RO94159B1 - Procedeu pentru prepararea unor derivati de pirazolsulfonamida - Google Patents

Procedeu pentru prepararea unor derivati de pirazolsulfonamida

Info

Publication number
RO94159B1
RO94159B1 RO121895A RO12189586A RO94159B1 RO 94159 B1 RO94159 B1 RO 94159B1 RO 121895 A RO121895 A RO 121895A RO 12189586 A RO12189586 A RO 12189586A RO 94159 B1 RO94159 B1 RO 94159B1
Authority
RO
Romania
Prior art keywords
page
derivatives
description
preparation
general formula
Prior art date
Application number
RO121895A
Other languages
English (en)
Other versions
RO94159A2 (ro
Inventor
Susumu Yamamoto
Takuya Kakuta
Toshiaki Sato
Morimoto Katsushi
Oyo Eiichi
Ikai Takasi
Tsutomu Nawamaki
Original Assignee
Nissan Chemical Industries
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Nissan Chemical Industries filed Critical Nissan Chemical Industries
Publication of RO94159A2 publication Critical patent/RO94159A2/ro
Publication of RO94159B1 publication Critical patent/RO94159B1/ro

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D521/00—Heterocyclic compounds containing unspecified hetero rings
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/28—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N<
    • A01N47/36—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N< containing the group >N—CO—N< directly attached to at least one heterocyclic ring; Thio analogues thereof
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/40—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having a double or triple bond to nitrogen, e.g. cyanates, cyanamides
    • A01N47/42—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having a double or triple bond to nitrogen, e.g. cyanates, cyanamides containing —N=CX2 groups, e.g. isothiourea
    • A01N47/44—Guanidine; Derivatives thereof

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Environmental Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

Abstract

Inventia se refera la un procedeu pentru prepararea unor derivati de pirozolsulfonamida cu formula generala I (vezi formula în pag.1 a descrierii) în care A, B, D, X, Y si Z au diferite semnificatii, prin tratarea unui derivat de pirazolsulfonil izocianat cu formula generala II (vezi formula în pag.1 a descrierii) cu un derivat de aminopirimidina cu formula generala III (vezi formula în pag.1 a descrierii) în mediu de solvent organic ales dintre toluen, dioxan si acetonitril, la temperatura de reflux, eventual în prezenta unui acceptor de acizi ales dintre trietilamina, trietilendiamina, piridina, alcoxid de sodiu sau hidrura de sodiu.
RO121895A 1985-01-18 1986-01-17 Procedeu pentru prepararea unor derivati de pirazolsulfonamida RO94159B1 (ro)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP680085 1985-01-18
JP7878485 1985-04-13
JP23678085 1985-10-22

Publications (2)

Publication Number Publication Date
RO94159A2 RO94159A2 (ro) 1988-03-30
RO94159B1 true RO94159B1 (ro) 1988-03-31

Family

ID=27277351

Family Applications (1)

Application Number Title Priority Date Filing Date
RO121895A RO94159B1 (ro) 1985-01-18 1986-01-17 Procedeu pentru prepararea unor derivati de pirazolsulfonamida

Country Status (18)

Country Link
US (1) US4881965A (ro)
EP (2) EP0318602B1 (ro)
CN (1) CN86100911A (ro)
AT (1) ATE88703T1 (ro)
AU (1) AU595176B2 (ro)
BR (1) BR8600183A (ro)
DE (1) DE3688374T2 (ro)
DK (1) DK25386A (ro)
ES (1) ES8706324A1 (ro)
FI (1) FI855180A7 (ro)
GR (1) GR860049B (ro)
HU (1) HU200596B (ro)
IN (1) IN165281B (ro)
PL (1) PL151526B1 (ro)
RO (1) RO94159B1 (ro)
SU (1) SU1701104A3 (ro)
TR (1) TR22668A (ro)
YU (1) YU45761B (ro)

