RO86363A - Procedeu pentru prepararea unor derivati de metiltiopirimidina - Google Patents

Procedeu pentru prepararea unor derivati de metiltiopirimidina

Info

Publication number
RO86363A
RO86363A RO83109750A RO10975083A RO86363A RO 86363 A RO86363 A RO 86363A RO 83109750 A RO83109750 A RO 83109750A RO 10975083 A RO10975083 A RO 10975083A RO 86363 A RO86363 A RO 86363A
Authority
RO
Romania
Prior art keywords
preparation
methylthiopyrimidine
derivatives
methylthiopyrimidine derivatives
Prior art date
Application number
RO83109750A
Other languages
English (en)
French (fr)
Other versions
RO86363B (ro
Inventor
Ishikawa Katsutoshi
Shimotori Hitoshi
Lida Noburi
Anihiro Kazuo Kazuo
Shuji Ozawa
Original Assignee
Mitsui Toatsu Chemicals Inc,Jp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Mitsui Toatsu Chemicals Inc,Jp filed Critical Mitsui Toatsu Chemicals Inc,Jp
Publication of RO86363A publication Critical patent/RO86363A/ro
Publication of RO86363B publication Critical patent/RO86363B/ro

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D407/00Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00
    • C07D407/02Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings
    • C07D407/12Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/541,3-Diazines; Hydrogenated 1,3-diazines
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/60Three or more oxygen or sulfur atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Dentistry (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Agronomy & Crop Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
RO109750A 1982-01-20 1983-01-17 Procedeu pentru prepararea unor derivati de metiltiopirimidina RO86363B (ro)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP57006142A JPS58124773A (ja) 1982-01-20 1982-01-20 5−メチルチオピリミジン誘導体とその製造法と農園芸用殺菌剤

Publications (2)

Publication Number Publication Date
RO86363A true RO86363A (ro) 1985-03-15
RO86363B RO86363B (ro) 1985-03-31

Family

ID=11630260

Family Applications (4)

Application Number Title Priority Date Filing Date
RO83116657A RO89716A (ro) 1982-01-20 1983-01-17 Compozitie fungicida lichida
RO83116656A RO89715A (ro) 1982-01-20 1983-01-17 Compozitie fungicida solida
RO83116655A RO89714A (ro) 1982-01-20 1983-01-17 Procedeu de preparare a unor derivati de 5-metiltiopirimidina
RO109750A RO86363B (ro) 1982-01-20 1983-01-17 Procedeu pentru prepararea unor derivati de metiltiopirimidina

Family Applications Before (3)

Application Number Title Priority Date Filing Date
RO83116657A RO89716A (ro) 1982-01-20 1983-01-17 Compozitie fungicida lichida
RO83116656A RO89715A (ro) 1982-01-20 1983-01-17 Compozitie fungicida solida
RO83116655A RO89714A (ro) 1982-01-20 1983-01-17 Procedeu de preparare a unor derivati de 5-metiltiopirimidina

Country Status (11)

Country Link
US (1) US4540698A (ro)
JP (1) JPS58124773A (ro)
DD (2) DD209447A5 (ro)
DE (1) DE3301106A1 (ro)
FR (1) FR2519983B1 (ro)
GB (1) GB2113216B (ro)
IN (1) IN157931B (ro)
IT (1) IT1163039B (ro)
NL (1) NL8300193A (ro)
PL (1) PL138343B1 (ro)
RO (4) RO89716A (ro)

