RU2011111117A - Лечение аутоиммунных заболеваний - Google Patents
Лечение аутоиммунных заболеваний Download PDFInfo
- Publication number
- RU2011111117A RU2011111117A RU2011111117/15A RU2011111117A RU2011111117A RU 2011111117 A RU2011111117 A RU 2011111117A RU 2011111117/15 A RU2011111117/15 A RU 2011111117/15A RU 2011111117 A RU2011111117 A RU 2011111117A RU 2011111117 A RU2011111117 A RU 2011111117A
- Authority
- RU
- Russia
- Prior art keywords
- treatment
- formula
- use according
- guillain
- uveitis
- Prior art date
Links
- 208000023275 Autoimmune disease Diseases 0.000 title 1
- 206010002026 amyotrophic lateral sclerosis Diseases 0.000 claims abstract 10
- 239000003814 drug Substances 0.000 claims abstract 10
- 208000035895 Guillain-Barré syndrome Diseases 0.000 claims abstract 8
- 206010049567 Miller Fisher syndrome Diseases 0.000 claims abstract 8
- 206010046851 Uveitis Diseases 0.000 claims abstract 8
- 150000001875 compounds Chemical class 0.000 claims abstract 8
- 229940079593 drug Drugs 0.000 claims abstract 8
- 238000000034 method Methods 0.000 claims abstract 8
- 150000003839 salts Chemical class 0.000 claims abstract 6
- 125000002467 phosphate group Chemical class [H]OP(=O)(O[H])O[*] 0.000 claims abstract 4
Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
- A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/66—Phosphorus compounds
- A61K31/661—Phosphorus acids or esters thereof not having P—C bonds, e.g. fosfosal, dichlorvos, malathion or mevinphos
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
- A61P21/02—Muscle relaxants, e.g. for tetanus or cramps
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Epidemiology (AREA)
- Immunology (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Emergency Medicine (AREA)
- Pain & Pain Management (AREA)
- Transplantation (AREA)
- Psychiatry (AREA)
- Rheumatology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Hospice & Palliative Care (AREA)
- Ophthalmology & Optometry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
1. Применение соединения формулы Ia ! ! или его фосфатного производного формулы ! ! или их фармацевтически приемлемых солей при приготовлении лекарственного средства для лечения бокового амиотрофического склероза (болезни Лу Герига), синдрома Гийена-Барре и увеита. ! 2. Применение по п.1, в котором указанное соединение представлено соединением формулы Ia ! ! или его фармацевтически приемлемой солью. ! 3. Применение по п.1, в котором указанное лекарственное средство предназначено для лечения увеита. ! 4. Применение по п.1, в котором указанное лекарственное средство предназначено для лечения бокового амиотрофического склероза. ! 5. Применение по п.1, в котором указанное лекарственное средство предназначено для лечения синдрома Гийена-Барре. ! 6. Применение по одному из пп.1, 2 или 3, которое заключается в совместном введении субъекту, одновременно или последовательно, по крайней мере одного второго лекарственного средства. ! 7. Способ лечения бокового амиотрофического склероза, синдрома Гийена-Барре и увеита, который заключается во введении субъекту, нуждающемуся в таком лечении, эффективного количества соединения формулы Ia ! ! или его фосфатного производного формулы ! ! или их фармацевтически приемлемой соли. ! 8. Способ п.7, в котором указанное лечение направлено на увеит. ! 9. Способ п.7, в котором указанное лечение направлено на боковой амиотрофический склероз. ! 10. Способ п.7, в котором указанное лечение направлено на синдром Гийена-Барре.
Claims (10)
3. Применение по п.1, в котором указанное лекарственное средство предназначено для лечения увеита.
4. Применение по п.1, в котором указанное лекарственное средство предназначено для лечения бокового амиотрофического склероза.
5. Применение по п.1, в котором указанное лекарственное средство предназначено для лечения синдрома Гийена-Барре.
6. Применение по одному из пп.1, 2 или 3, которое заключается в совместном введении субъекту, одновременно или последовательно, по крайней мере одного второго лекарственного средства.
8. Способ п.7, в котором указанное лечение направлено на увеит.