Families Citing this family (28)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4690705A (en) * 1984-11-30 1987-09-01 E. I. Du Pont De Nemours And Company Herbicidal sulfonamides
GB8820115D0 (en) * 1988-08-24 1988-09-28 Ici Plc Insecticidal compounds
JP3231429B2 (ja) * 1992-11-06 2001-11-19 株式会社日立製作所 中央処理装置と乗算器とを有する半導体集積回路装置
EP0837632B1 (en) 1995-07-11 1999-09-22 Novartis AG Selective herbicidal composition
BR0108908A (pt) * 2000-03-03 2002-12-24 Pfizer Prod Inc Derivados de éteres de pirazol como agentes antiinflamatórios/analgésicos
EP2052606A1 (de) 2007-10-24 2009-04-29 Bayer CropScience AG Herbizid-Kombination
DE102008037620A1 (de) 2008-08-14 2010-02-18 Bayer Crop Science Ag Herbizid-Kombination mit Dimethoxytriazinyl-substituierten Difluormethansulfonylaniliden
JP5756457B2 (ja) * 2009-04-06 2015-07-29 アジオス ファーマシューティカルズ， インコーポレイテッド ピルビン酸キナーゼｍ２調節剤、治療組成物および関連する使用方法
CA2944788C (en) 2009-06-29 2023-08-22 Agios Pharmaceuticals, Inc. Compounds, and compositions thereof, which modulate pyruvate kinase m2, and methods of making same
DK2448581T3 (en) 2009-06-29 2017-03-13 Agios Pharmaceuticals Inc Therapeutic compositions and methods for their applications
CN101940217A (zh) * 2010-09-13 2011-01-12 尹小根 含有唑嘧磺隆的除草组合物
MX2013006900A (es) 2010-12-17 2013-10-17 Agios Pharmaceuticals Inc Nuevos derivados n-(4-(azetidina-1-carbonil)fenil)-(hetero-)arilsu lfonamida como moduladores piruvato quinasa m2 (pmk2).
US9328077B2 (en) 2010-12-21 2016-05-03 Agios Pharmaceuticals, Inc Bicyclic PKM2 activators
TWI549947B (zh) 2010-12-29 2016-09-21 阿吉歐斯製藥公司 治療化合物及組成物
WO2012151440A1 (en) 2011-05-03 2012-11-08 Agios Pharmaceuticals, Inc. Pyruvate kinase activators for use for increasing lifetime of the red blood cells and treating anemia
CN103764147B (zh) 2011-05-03 2018-05-22 安吉奥斯医药品有限公司 用于治疗的丙酮酸激酶活化剂
EP2928471B1 (en) 2012-12-06 2020-10-14 Celgene Quanticel Research, Inc. Histone demethylase inhibitors
WO2014139144A1 (en) 2013-03-15 2014-09-18 Agios Pharmaceuticals, Inc. Therapeutic compounds and compositions
PE20221627A1 (es) 2015-02-16 2022-10-19 Univ Queensland Sulfonilureas y compuestos relacionados y uso de estos
PT3307271T (pt) 2015-06-11 2023-10-10 Agios Pharmaceuticals Inc Métodos de utilização de ativadores da piruvato-cinase
AU2017416068A1 (en) 2017-05-24 2019-10-31 The Provost, Fellows, Foundation Scholars, And Other Members Of Board, Of The College Of The Holy And Undivided Trinity Of Queen Elizabeth Near Dublin Novel compounds and uses
PE20212077A1 (es) 2017-07-07 2021-10-28 Inflazome Ltd Nuevos compuestos sulfonamida de carboxamida
EP3668842A1 (en) 2017-08-15 2020-06-24 Inflazome Limited Sulfonylureas and sulfonylthioureas as nlrp3 inhibitors
US11926600B2 (en) 2017-08-15 2024-03-12 Inflazome Limited Sulfonylureas and sulfonylthioureas as NLRP3 inhibitors
TW201910316A (zh) 2017-08-15 2019-03-16 愛爾蘭商英弗雷佐姆有限公司 新穎化合物
MA50567A (fr) * 2017-11-09 2020-09-16 Inflazome Ltd Nouveaux composés de sulfonamide carboxamide
US12221434B2 (en) 2017-11-09 2025-02-11 Inflazome Limited Sulfonamide carboxamide compounds
WO2019166619A1 (en) 2018-03-02 2019-09-06 Inflazome Limited Novel compounds

