03-15 | 2018-09-20 | Glycomimetics, Inc. | Galactopyranosyl-cyclohexyl derivatives as e-selectin antagonists |
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| CN111566117A (zh) | 2017-12-29 | 2020-08-21 | 糖模拟物有限公司 | E-选择蛋白和半乳凝素-3的异双功能抑制剂 |
| WO2019173229A1 (en) | 2018-03-05 | 2019-09-12 | Glycomimetics, Inc. | Methods for treating acute myeloid leukemia and related conditions |
| US11845771B2 (en) | 2018-12-27 | 2023-12-19 | Glycomimetics, Inc. | Heterobifunctional inhibitors of E-selectin and galectin-3 |
| CA3174634A1 (en) * | 2020-03-11 | 2021-09-16 | Biolinerx Ltd. | Cxcr4 inhibitor for the treatment of acute respiratory distress syndrome and viral infections |
| MX2023003409A (es) * | 2020-09-28 | 2023-06-26 | Ermium Therapeutics | Derivados de isotiourea ciclica como moduladores de cxcr4. |
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- 2005-02-25 EP EP05715554A patent/EP1720845A1/en not_active Withdrawn
- 2005-02-25 WO PCT/EP2005/002014 patent/WO2005085219A1/en not_active Ceased
- 2005-02-25 US US10/590,399 patent/US7671078B2/en not_active Expired - Fee Related
- 2005-02-25 RU RU2006134019/04A patent/RU2376297C2/ru not_active IP Right Cessation
- 2005-02-25 JP JP2007500168A patent/JP2007523941A/ja active Pending
- 2005-02-25 CA CA002556386A patent/CA2556386A1/en not_active Abandoned
- 2005-02-25 AU AU2005219531A patent/AU2005219531B2/en not_active Ceased
- 2005-02-25 CN CNA2005800060942A patent/CN1922158A/zh active Pending
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2503450C1 (ru) * | 2012-04-19 | 2014-01-10 | Федеральное Государственное Бюджетное Учреждение "Медицинский Радиологический Научный Центр" Министерства Здравоохранения и Социального Развития Российской Федерации (ФГБУ МРНЦ Минздравсоцразвития России) | Противоопухолевое средство |
Also Published As
| Publication number | Publication date |
|---|---|
| GB0404434D0 (en) | 2004-03-31 |
| RU2006134019A (ru) | 2008-04-10 |
| CN1922158A (zh) | 2007-02-28 |
| US20070161618A1 (en) | 2007-07-12 |
| CA2556386A1 (en) | 2005-09-15 |
| US7671078B2 (en) | 2010-03-02 |
| WO2005085219A1 (en) | 2005-09-15 |
| JP2007523941A (ja) | 2007-08-23 |
| KR20060124722A (ko) | 2006-12-05 |
| AU2005219531B2 (en) | 2009-01-15 |
| AU2005219531A1 (en) | 2005-09-15 |
| EP1720845A1 (en) | 2006-11-15 |
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