9. Способ п.7, в котором указанное лечение направлено на боковой амиотрофический склероз.
10. Способ п.7, в котором указанное лечение направлено на синдром Гийена-Барре.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US71599005P | 2005-09-09 | 2005-09-09 | |
US60/715,990 | 2005-09-09 |
Related Parent Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
RU2008113187/15A Division RU2424795C2 (ru) | 2005-09-09 | 2006-09-07 | Лечение аутоиммунных заболеваний |
Publications (2)
Publication Number | Publication Date |
---|---|
RU2011111117A true RU2011111117A (ru) | 2012-09-27 |
RU2493840C2 RU2493840C2 (ru) | 2013-09-27 |
Family
ID=37056992
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
RU2008113187/15A RU2424795C2 (ru) | 2005-09-09 | 2006-09-07 | Лечение аутоиммунных заболеваний |
RU2011111117/15A RU2493840C2 (ru) | 2005-09-09 | 2006-09-07 | Лечение аутоиммунных заболеваний |
Family Applications Before (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
RU2008113187/15A RU2424795C2 (ru) | 2005-09-09 | 2006-09-07 | Лечение аутоиммунных заболеваний |
Country Status (29)
Country | Link |
---|---|
US (1) | US20080200438A1 (ru) |
EP (2) | EP1926483B1 (ru) |
JP (4) | JP5244598B2 (ru) |
KR (3) | KR101476591B1 (ru) |
CN (1) | CN101257899B (ru) |
AT (1) | ATE489948T1 (ru) |
AU (2) | AU2006289100B2 (ru) |
BR (1) | BRPI0615906A2 (ru) |
CA (2) | CA2620554C (ru) |
CY (1) | CY1111285T1 (ru) |
DE (1) | DE602006018629D1 (ru) |
DK (2) | DK2295049T3 (ru) |
ES (2) | ES2529724T3 (ru) |
HK (1) | HK1149906A1 (ru) |
IL (2) | IL189665A (ru) |
JO (1) | JO2655B1 (ru) |
MA (1) | MA29787B1 (ru) |
MX (1) | MX2008003170A (ru) |
NO (1) | NO20081727L (ru) |
NZ (2) | NZ588372A (ru) |
PL (2) | PL2295049T3 (ru) |
PT (2) | PT2295049E (ru) |
RU (2) | RU2424795C2 (ru) |
SG (1) | SG165364A1 (ru) |
SI (2) | SI1926483T1 (ru) |
TN (1) | TNSN08103A1 (ru) |
TW (2) | TWI372620B (ru) |
WO (1) | WO2007028821A2 (ru) |
ZA (1) | ZA200801694B (ru) |
Families Citing this family (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
PL1772145T3 (pl) * | 2004-07-16 | 2011-08-31 | Kyorin Seiyaku Kk | Sposób skutecznego stosowania leku i sposób dotyczący zapobiegania efektom ubocznym |
KR101181090B1 (ko) | 2004-10-12 | 2012-09-07 | 교린 세이야꾸 가부시키 가이샤 | 2-아미노-2-[2-[4-(3-벤질옥시페닐티오)-2-클로로페닐]에틸]-1,3-프로판디올 염산염 또는 그 수화물의 제조방법 및 그 제조 중간체 |
PT1932522E (pt) * | 2005-10-07 | 2012-06-26 | Kyorin Seiyaku Kk | Agente terapêutico para doenças do fígado contendo, como princípio activo, um derivado de 2- amino-1,3-propanodiol |
TWI389683B (zh) * | 2006-02-06 | 2013-03-21 | Kyorin Seiyaku Kk | A therapeutic agent for an inflammatory bowel disease or an inflammatory bowel disease treatment using a 2-amino-1,3-propanediol derivative as an active ingredient |
NZ574011A (en) * | 2006-08-08 | 2011-10-28 | Kyorin Seiyaku Kk | Aminophosphoric acid ester derivative and s1p receptor modulator containing the same as active ingredient |
MY146775A (en) * | 2006-08-08 | 2012-09-28 | Kyorin Seiyaku Kk | Amino alcohol derivative and immunosuppressive agent having same as an active ingredient |
JP5198293B2 (ja) * | 2007-02-13 | 2013-05-15 | 杏林製薬株式会社 | アミノアルコール誘導体を有効成分とする脱髄性疾患の治療剤又は予防剤 |
