RS56538B1 - (tieno[2,3-b][1,5]benzoksazepin-4-il)piperazin-1-il jedinjenja kao dvostruko delujućih h1 inverzni agonisti/5-ht2a antagonisti - Google Patents
(tieno[2,3-b][1,5]benzoksazepin-4-il)piperazin-1-il jedinjenja kao dvostruko delujućih h1 inverzni agonisti/5-ht2a antagonistiInfo
- Publication number
- RS56538B1 RS56538B1 RS20171134A RSP20171134A RS56538B1 RS 56538 B1 RS56538 B1 RS 56538B1 RS 20171134 A RS20171134 A RS 20171134A RS P20171134 A RSP20171134 A RS P20171134A RS 56538 B1 RS56538 B1 RS 56538B1
- Authority
- RS
- Serbia
- Prior art keywords
- benzoxazepin
- thieno
- piperazin
- compounds
- inverse agonists
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
- Biomedical Technology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Anesthesiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Epidemiology (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201361752203P | 2013-01-14 | 2013-01-14 | |
PCT/US2014/010577 WO2014110065A1 (en) | 2013-01-14 | 2014-01-08 | (THIENO[2,3-b][1,5]BENZOXAZEPIN-4-YL)PIPERAZIN-1-YL COMPOUNDS AS DUAL ACTIVITY H1 INVERSE AGONISTS/5-HT2A ANTAGONISTS |
EP14701636.4A EP2943498B1 (en) | 2013-01-14 | 2014-01-08 | (thieno[2,3-b][1,5]benzoxazepin-4-yl)piperazin-1-yl compounds as dual activity h1 inverse agonists/5-ht2a antagonists |
Publications (1)
Publication Number | Publication Date |
---|---|
RS56538B1 true RS56538B1 (sr) | 2018-02-28 |
Family
ID=50023875
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
RS20171134A RS56538B1 (sr) | 2013-01-14 | 2014-01-08 | (tieno[2,3-b][1,5]benzoksazepin-4-il)piperazin-1-il jedinjenja kao dvostruko delujućih h1 inverzni agonisti/5-ht2a antagonisti |
Country Status (25)
Country | Link |
---|---|
US (1) | US9562057B2 (hu) |
EP (1) | EP2943498B1 (hu) |
JP (1) | JP6100400B2 (hu) |
KR (1) | KR101735458B1 (hu) |
CN (1) | CN104955827B (hu) |
AU (1) | AU2014205616B2 (hu) |
BR (1) | BR112015015491A8 (hu) |
CA (1) | CA2893106C (hu) |
CY (1) | CY1119517T1 (hu) |
DK (1) | DK2943498T3 (hu) |
EA (1) | EA026328B1 (hu) |
ES (1) | ES2647523T3 (hu) |
HR (1) | HRP20171731T1 (hu) |
HU (1) | HUE037363T2 (hu) |
LT (1) | LT2943498T (hu) |
ME (1) | ME02898B (hu) |
MX (1) | MX365594B (hu) |
NO (1) | NO2971205T3 (hu) |
PL (1) | PL2943498T3 (hu) |
PT (1) | PT2943498T (hu) |
RS (1) | RS56538B1 (hu) |
SA (1) | SA515360750B1 (hu) |
SI (1) | SI2943498T1 (hu) |
WO (1) | WO2014110065A1 (hu) |
ZA (1) | ZA201504041B (hu) |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5602124A (en) * | 1994-12-12 | 1997-02-11 | Allelix Biopharmaceuticals, Inc. | 5-HT2 receptor ligands |
HU226410B1 (en) * | 2003-04-22 | 2008-11-28 | Egis Gyogyszergyar Nyilvanosan | Novel polymorphous forms of olanzapine hydrochlorides, process for producing them, use thereof and pharmaceutical compositions containing them |
CA2536107A1 (en) * | 2003-09-09 | 2005-03-24 | Eli Lilly And Company | Substituted piperazines of azepines, oxazepines, and thiazepines |
US7807828B2 (en) * | 2005-08-11 | 2010-10-05 | Hypnion, Inc. | Olanzapine analogs and methods of use thereof |
AR084867A1 (es) * | 2011-02-07 | 2013-07-10 | Lilly Co Eli | Compuestos de acido [(5h-pirrolo[2,1-c][1,4]benzodiazepin-11-il)piperazin-1-il]-2,2-dimetilpropanoico sustituido como antagonistas de 5-ht/agonistas inversos de actividad dual |
AU2012283035B2 (en) * | 2011-07-08 | 2015-07-30 | Eli Lilly & Company | (thieno[2,3-b][1,5]benzoxazepin-4-yl)piperazin-1-yl compounds as dual activity H1 inverse agonists/5-HT2A antagonists |
SI2751115T1 (sl) * | 2011-08-30 | 2017-11-30 | Eli Lilly And Company | SPOJINE (TIENO(2,3-b)(1,5)BENZOKSAZEPIN-4-IL)PIPERAZIN-1-OLA KOT DVOJNO AKTIVNI H1 INVERZNI AGONISTI/5-HT2A ANTAGONISTI |
-
2014
- 2014-01-08 US US14/758,023 patent/US9562057B2/en not_active Expired - Fee Related
- 2014-01-08 BR BR112015015491A patent/BR112015015491A8/pt not_active IP Right Cessation
- 2014-01-08 HU HUE14701636A patent/HUE037363T2/hu unknown
- 2014-01-08 AU AU2014205616A patent/AU2014205616B2/en not_active Ceased
- 2014-01-08 CA CA2893106A patent/CA2893106C/en not_active Expired - Fee Related
- 2014-01-08 PL PL14701636T patent/PL2943498T3/pl unknown
- 2014-01-08 DK DK14701636.4T patent/DK2943498T3/en active
- 2014-01-08 EA EA201591099A patent/EA026328B1/ru not_active IP Right Cessation
- 2014-01-08 LT LTEP14701636.4T patent/LT2943498T/lt unknown
- 2014-01-08 WO PCT/US2014/010577 patent/WO2014110065A1/en active Application Filing
- 2014-01-08 KR KR1020157018420A patent/KR101735458B1/ko active IP Right Grant
- 2014-01-08 MX MX2015008970A patent/MX365594B/es active IP Right Grant
- 2014-01-08 PT PT147016364T patent/PT2943498T/pt unknown
- 2014-01-08 JP JP2015551850A patent/JP6100400B2/ja not_active Expired - Fee Related
- 2014-01-08 SI SI201430378T patent/SI2943498T1/sl unknown
- 2014-01-08 ES ES14701636.4T patent/ES2647523T3/es active Active
- 2014-01-08 EP EP14701636.4A patent/EP2943498B1/en active Active
- 2014-01-08 RS RS20171134A patent/RS56538B1/sr unknown
- 2014-01-08 ME MEP-2017-239A patent/ME02898B/me unknown
- 2014-01-08 CN CN201480004741.5A patent/CN104955827B/zh not_active Expired - Fee Related
- 2014-03-14 NO NO14777943A patent/NO2971205T3/no unknown
-
2015
- 2015-06-05 ZA ZA2015/04041A patent/ZA201504041B/en unknown
- 2015-07-13 SA SA515360750A patent/SA515360750B1/ar unknown
-
2017
- 2017-11-01 CY CY20171101141T patent/CY1119517T1/el unknown
- 2017-11-13 HR HRP20171731TT patent/HRP20171731T1/hr unknown
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