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2552261B2 (ja) 1978-05-30 1996-11-06 イー・アイ・デユポン・ドウ・ヌムール・アンド・カンパニー 農業用スルホンアミド類およびその製造法
US4347251A (en) 1981-07-13 1982-08-31 American Cyanamid Company Novel 3-substituted amino-1-substituted heteroaryl-2-pyrazolines
US4954164A (en) * 1982-02-27 1990-09-04 Nissan Chemical Industries, Ltd. Pyrazolesulfonylurea derivatives, preparation thereof, herbicide containing said derivative as active ingredient and herbicidal method by use thereof
EP0096003B2 (de) * 1982-05-28 1994-06-15 Ciba-Geigy Ag Neue Sulfonyl(thio)harnstoffe, Verfahren zu deren Herstellung und deren Verwendung als Herbizide und/oder Wachstumsregulatoren
DE3379462D1 (de) * 1982-06-01 1989-04-27 Du Pont Herbicidal imidazole, pyrazole, thiazole and isothiazole derivatives
US4534790A (en) * 1982-10-07 1985-08-13 E. I. Du Pont De Nemours And Company Herbicidal sulfonamides
JPS59167570A (ja) 1983-03-04 1984-09-21 バイエル・アクチエンゲゼルシヤフト グアニジン誘導体
JPS606654A (ja) 1983-06-24 1985-01-14 Nippon Tokushu Noyaku Seizo Kk 置換フエニルスルホニルグアニジン誘導体、その中間体、それらの製法及び除草剤
JPS6036467A (ja) 1983-08-10 1985-02-25 Nippon Tokushu Noyaku Seizo Kk 置換フエニルスルホニルグアニジン誘導体、その中間体、それらの製法及び雑草防除剤
US4705558A (en) * 1984-10-19 1987-11-10 E. I. Du Pont De Nemours And Company Herbicidal pyrazolesulfonamides
AU578307B2 (en) * 1984-09-17 1988-10-20 E.I. Du Pont De Nemours And Company Herbicidal pyrazolesulfonamides
AU4789685A (en) * 1984-09-28 1986-04-10 E.I. Du Pont De Nemours And Company Heterocyclic sulphonamide derivatives
US4690705A (en) * 1984-11-30 1987-09-01 E. I. Du Pont De Nemours And Company Herbicidal sulfonamides

Also Published As

Publication number Publication date
EP0318602A1 (en) 1989-06-07
IN165281B (ro) 1989-09-09
ES8706324A1 (es) 1987-06-16
US4881965A (en) 1989-11-21
PL151526B1 (en) 1990-09-28
FI855180A0 (fi) 1985-12-30
CN86100911A (zh) 1986-09-24
FI855180L (fi) 1986-07-19
DE3688374D1 (de) 1993-06-03
BR8600183A (pt) 1986-09-30
PL257531A1 (en) 1987-09-21
AU595176B2 (en) 1990-03-29
EP0189069A2 (en) 1986-07-30
DK25386D0 (da) 1986-01-17
DE3688374T2 (de) 1993-10-21
HUT39727A (en) 1986-10-29
EP0189069A3 (en) 1986-12-30
GR860049B (en) 1986-05-12
TR22668A (tr) 1988-02-23
HU200596B (en) 1990-07-28
DK25386A (da) 1986-07-19
EP0318602B1 (en) 1993-04-28
FI855180A7 (fi) 1986-07-19
AU5211686A (en) 1986-07-24
ATE88703T1 (de) 1993-05-15
RO94159A2 (ro) 1988-03-30
YU45761B (sh) 1992-07-20
ES550931A0 (es) 1987-06-16
YU7086A (en) 1987-10-31
SU1701104A3 (ru) 1991-12-23

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