RS55505B1 - Farmaceutska kompozicija koja sadrži ne-nukleozidni inhibitor reverzne transkriptaze - Google Patents

Farmaceutska kompozicija koja sadrži ne-nukleozidni inhibitor reverzne transkriptaze

Info

Publication number
RS55505B1
RS55505B1 RS20161093A RSP20161093A RS55505B1 RS 55505 B1 RS55505 B1 RS 55505B1 RS 20161093 A RS20161093 A RS 20161093A RS P20161093 A RSP20161093 A RS P20161093A RS 55505 B1 RS55505 B1 RS 55505B1
Authority
RS
Serbia
Prior art keywords
pharmaceutical composition
reverse transcriptase
nucleoside reverse
transcriptase inhibitor
nucleoside
Prior art date
Application number
RS20161093A
Other languages
English (en)
Inventor
Jason Burch
Bernard Cote
Original Assignee
Merck Canada Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=44710363&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=RS55505(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Merck Canada Inc filed Critical Merck Canada Inc
Publication of RS55505B1 publication Critical patent/RS55505B1/sr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Virology (AREA)
  • Molecular Biology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • AIDS & HIV (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Saccharide Compounds (AREA)
RS20161093A 2010-03-30 2011-03-28 Farmaceutska kompozicija koja sadrži ne-nukleozidni inhibitor reverzne transkriptaze RS55505B1 (sr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US31882410P 2010-03-30 2010-03-30
US32157310P 2010-04-07 2010-04-07

Publications (1)

Publication Number Publication Date
RS55505B1 true RS55505B1 (sr) 2017-05-31

Family

ID=44710363

Family Applications (2)

Application Number Title Priority Date Filing Date
RS20150340A RS54017B1 (sr) 2010-03-30 2011-03-28 Ne-nukleozidni inhibitori reverzne transkriptaze
RS20161093A RS55505B1 (sr) 2010-03-30 2011-03-28 Farmaceutska kompozicija koja sadrži ne-nukleozidni inhibitor reverzne transkriptaze

Family Applications Before (1)

Application Number Title Priority Date Filing Date
RS20150340A RS54017B1 (sr) 2010-03-30 2011-03-28 Ne-nukleozidni inhibitori reverzne transkriptaze

Country Status (44)

Country Link
US (2) US8486975B2 (sr)
EP (2) EP2552902B1 (sr)
JP (2) JP5281718B2 (sr)
KR (1) KR101421861B1 (sr)
CN (1) CN102971308B (sr)
AR (1) AR080859A1 (sr)
AU (1) AU2011235568B2 (sr)
BR (1) BR112012024691B1 (sr)
CA (1) CA2794377C (sr)
CL (1) CL2012002744A1 (sr)
CO (1) CO6630126A2 (sr)
CR (1) CR20120503A (sr)
CY (3) CY1118774T1 (sr)
DK (2) DK2924034T3 (sr)
DO (1) DOP2012000256A (sr)
EA (1) EA024804B1 (sr)
EC (1) ECSP12012201A (sr)
ES (2) ES2609636T3 (sr)
FI (1) FIC20190021I1 (sr)
GE (1) GEP20156368B (sr)
HK (2) HK1175471A1 (sr)
HN (1) HN2012002039A (sr)
HR (2) HRP20150427T1 (sr)
HU (4) HUE025336T2 (sr)
IL (2) IL222030A (sr)
LT (3) LT2924034T (sr)
LU (1) LUC00114I2 (sr)
MA (1) MA34170B1 (sr)
ME (2) ME02181B (sr)
MX (1) MX2012011379A (sr)
MY (1) MY163979A (sr)
NI (1) NI201200146A (sr)
NL (1) NL300980I2 (sr)
NO (2) NO2019018I1 (sr)
NZ (1) NZ602670A (sr)
PE (1) PE20130158A1 (sr)
PL (2) PL2924034T3 (sr)
PT (2) PT2924034T (sr)
RS (2) RS54017B1 (sr)
SG (1) SG184347A1 (sr)
SI (2) SI2924034T1 (sr)
TN (1) TN2012000455A1 (sr)
TW (1) TWI458719B (sr)
WO (1) WO2011120133A1 (sr)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GEP20156368B (en) * 2010-03-30 2015-09-25 Merck Canada Inc Non-nucleoside reverse transcriptase inhibitors
US20140031250A1 (en) 2010-10-07 2014-01-30 David Tsai Ting Biomarkers of Cancer
MX362517B (es) * 2012-09-26 2019-01-21 Merck Sharp & Dohme Forma cristalina de un inhibidor de transcriptasa inversa.
JO3470B1 (ar) 2012-10-08 2020-07-05 Merck Sharp & Dohme مشتقات 5- فينوكسي-3h-بيريميدين-4-أون واستخدامها كمثبطات ناسخ عكسي ل hiv
EP2928472B1 (en) * 2012-12-05 2018-05-02 Merck Sharp & Dohme Corp. Process for making reverse transcriptase inhibitors
AU2014353177B2 (en) * 2013-11-22 2018-03-15 Merck Sharp & Dohme Llc Composition of a non-nucleoside reverse transcriptase inhibitor
ES2759976T3 (es) 2013-12-04 2020-05-12 Merck Sharp & Dohme Proceso para fabricar inhibidores de la transcriptasa inversa
BR112016022722B8 (pt) * 2014-04-01 2023-11-21 Merck Sharp & Dohme Composto, composição farmacêutica que o comprende e uso do mesmo
US10603282B2 (en) 2015-12-02 2020-03-31 Merck Sharp & Dohme Corp. Pharmaceutical compositions containing doravirine, tenofovir disoproxil fumarate and lamivudine
US11077050B2 (en) 2017-03-24 2021-08-03 Merck Sharp & Dohme Corp. Formulation for parenteral administration
JP2020517633A (ja) 2017-04-18 2020-06-18 シプラ・リミテッド レトロウイルス感染の治療に用いる併用療法
WO2019157087A1 (en) 2018-02-06 2019-08-15 The General Hospital Corporation Repeat rna as biomarkers of tumor immune response
CN110801455B (zh) * 2019-11-12 2020-06-02 河北医科大学第二医院 用于治疗mrsa的药物组合物及其应用
CN114163309B (zh) * 2021-12-27 2023-04-25 甘肃皓天医药科技有限责任公司 一种多拉韦林中间体的制备方法
CN114349690B (zh) * 2022-02-15 2023-04-25 甘肃皓天医药科技有限责任公司 一种多拉韦林中间体合成方法