TW200946105A (en) | 2008-02-07 | 2009-11-16 | Kyorin Seiyaku Kk | Therapeutic agent or preventive agent for inflammatory bowel disease containing amino alcohol derivative as active ingredient |
RU2505288C2 (ru) * | 2008-05-20 | 2014-01-27 | Киорин Фармасьютикал Ко., Лтд. | Средства поддержания индуцированной ремиссии |
JP5731384B2 (ja) * | 2008-08-18 | 2015-06-10 | ノバルティス アーゲー | 脱髄性末梢ニューロパシーの処置のためのアミノアルコール誘導体 |
CN102917698A (zh) * | 2010-05-06 | 2013-02-06 | 诺瓦提斯公司 | 二芳基硫醚衍生物的给药方案 |
BR112012028190A2 (pt) * | 2010-05-06 | 2016-08-02 | Novartis Ag | tratamento de doenças autoimunes |
Family Cites Families (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5141421A (en) * | 1991-12-17 | 1992-08-25 | Carrier Corporation | Nested coupling mechanism for scroll machines |
DE4428835A1 (de) * | 1994-08-01 | 1996-02-08 | Schering Ag | Neue 3-substituierte 3H-2,3-Benzodiazepinderivate, deren Herstellung und Verwendung als Arzneimittel |
EP0990440B1 (en) * | 1997-02-27 | 2008-10-29 | Novartis AG | Pharmaceutical composition comprising 2-amino-2-[2-(4-octylphenyl)ethyl]propane-1,3-diol, a lecithin and a saccharide |
JP4152884B2 (ja) * | 2001-09-27 | 2008-09-17 | 杏林製薬株式会社 | ジアリールエーテル誘導体とその付加塩及び免疫抑制剤 |
MXPA04002679A (es) * | 2001-09-27 | 2004-07-30 | Kyorin Seiyaku Kk | Derivados de sulfuro de diarilo, sales de los mismos y agentes inmunosupresores que utilizan los mismos. |
CA2498944C (en) * | 2002-09-19 | 2011-05-17 | Yasushi Kohno | Amino alcohol derivatives, salts thereof and immunosuppressive agents |
KR20080103117A (ko) * | 2002-09-24 | 2008-11-26 | 노파르티스 아게 | 탈수초성 장애의 치료에 있어서의 스핑고신-1-포스페이트 수용체 아고니스트 |
KR20050071517A (ko) * | 2002-09-28 | 2005-07-07 | 맥네일-피피씨, 인코포레이티드 | 코어를 2개 갖는 개질된 방출성 투여 제형 |
KR101005171B1 (ko) * | 2003-02-18 | 2011-01-04 | 교린 세이야꾸 가부시키 가이샤 | 아미노포스폰산 유도체와 그 부가염 및 s1p 수용체조절제 |
HUE028247T2 (en) * | 2003-04-08 | 2016-12-28 | Novartis Ag | A solid oral composition comprising S1P receptor agonist and sugar alcohol |
WO2005014525A2 (en) * | 2003-08-12 | 2005-02-17 | Mitsubishi Pharma Corporation | Bi-aryl compound having immunosuppressive activity |
WO2005021503A1 (en) * | 2003-08-28 | 2005-03-10 | Novartis Ag | Aminopropanol derivatives |
PL1772145T3 (pl) * | 2004-07-16 | 2011-08-31 | Kyorin Seiyaku Kk | Sposób skutecznego stosowania leku i sposób dotyczący zapobiegania efektom ubocznym |
JP2008521827A (ja) * | 2004-11-29 | 2008-06-26 | ノバルティス アクチエンゲゼルシャフト | S1p受容体アゴニストの投与レジメン |
GB0504544D0 (en) * | 2005-03-04 | 2005-04-13 | Novartis Ag | Organic compounds |
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2006
- 2006-09-07 KR KR1020147001496A patent/KR101476591B1/ko not_active IP Right Cessation
- 2006-09-07 WO PCT/EP2006/066150 patent/WO2007028821A2/en active Application Filing
- 2006-09-07 JO JO2006298A patent/JO2655B1/en active
- 2006-09-07 ES ES10174280.7T patent/ES2529724T3/es active Active
- 2006-09-07 MX MX2008003170A patent/MX2008003170A/es active IP Right Grant
- 2006-09-07 SI SI200630937T patent/SI1926483T1/sl unknown
- 2006-09-07 SG SG201006580-3A patent/SG165364A1/en unknown
