RS53152B - Novi antibakterijski agensi za lečenje gram pozitivnih infekcija - Google Patents

Novi antibakterijski agensi za lečenje gram pozitivnih infekcija

Info

Publication number
RS53152B
RS53152B RS20140021A RSP20140021A RS53152B RS 53152 B RS53152 B RS 53152B RS 20140021 A RS20140021 A RS 20140021A RS P20140021 A RSP20140021 A RS P20140021A RS 53152 B RS53152 B RS 53152B
Authority
RS
Serbia
Prior art keywords
compounds
compound
pharmaceutical composition
acid
formula
Prior art date
Application number
RS20140021A
Other languages
English (en)
Serbian (sr)
Inventor
Andre Lee Pearson
Chester A. Metcalf Iii
Jing Li
Original Assignee
Cubist Pharmaceuticals Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Cubist Pharmaceuticals Inc. filed Critical Cubist Pharmaceuticals Inc.
Publication of RS53152B publication Critical patent/RS53152B/sr

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/02Peptides of undefined number of amino acids; Derivatives thereof
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/50Cyclic peptides containing at least one abnormal peptide link
    • C07K7/54Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/04Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/12Cyclic peptides, e.g. bacitracins; Polymyxins; Gramicidins S, C; Tyrocidins A, B or C
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/04Immunostimulants
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04Linear peptides containing only normal peptide links
    • C07K7/08Linear peptides containing only normal peptide links having 12 to 20 amino acids
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/50Cyclic peptides containing at least one abnormal peptide link
    • C07K7/54Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring
    • C07K7/60Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring the cyclisation occurring through the 4-amino group of 2,4-diamino-butanoic acid
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/64Cyclic peptides containing only normal peptide links
    • C07K7/645Cyclosporins; Related peptides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Immunology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
RS20140021A 2008-12-22 2009-12-18 Novi antibakterijski agensi za lečenje gram pozitivnih infekcija RS53152B (sr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US13987508P 2008-12-22 2008-12-22
PCT/US2009/068747 WO2010075215A1 (en) 2008-12-22 2009-12-18 Novel antibacterial agents for the treatment of gram positive infections

Publications (1)

Publication Number Publication Date
RS53152B true RS53152B (sr) 2014-06-30

Family

ID=41718893

Family Applications (1)

Application Number Title Priority Date Filing Date
RS20140021A RS53152B (sr) 2008-12-22 2009-12-18 Novi antibakterijski agensi za lečenje gram pozitivnih infekcija

Country Status (26)

Country Link
US (3) US8507647B2 (https=)
EP (2) EP2674437A1 (https=)
JP (1) JP5670914B2 (https=)
KR (1) KR101717795B1 (https=)
CN (1) CN102325787B (https=)
AR (1) AR074833A1 (https=)
AU (1) AU2009330245C1 (https=)
BR (1) BRPI0923567A2 (https=)
CA (1) CA2747965C (https=)
CY (1) CY1114883T1 (https=)
DK (1) DK2379580T3 (https=)
ES (1) ES2442167T3 (https=)
HR (1) HRP20131170T1 (https=)
IL (1) IL213638A0 (https=)
MX (1) MX2011006803A (https=)
NZ (1) NZ594019A (https=)
PL (1) PL2379580T3 (https=)
PT (1) PT2379580E (https=)
RS (1) RS53152B (https=)
RU (1) RU2512396C2 (https=)
SG (1) SG172299A1 (https=)
SI (1) SI2379580T1 (https=)
SM (1) SMT201400037B (https=)
TW (1) TWI444198B (https=)
WO (1) WO2010075215A1 (https=)
ZA (1) ZA201104693B (https=)

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MX2013013760A (es) * 2011-05-26 2014-01-08 Cubist Pharm Inc Composiciones de cb-183, 315 y metodos relacionados.
US10377699B2 (en) * 2013-11-06 2019-08-13 The University Of Hong Kong Daptomycin analogues and a method for the preparation of daptomycin or a daptomycin analogue
WO2015172047A1 (en) * 2014-05-08 2015-11-12 Merck Sharp & Dohme Corp. Cyclic peptide compounds and related methods, salts and compositions
US11667674B2 (en) 2016-04-08 2023-06-06 Versitech Limited Antibacterial cyclic lipopeptides
US10647746B2 (en) 2016-04-08 2020-05-12 Versitech Limited Antibacterial cyclic lipopeptides
PT3445767T (pt) * 2016-04-22 2020-05-13 Astrazeneca Ab Inibidores de mcl-1 macrocíclicos para o tratamento de cancro
US10098890B2 (en) 2016-10-29 2018-10-16 Cipla Limited Stable carfilzomib formulations
IT201600127655A1 (it) 2016-12-16 2018-06-16 Gnosis Spa Processo per la purificazione di antibiotici lipopolipeptidici
US10072045B1 (en) 2017-06-26 2018-09-11 Ramapo Pharmaceuticals, Inc. Antibacterial lipopeptides and methods for their preparation and use
US10526343B2 (en) 2018-03-26 2020-01-07 University Of Sharjah Heterocyclic systems and pharmaceutical applications thereof
RU2762182C1 (ru) * 2020-12-08 2021-12-16 Федеральное государственное бюджетное научное учреждение "Научно-исследовательский институт по изысканию новых антибиотиков имени Г.Ф. Гаузе" Гауземицины А и В - гликолипопептидные антибактериальные антибиотики и способ их получения

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Also Published As

Publication number Publication date
TW201028161A (en) 2010-08-01
DK2379580T3 (da) 2014-01-20
JP2012513467A (ja) 2012-06-14
PT2379580E (pt) 2014-01-20
AU2009330245C1 (en) 2013-09-26
US20150337013A1 (en) 2015-11-26
MX2011006803A (es) 2011-09-06
BRPI0923567A2 (pt) 2016-09-27
US8507647B2 (en) 2013-08-13
HRP20131170T1 (hr) 2014-01-03
EP2674437A1 (en) 2013-12-18
SMT201400037B (it) 2014-05-07
ZA201104693B (en) 2013-01-30
US20100184649A1 (en) 2010-07-22
KR20110114592A (ko) 2011-10-19
SI2379580T1 (sl) 2014-02-28
RU2512396C2 (ru) 2014-04-10
CN102325787A (zh) 2012-01-18
ES2442167T3 (es) 2014-02-10
HK1161886A1 (en) 2012-08-10
EP2379580B1 (en) 2013-10-23
CA2747965A1 (en) 2010-07-01
CA2747965C (en) 2017-06-27
WO2010075215A1 (en) 2010-07-01
CY1114883T1 (el) 2016-12-14
NZ594019A (en) 2013-08-30
IL213638A0 (en) 2011-07-31
US20140073558A1 (en) 2014-03-13
TWI444198B (zh) 2014-07-11
JP5670914B2 (ja) 2015-02-18
SG172299A1 (en) 2011-07-28
CN102325787B (zh) 2014-05-28
AU2009330245B2 (en) 2013-05-02
RU2011130278A (ru) 2013-01-27
KR101717795B1 (ko) 2017-03-17
AR074833A1 (es) 2011-02-16
AU2009330245A1 (en) 2011-08-04
PL2379580T3 (pl) 2014-05-30
EP2379580A1 (en) 2011-10-26

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