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE9904045D0 (sv) 1999-11-09 1999-11-09 Astra Ab Compounds
TW200423930A (en) * 2003-02-18 2004-11-16 Hoffmann La Roche Non-nucleoside reverse transcriptase inhibitors
RU2344128C2 (ru) 2003-03-24 2009-01-20 Ф.Хоффманн-Ля Рош Аг Бензилпиридазиноны как ингибиторы обратной транскриптазы
TW200505441A (en) 2003-03-24 2005-02-16 Hoffmann La Roche Non-nucleoside reverse transcriptase inhibitorsⅠ
WO2005102989A1 (en) 2004-04-23 2005-11-03 F. Hoffmann-La Roche Ag Non-nucleoside reverse transcriptase inhibitors
US7166738B2 (en) 2004-04-23 2007-01-23 Roche Palo Alto Llc Non-nucleoside reverse transcriptase inhibitors
JP2008525419A (ja) 2004-12-22 2008-07-17 ファイザー・リミテッド Hiv−1逆転写酵素の非ヌクレオシド阻害剤
AR057455A1 (es) 2005-07-22 2007-12-05 Merck & Co Inc Inhibidores de la transcriptasa reversa de vih y composicion farmaceutica
BRPI0617482A2 (pt) 2005-10-19 2011-07-26 Hoffmann La Roche compostos inibidores de transcriptase reversa nço-nucleosÍdeos de n-fenil fenilacetamida, composiÇço farmacÊutica contendo os referidos compostos bem como seus usos
WO2007045573A1 (en) 2005-10-19 2007-04-26 F. Hoffmann-La Roche Ag Phenyl-acetamide nnrt inhibitors
TW200831085A (en) 2006-12-13 2008-08-01 Merck & Co Inc Non-nucleoside reverse transcriptase inhibitors
WO2009067166A2 (en) * 2007-11-20 2009-05-28 Merck & Co., Inc. Non-nucleoside reverse transcriptase inhibitors
GEP20156368B (en) * 2010-03-30 2015-09-25 Merck Canada Inc Non-nucleoside reverse transcriptase inhibitors