- 2006-09-07 CN CN2006800328984A patent/CN101257899B/zh not_active Expired - Fee Related
- 2006-09-07 ES ES06793341T patent/ES2357426T3/es active Active
- 2006-09-07 BR BRPI0615906-0A patent/BRPI0615906A2/pt not_active IP Right Cessation
- 2006-09-07 PT PT10174280T patent/PT2295049E/pt unknown
- 2006-09-07 CA CA2620554A patent/CA2620554C/en not_active Expired - Fee Related
- 2006-09-07 RU RU2008113187/15A patent/RU2424795C2/ru not_active IP Right Cessation
- 2006-09-07 AT AT06793341T patent/ATE489948T1/de active
- 2006-09-07 DE DE602006018629T patent/DE602006018629D1/de active Active
- 2006-09-07 NZ NZ588372A patent/NZ588372A/en not_active IP Right Cessation
- 2006-09-07 EP EP06793341A patent/EP1926483B1/en active Active
- 2006-09-07 PL PL10174280T patent/PL2295049T3/pl unknown
- 2006-09-07 US US12/065,096 patent/US20080200438A1/en not_active Abandoned
- 2006-09-07 RU RU2011111117/15A patent/RU2493840C2/ru not_active IP Right Cessation
- 2006-09-07 AU AU2006289100A patent/AU2006289100B2/en not_active Ceased
- 2006-09-07 SI SI200631889T patent/SI2295049T1/sl unknown
- 2006-09-07 DK DK10174280.7T patent/DK2295049T3/en active
- 2006-09-07 EP EP10174280.7A patent/EP2295049B1/en active Active
- 2006-09-07 CA CA2820510A patent/CA2820510A1/en not_active Abandoned
- 2006-09-07 PT PT06793341T patent/PT1926483E/pt unknown
- 2006-09-07 PL PL06793341T patent/PL1926483T3/pl unknown
- 2006-09-07 DK DK06793341.6T patent/DK1926483T3/da active
- 2006-09-07 KR KR1020147026128A patent/KR20140117704A/ko not_active Application Discontinuation
- 2006-09-07 JP JP2008529636A patent/JP5244598B2/ja active Active
- 2006-09-07 NZ NZ566137A patent/NZ566137A/en not_active IP Right Cessation
- 2006-09-08 TW TW099117063A patent/TWI372620B/zh not_active IP Right Cessation
- 2006-09-08 TW TW095133326A patent/TWI376223B/zh active
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2008
- 2008-02-21 IL IL189665A patent/IL189665A/en not_active IP Right Cessation
- 2008-02-21 ZA ZA200801694A patent/ZA200801694B/xx unknown
- 2008-03-06 TN TNP2008000103A patent/TNSN08103A1/en unknown
- 2008-03-17 MA MA30758A patent/MA29787B1/fr unknown
- 2008-04-07 NO NO20081727A patent/NO20081727L/no not_active Application Discontinuation
- 2008-04-08 KR KR1020087008413A patent/KR101476451B1/ko not_active IP Right Cessation
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2010
- 2010-09-21 AU AU2010224355A patent/AU2010224355B2/en not_active Ceased
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2011
- 2011-03-01 CY CY20111100242T patent/CY1111285T1/el unknown
- 2011-04-27 HK HK11104200A patent/HK1149906A1/xx unknown
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2012
- 2012-10-17 JP JP2012230044A patent/JP6077265B2/ja not_active Expired - Fee Related
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2014
- 2014-06-23 IL IL233328A patent/IL233328A0/en unknown
- 2014-09-29 JP JP2014199069A patent/JP2015025002A/ja not_active Withdrawn
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2016
- 2016-09-30 JP JP2016193400A patent/JP2017019854A/ja not_active Withdrawn
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