RS52304B - SUBSTITUTED INDOLYL ALKYL AMINO DERIVATIVES AS NEW HISTON DEACETYLASE INHIBITORS - Google Patents

SUBSTITUTED INDOLYL ALKYL AMINO DERIVATIVES AS NEW HISTON DEACETYLASE INHIBITORS

Info

Publication number
RS52304B
RS52304B RS20120165A RSP20120165A RS52304B RS 52304 B RS52304 B RS 52304B RS 20120165 A RS20120165 A RS 20120165A RS P20120165 A RSP20120165 A RS P20120165A RS 52304 B RS52304 B RS 52304B
Authority
RS
Serbia
Prior art keywords
alkyl
hydrogen
6alkyl
amino
alkyl amino
Prior art date
Application number
RS20120165A
Other languages
English (en)
Serbian (sr)
Inventor
Marc Gustaaf C. Verdonck
Patrick René ANGIBAUD
Bruno Roux
Isabelle Noëlle Constance PILATTE
Peter Ten Holte
Janine Arts
Kristof Van Emelen
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Priority claimed from PCT/EP2005/053612 external-priority patent/WO2006010750A1/en
Publication of RS52304B publication Critical patent/RS52304B/en

Links

Landscapes

  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
RS20120165A 2004-07-28 2005-07-25 SUBSTITUTED INDOLYL ALKYL AMINO DERIVATIVES AS NEW HISTON DEACETYLASE INHIBITORS RS52304B (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP04077172 2004-07-28
US59218204P 2004-07-29 2004-07-29
PCT/EP2005/053612 WO2006010750A1 (en) 2004-07-28 2005-07-25 Substituted indolyl alkyl amino derivatives as novel inhibitors of histone deacetylase

Publications (1)

Publication Number Publication Date
RS52304B true RS52304B (en) 2012-12-31

Family

ID=34928411

Family Applications (1)

Application Number Title Priority Date Filing Date
RS20120165A RS52304B (en) 2004-07-28 2005-07-25 SUBSTITUTED INDOLYL ALKYL AMINO DERIVATIVES AS NEW HISTON DEACETYLASE INHIBITORS

Country Status (10)

Country Link
CN (1) CN1993353B (me)
AT (1) ATE542812T1 (me)
DK (1) DK1781639T3 (me)
ES (1) ES2381117T3 (me)
ME (1) ME01444B (me)
PT (1) PT1781639E (me)
RS (1) RS52304B (me)
SI (1) SI1781639T1 (me)
UA (1) UA93352C2 (me)
ZA (1) ZA200700764B (me)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN107095871A (zh) * 2016-02-22 2017-08-29 中国科学院上海巴斯德研究所 Quisinostat,一种新型的高效抗疟药物
CN107721980B (zh) * 2017-08-25 2019-07-12 南京医科大学 一类氟尿嘧啶和Quisinosta的乏氧靶向前药及其应用
CN112485233B (zh) * 2020-11-03 2022-08-26 山东师范大学 一种检测去乙酰化酶用纳米传感器及其检测方法和应用

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE60321548D1 (de) * 2002-03-13 2008-07-24 Janssen Pharmaceutica Nv Carbonylamino- derivativate als neue inhibitoren von histone deacetylase

Also Published As

Publication number Publication date
UA93352C2 (ru) 2011-02-10
DK1781639T3 (da) 2012-05-14
PT1781639E (pt) 2012-05-02
SI1781639T1 (sl) 2012-06-29
ME01444B (me) 2013-12-20
ZA200700764B (en) 2008-09-25
ES2381117T3 (es) 2012-05-23
ATE542812T1 (de) 2012-02-15
CN1993353A (zh) 2007-07-04
CN1993353B (zh) 2010-12-01

Similar Documents

Publication Publication Date Title
HRP20090162T1 (en) Quinolinone-carboxamide compounds as 5-ht4 receptor agonists
CO5200848A1 (es) Derivados de 3(5)-ureido-pirazol, proceso para su prepa- racion y su utilizacion como agentes antitumorales
CY1107221T1 (el) Παραγωγα τριαζολιου ως ανταγωνιστες υποδοχεα ταχυκινινης
RS53627B1 (en) N- (3-Amino-quinoxalin-2-yl) -sulfonamide derivatives and their use as phosphatidylinositol 3-kinase inhibitors
MEP61208A (en) Novel compounds having inhibitory activity against sodium-dependant transporter
AR057023A1 (es) Compuestos heterociclicos con propiedades inhibidoras de hiv-integrasa
ATE404536T1 (de) Substituierte chinolinderivate als inhibitoren von mitotischem kinesin
AR060545A1 (es) Compuestos de benzoaxol y benzotiazol 6-0- sustituidos y metodos de inhibicion de la senalizacion de csf-1r. composiciones farmaceuticas
AR054799A1 (es) Derivados de oxindol
NO20091889L (no) Inhibitorer av spiroketon acetyl-CoA karboksylase
CO5640098A2 (es) Acidos biariloximetilaren-carboxilicos
RS52261B (en) AMIDOPHENOX INDASOLS AS A USEFUL C-MET INHIBITOR
CL2004000655A1 (es) Compuestos derivados de piperidin-2-ona 1,6-disustituidos, sus sales, composicion farmaceutica, agonistas del receptor ep4; uso de los compuestos para tratar hipertension ocular, glaucoma.
AR055959A1 (es) Derivados espiro para la modulacion de actividad de crth2
DE602006011752D1 (de) Als antikoagulationsmittel geeignete phenylglycinamid- und pyridylglycinamidderivate
EA200900924A1 (ru) Циклизованные производные как ингибиторы eg-5
CR11483A (es) Inhibidores de peptido desformilasa
RS51674B (en) PIPERIDIN-4-IL-PIRIDAZIN-3-ILAMINE DERIVATIVES AS A FAST DISSOCATING DOPAMIN 2 RECEIVER ANTAGONISTS
EA201000101A1 (ru) Производные пиримидина 934
RS51226B (sr) Derivati azapeptida kao inhibitori hiv proteaze
RS51193B (sr) Hidantoinski derivati korisni kao inhibitori metaloproteinaza
DK1485377T5 (da) Pyranoner egnede som ATM-inhibitorer
ATE409179T1 (de) Tetralin- und indanderivate und deren anwendungen als 5-ht-antagonisten
EA200401455A1 (ru) Производные бензоксазина в качестве модуляторов 5-htи их применение
RS52518B (en) 4-ALCOXYPYRIDASINE DERIVATIVES AS A FAST DISSOCATING DOPAMINE 2 RECEPTOR ANTAGONISTS