Also Published As

Publication number Publication date
HK1175471A1 (en) 2013-07-05
CY2019025I1 (el) 2019-11-27
CY2019026I2 (el) 2020-05-29
IL233334A0 (en) 2014-09-01
FIC20190021I1 (fi) 2019-04-17
CY2019025I2 (el) 2019-11-27
CR20120503A (es) 2013-01-09
DOP2012000256A (es) 2012-12-15
GEP20156368B (en) 2015-09-25
LT2924034T (lt) 2016-12-27
JP5281718B2 (ja) 2013-09-04
SI2552902T1 (sl) 2015-10-30
ES2536295T3 (es) 2015-05-22
PL2552902T3 (pl) 2015-10-30
MX2012011379A (es) 2012-11-30
PE20130158A1 (es) 2013-02-28
NO2019019I1 (no) 2019-04-24
AR080859A1 (es) 2012-05-16
CA2794377C (en) 2015-06-16
CN102971308B (zh) 2015-02-04
HRP20150427T1 (hr) 2015-07-03
SG184347A1 (en) 2012-11-29
DK2552902T3 (en) 2015-06-15
EP2552902A4 (en) 2013-09-04
CY1118774T1 (el) 2017-07-12
JP2013209405A (ja) 2013-10-10
JP5886790B2 (ja) 2016-03-16
WO2011120133A1 (en) 2011-10-06
US8486975B2 (en) 2013-07-16
HN2012002039A (es) 2015-08-24
LTC2552902I2 (lt) 2019-12-10
LUC00114I1 (sr) 2019-04-17
NL300980I1 (nl) 2019-04-24
TWI458719B (zh) 2014-11-01
EP2924034A1 (en) 2015-09-30
CA2794377A1 (en) 2011-10-06
PL2924034T3 (pl) 2017-07-31
IL233334A (en) 2015-09-24
EA201290976A1 (ru) 2013-03-29
ME02181B (me) 2015-10-20
ME02570B (me) 2017-06-20
US20130296382A1 (en) 2013-11-07
SI2924034T1 (sl) 2017-05-31
MA34170B1 (fr) 2013-04-03
DK2924034T3 (en) 2017-02-06
NI201200146A (es) 2013-03-18
LTPA2019507I1 (lt) 2019-04-25
HUE031785T2 (en) 2017-08-28
US20110245296A1 (en) 2011-10-06
PT2552902E (pt) 2015-06-02
LUC00114I2 (sr) 2020-07-10
EP2924034B1 (en) 2016-11-02
AU2011235568A1 (en) 2012-11-01
ECSP12012201A (es) 2012-10-30
BR112012024691B1 (pt) 2020-11-17
RS54017B1 (sr) 2015-10-30
NL300980I2 (nl) 2021-06-17
HRP20161680T1 (hr) 2017-01-27
CY2019026I1 (el) 2020-05-29
BR112012024691A2 (pt) 2019-07-02
CL2012002744A1 (es) 2012-12-14
HUE025336T2 (en) 2016-03-29
EA024804B1 (ru) 2016-10-31
EP2552902A1 (en) 2013-02-06
HK1209121A1 (en) 2016-03-24
IL222030A (en) 2014-07-31
NO2019018I1 (no) 2019-04-24
HUS1900021I1 (hu) 2019-05-28
HUS1900022I1 (hu) 2019-05-28
TW201139409A (en) 2011-11-16
EP2552902B1 (en) 2015-03-11
TN2012000455A1 (en) 2014-01-30
KR101421861B1 (ko) 2014-07-22
AU2011235568B2 (en) 2013-09-12
PT2924034T (pt) 2017-01-06
CO6630126A2 (es) 2013-03-01
KR20120128703A (ko) 2012-11-27
CN102971308A (zh) 2013-03-13
ES2609636T3 (es) 2017-04-21
JP2013510800A (ja) 2013-03-28
LTC2924034I2 (lt) 2020-10-12
MY163979A (en) 2017-11-15
LTPA2019506I1 (lt) 2019-04-25
NZ602670A (en) 2014-09-26

Similar Documents

Publication Publication Date Title
HUS1900022I1 (hu) Gyógyszerészeti kompozíció, amely tartalmaz nem nukleozid reverz transzkriptáz inhibitort
EP2604688A4 (en) VARIANTE REVERSE TRANSKRIPTASE
IL220863A (en) Oxazole derivatives of kinase inhibitors, medicinal preparations containing them and their uses
EP2217069A4 (en) INHIBITORS OF NON-NUCLEOSIDE INHIBITORS OF THE REVERSE TRANSCRIPTASE
HUE031336T2 (hu) Gyógyszerészeti készítmények
IL205386A0 (en) Non - nucleoside reverse transcriptase inhibitors
ZA201208726B (en) High-temperature stable oxygen-carrier-containing pharmaceutical composition
BR112013013571A2 (pt) comprimido para a desintegração oral
ZA201304633B (en) A pharmaceutical composition
ZA201101850B (en) Composition having a sirtuin activator
IL200886A0 (en) Non-nucleoside reverse transcriptase inhibitors
HUE051133T2 (hu) Gyógyászati készítmények
ZA201207797B (en) Injectable formulation of a reverse transcriptase inhibitor for the treatment cancer
IL202143A0 (en) Non-nucleoside reverse transcriptase inhibitors
EP2560678A4 (en) PHARMACEUTICAL COMPOSITIONS
ZA201201003B (en) A pharmaceutical composition
IL226378A0 (en) preparations@rokkhot
GB201008590D0 (en) Pharmaceutical compositions