Families Citing this family (30)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS59227867A (ja) * 1983-06-09 1984-12-21 Mitsui Toatsu Chem Inc 5―メチルチオピリミジン誘導体とその製造法と農園芸用殺菌剤
JPH0635450B2 (ja) * 1984-03-16 1994-05-11 三井東圧化学株式会社 チオシアノピリミジン誘導体、その製造法および農園芸用殺菌剤
JPS6345269A (ja) * 1986-04-28 1988-02-26 Mitsui Toatsu Chem Inc ジハロゲン置換チオシアノピリミジン誘導体、その製造法および農園芸用殺菌剤
JPS63112566A (ja) * 1986-10-28 1988-05-17 Nissan Chem Ind Ltd ピリミジノン誘導体、その製法および殺虫・殺ダニ・殺菌剤
JPH0827122A (ja) * 1994-07-15 1996-01-30 Kureha Chem Ind Co Ltd 2−(ベンジルオキシ)(フェノキシ)ピリミジン誘導体、その製造方法及び除草剤
US6090815A (en) * 1996-10-31 2000-07-18 Kumiai Chemical Industry Co., Ltd. Pyrimidinyloxyalkanoic amide derivatives and fungicides for agricultural and horticultural use
US7473691B2 (en) * 2000-09-15 2009-01-06 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
US6660731B2 (en) * 2000-09-15 2003-12-09 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
CA2422367C (en) * 2000-09-15 2010-05-18 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
WO2002059111A2 (en) * 2000-12-21 2002-08-01 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
EP2322521B1 (en) * 2002-02-06 2013-09-04 Vertex Pharmaceuticals, Inc. Heteroaryl compounds useful as inhibitors of GSK-3
US20040009981A1 (en) * 2002-03-15 2004-01-15 David Bebbington Compositions useful as inhibitors of protein kinases
MY141867A (en) * 2002-06-20 2010-07-16 Vertex Pharma Substituted pyrimidines useful as protein kinase inhibitors
JP4733388B2 (ja) * 2002-08-02 2011-07-27 バーテックス ファーマシューティカルズ インコーポレイテッド Gsk−3のインヒビターとして有用なピラゾール組成物
WO2004072029A2 (en) * 2003-02-06 2004-08-26 Vertex Pharmaceuticals Incorporated Pyrazolopyridazines useful as inhibitors of protein kinases
CN1902193B (zh) * 2003-12-04 2011-07-13 沃泰克斯药物股份有限公司 可用作蛋白激酶抑制剂的喹喔啉
AU2006279376B2 (en) * 2005-08-18 2011-04-14 Vertex Pharmaceuticals Incoporated Pyrazine kinase inhibitors
BRPI0619706A2 (pt) * 2005-11-03 2011-10-11 Vertex Pharma composto, composição, método para inibir a atividade da proteìna aurora quinase numa amostra biológica, método para tratar um distúrbio proliferativo num paciente, método para tratar cáncer num indivìduo
MX2009004807A (es) * 2006-11-02 2009-06-15 Vertex Pharma Aminopiridinas y aminopirimidinas utiles como inhibidores de proteina cinasa.
EP2099787B1 (en) * 2006-12-19 2010-07-21 Vertex Pharmaceuticals, Inc. Aminopyrimidines useful as inhibitors of protein kinases
JP2010520887A (ja) 2007-03-09 2010-06-17 バーテックス ファーマシューティカルズ インコーポレイテッド 蛋白キナーゼの阻害剤として有用なアミノピリジン
JP5520057B2 (ja) * 2007-03-09 2014-06-11 バーテックス ファーマシューティカルズ インコーポレイテッド 蛋白キナーゼの阻害剤として有用なアミノピリミジン
JP5393489B2 (ja) * 2007-03-09 2014-01-22 バーテックス ファーマシューティカルズ インコーポレイテッド 蛋白キナーゼの阻害剤として有用なアミノピリミジン
NZ580343A (en) 2007-04-13 2012-03-30 Vertex Pharma Aminopyrimidines useful as kinase inhibitors
CA2694381A1 (en) * 2007-05-02 2008-11-13 Vertex Pharmaceuticals Incorporated Aminopyrimidines useful as kinase inhibitors
MX2009011810A (es) * 2007-05-02 2010-01-14 Vertex Pharma Tiazoles y pirazoles utiles como inhibidores de cinasa.
CA2688584A1 (en) * 2007-05-02 2008-11-13 Vertex Pharmaceuticals Incorporated Aminopyrimidines useful as kinase inhibitors
AU2008257044A1 (en) * 2007-05-24 2008-12-04 Vertex Pharmaceuticals Incorporated Thiazoles and pyrazoles useful as kinase inhibitors
WO2009018415A1 (en) * 2007-07-31 2009-02-05 Vertex Pharmaceuticals Incorporated Process for preparing 5-fluoro-1h-pyrazolo [3, 4-b] pyridin-3-amine and derivatives thereof
RU2011112802A (ru) * 2008-09-03 2012-10-10 Вертекс Фармасьютикалз Инкорпорейтед (Us) Сокристаллы и содержащие их фармацевтические композиции

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4199583A (en) * 1970-07-13 1980-04-22 The Upjohn Company Antifungal method, formulations and compounds
US4126459A (en) * 1976-05-14 1978-11-21 Polaroid Corporation Thioether substituted silver halide solvents
US4211559A (en) * 1976-09-30 1980-07-08 Texas Instruments Incorporated Photographic processes and compositions employing thioether containing silver halide solvents

Also Published As

Publication number Publication date
US4540698A (en) 1985-09-10
GB2113216B (en) 1985-12-04
FR2519983B1 (fr) 1985-12-06
DD209447A5 (de) 1984-05-09
DD219654A5 (de) 1985-03-13
RO89716A (ro) 1986-07-30
RO89714A (ro) 1986-07-30
FR2519983A1 (fr) 1983-07-22
IT1163039B (it) 1987-04-08
NL8300193A (nl) 1983-08-16
RO86363B (ro) 1985-03-31
PL138343B1 (en) 1986-09-30
GB2113216A (en) 1983-08-03
PL240209A1 (en) 1984-06-18
JPH0378383B2 (ro) 1991-12-13
JPS58124773A (ja) 1983-07-25
DE3301106A1 (de) 1983-07-28
RO89715A (ro) 1986-07-30
IT8319164A0 (it) 1983-01-18
GB8300400D0 (en) 1983-02-09
IN157931B (ro) 1986-07-26

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