RS50642B - Derivati triazolopiridinilsulfanila kao inhibitori p38 map kinaze - Google Patents

Derivati triazolopiridinilsulfanila kao inhibitori p38 map kinaze

Info

Publication number
RS50642B
RS50642B RSP-2008/0599A RSP20080599A RS50642B RS 50642 B RS50642 B RS 50642B RS P20080599 A RSP20080599 A RS P20080599A RS 50642 B RS50642 B RS 50642B
Authority
RS
Serbia
Prior art keywords
independently selected
optionally substituted
halo
alkyl
conr5r6
Prior art date
Application number
RSP-2008/0599A
Other languages
English (en)
Inventor
John Paul Mathias
David Simon Millan
Russell Andrew Lewthwaite
Christopher Phillips
Original Assignee
Pfizer Inc.
Pfizer Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Inc., Pfizer Limited filed Critical Pfizer Inc.
Priority claimed from PCT/IB2005/002574 external-priority patent/WO2006018718A2/en
Publication of RS50642B publication Critical patent/RS50642B/sr

Links

RSP-2008/0599A 2004-08-12 2005-08-09 Derivati triazolopiridinilsulfanila kao inhibitori p38 map kinaze RS50642B (sr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB0418015A GB0418015D0 (en) 2004-08-12 2004-08-12 New compounds
US69155905P 2005-06-17 2005-06-17
PCT/IB2005/002574 WO2006018718A2 (en) 2004-08-12 2005-08-09 Triazolopyridinylsulfanyl derivatives as p38 map kinase inhibitors

Publications (1)

Publication Number Publication Date
RS50642B true RS50642B (sr) 2010-06-30

Family

ID=33017410

Family Applications (1)

Application Number Title Priority Date Filing Date
RSP-2008/0599A RS50642B (sr) 2004-08-12 2005-08-09 Derivati triazolopiridinilsulfanila kao inhibitori p38 map kinaze

Country Status (9)

Country Link
CN (1) CN101006087B (sr)
GB (1) GB0418015D0 (sr)
ME (1) ME01360B (sr)
NI (1) NI200700039A (sr)
PE (1) PE20060618A1 (sr)
RS (1) RS50642B (sr)
TW (1) TWI295926B (sr)
UA (1) UA93032C2 (sr)
ZA (1) ZA200700923B (sr)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20130087048A (ko) * 2008-02-04 2013-08-05 화이자 리미티드 염증성 질환을 치료하기 위한 [1,2,4]트라이아졸로[4,3-a]피리딘 유도체의 다형체 형태
MX2011008496A (es) * 2009-02-17 2011-11-18 Chiesi Farma Spa Derivados de triazolopiridina como inhibidores de proteinas cinasas activadas por mitogeno p38 (map).
GB201009731D0 (en) * 2010-06-10 2010-07-21 Pulmagen Therapeutics Inflamma Kinase inhibitors
CN105968110B (zh) * 2011-12-09 2018-04-27 奇斯药制品公司 激酶抑制剂
CN105646484A (zh) * 2016-03-01 2016-06-08 孙霖 晶型b及制备方法
CN105693716A (zh) * 2016-03-01 2016-06-22 孙霖 晶型a及制备方法

Also Published As

Publication number Publication date
NI200700039A (es) 2008-03-07
ZA200700923B (en) 2008-09-25
UA93032C2 (uk) 2011-01-10
CN101006087B (zh) 2010-09-29
TWI295926B (en) 2008-04-21
CN101006087A (zh) 2007-07-25
TW200610529A (en) 2006-04-01
ME01360B (me) 2010-06-30
PE20060618A1 (es) 2006-07-14
GB0418015D0 (en) 2004-09-15

Similar Documents

Publication Publication Date Title
HRP20080608T3 (en) Triazolopyridinylsulfanyl derivatives as p38 map kinase inhibitors
RS52166B (sr) Amino-heterociklična jedinjenja
AR060316A1 (es) Azaindoles de utilidad como inhibidores de janus quinasas
RS50642B (sr) Derivati triazolopiridinilsulfanila kao inhibitori p38 map kinaze
CY1110232T1 (el) Παραγωγα 2-αρυλ-6-φαινυλ-ιμιδαζο[1,2-α]πυριδιν, η παρασκευη τους και η εφαρμογη τους στη θεραπευτικη αγωγη
NO20061456L (no) Use of CRTH2 antagonist compounds in therapy
HRP20080477T3 (en) Aryl-pyridine derivatives as 11-beta-hsd1 inhibitors
RS53342B (sr) Derivati tieno-piridina kao inhibitori mek
WO2005070910A3 (fr) Derives de 1 -piperazine- et 1-homopiperazine-carboxylates, leur preparation et leur application en tant qu’ inhibiteurs de l’enzyme faah
MY189118A (en) Pyrazolo[1,5-a]pyrazin-4-yl derivatives
ATE442356T1 (de) 1-essigsäureindolderivate mit pgd2- antagonistischer wirkung
RS52702B (sr) Jedinjenja karbazola i terapeutske upotrebe jedinjenja
AR091022A1 (es) Inhibidores del nampt
HRP20020317B1 (en) Pharmaceutically active compounds
MX344276B (es) Compuesto de piperidina novedoso o sal del mismo.
HRP20080311T3 (en) Pyrazole derivatives, compositions containing such compounds and methods of use
AR067599A1 (es) Derivados de indazol sustituido activos como inhibidores de quinasa
RS52964B (sr) Derivat 7-piperidinoalkil-3,4-dihidrokvinolona
EP1867649A4 (en) PIPERIDYL-2,6-DION DERIVATIVES USED TO INHIBIT THE RELEASE OF TUMOR NECROSIS FACTOR FROM CELLS
ATE556058T1 (de) 1-(2h)-isochinolonderivat
HRP20050682B1 (hr) Derivati pirazolopiridina
RS52326B (sr) Fenil-piperazin derivati kao inhibitori resorbcije serotonina
CO5550450A2 (es) Derivados de 1-acil-pirrolidina para el tratamiento de infec ciones virales
EA201000413A1 (ru) Способ получения производных лактамида, новые производные лактамида и препараты, содержащие производные лактамида
RS52949B (sr) Adicione soli amina koji sadrže hidroksilne i/ili karboksilne grupe s derivatima aminonikotinske kiseline kao dhodh inhibitorima