RO84361A - Procedeu pentru prepararea unor derivati peptidici antagonisti ai actiunii antidiuretice si/sau vasopresoare a argininvasopresiunei - Google Patents

Procedeu pentru prepararea unor derivati peptidici antagonisti ai actiunii antidiuretice si/sau vasopresoare a argininvasopresiunei

Info

Publication number
RO84361A
RO84361A RO82107007A RO10700782A RO84361A RO 84361 A RO84361 A RO 84361A RO 82107007 A RO82107007 A RO 82107007A RO 10700782 A RO10700782 A RO 10700782A RO 84361 A RO84361 A RO 84361A
Authority
RO
Romania
Prior art keywords
vasopresous
argininvasopression
durably
diabetes
preparation
Prior art date
Application number
RO82107007A
Other languages
English (en)
French (fr)
Other versions
RO84361B (ro
Inventor
Maurice Manning
Wilbur H Sawyer
Original Assignee
Medical College Of Ohio,The Trustees Of Columbia University,Us
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US06/247,008 external-priority patent/US4367225A/en
Application filed by Medical College Of Ohio,The Trustees Of Columbia University,Us filed Critical Medical College Of Ohio,The Trustees Of Columbia University,Us
Publication of RO84361A publication Critical patent/RO84361A/ro
Publication of RO84361B publication Critical patent/RO84361B/ro

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04Linear peptides containing only normal peptide links
    • C07K7/16Oxytocins; Vasopressins; Related peptides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10STECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10S930/00Peptide or protein sequence
    • Y10S930/01Peptide or protein sequence
    • Y10S930/15Oxytocin or vasopressin; related peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Immunology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
RO107007A 1981-03-24 1982-03-23 Procedeu pentru prepararea unor derivati peptidici antagonisti ai actiunii antidiuretice si/sau vasopresoare a argininvasopresiunei RO84361B (ro)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US06/247,008 US4367225A (en) 1981-03-24 1981-03-24 Novel antagonists of the antidiuretic and/or vasopressor action of arginine vasopressin
US06/322,071 US4399125A (en) 1981-03-24 1981-11-16 Novel antagonists of the antidiuretic action of arginine vasopressin

Publications (2)

Publication Number Publication Date
RO84361A true RO84361A (ro) 1984-05-23
RO84361B RO84361B (ro) 1984-07-30

Family

ID=26938391

Family Applications (1)

Application Number Title Priority Date Filing Date
RO107007A RO84361B (ro) 1981-03-24 1982-03-23 Procedeu pentru prepararea unor derivati peptidici antagonisti ai actiunii antidiuretice si/sau vasopresoare a argininvasopresiunei

Country Status (21)

Country Link
US (1) US4399125A (ro)
EP (1) EP0061356B1 (ro)
KR (1) KR880000758B1 (ro)
AU (1) AU546865B2 (ro)
BG (1) BG38487A3 (ro)
CA (1) CA1185235A (ro)
DD (2) DD202695A5 (ro)
DE (1) DE3264734D1 (ro)
DK (1) DK130182A (ro)
ES (2) ES8604264A1 (ro)
FI (1) FI77047C (ro)
HU (1) HU189127B (ro)
IE (1) IE52624B1 (ro)
IL (1) IL65211A (ro)
NO (1) NO162024C (ro)
NZ (1) NZ199908A (ro)
PH (1) PH19237A (ro)
PT (1) PT74615B (ro)
RO (1) RO84361B (ro)
YU (1) YU63482A (ro)
ZW (1) ZW4882A1 (ro)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4491577A (en) * 1981-11-16 1985-01-01 The Medical College Of Ohio Antagonists of the antidiuretic action of arginine vasopressin
DK153883A (da) * 1982-04-20 1983-10-21 Ceskoslovenska Akademie Ved Vasopressin-analoge
US4587045A (en) * 1983-02-16 1986-05-06 Smithkline Beckman Corporation Intermediates for preparing octapeptide vasopressin antagonists
US4469679A (en) * 1983-02-16 1984-09-04 Smithkline Beckman Corporation Octapeptide vasopressin antagonists
US4483794A (en) * 1983-05-10 1984-11-20 Ceskoslovenska Akademie Ved Analogs of neurohypophysial hormones
CA1238314A (en) * 1983-09-22 1988-06-21 James F. Callahan Process for preparing basic heptapeptide vasopressin antagonists
US4551445A (en) * 1983-10-14 1985-11-05 The Medical College Of Ohio Derivatives of arginine vasopressin antagonists
US4649130A (en) * 1984-01-26 1987-03-10 Medical College Of Ohio Novel derivatives of arginine vasopressin antagonists
US4714696A (en) * 1984-01-26 1987-12-22 Medical College Of Ohio Novel derivatives of arginine vasopressin antagonists
CA1249397A (en) * 1984-03-07 1989-01-24 Fadia E. Ali Process for preparing des-proline vasopressin antagonists
US4481193A (en) * 1984-03-07 1984-11-06 Smithkline Beckman Corporation Des-proline vasopressin antagonists
US4481194A (en) * 1984-03-07 1984-11-06 Smithkline Beckman Corporation Des-proline-des-glycine vasopressin antagonists
US4597901A (en) * 1984-12-14 1986-07-01 Smithkline Beckman Corporation β-indolylalanyl or β-indolylglycinyl vasopressin antagonists
US4719199A (en) * 1984-12-14 1988-01-12 Smithkline Beckman Corporation Diuretic compositions and methods of producing diuresis
US4684716A (en) * 1984-12-14 1987-08-04 Smithkline Beckman Corporation Polypeptide intermediates
US4624943A (en) * 1985-03-20 1986-11-25 Smithkline Beckman Corporation Aromatic basic-tailed vasopressin antagonists
WO1987002676A1 (en) * 1985-10-25 1987-05-07 Gibson-Stephens Neuropharmaceuticals, Inc. Conformationally constrained oxytocin antagonists with prolonged biological activities
PT84342B (pt) * 1986-02-25 1989-09-14 Smithkline Beecham Corp Processo de preparacao de compostos de vasopressina
US4762820A (en) * 1986-03-03 1988-08-09 Trustees Of Boston University Therapeutic treatment for congestive heart failure
WO1988005661A1 (en) * 1987-01-30 1988-08-11 Biomed Research Consultants, Limited Vasopressin-based pharmaceutical compositions
US5055448A (en) * 1987-06-25 1991-10-08 Medical College Of Ohio Linear derivatives of arginine vasopressin antagonists
AT398766B (de) * 1988-05-26 1995-01-25 Gebro Broschek Gmbh Verfahren zur intramolekularen oxidation von zwei -sh gruppen in einer peptidverbindung zu einer disulfidbrücke
US5070187A (en) * 1989-11-03 1991-12-03 Trustees Of Boston University Pharmacologically effective antagonists of arginine-vasopressin
US5051400A (en) * 1990-06-28 1991-09-24 Smithkline Beecham Corporation Method of treating nausea and emesis related to motion sickness with vasopressin antagonists
RU2342949C1 (ru) * 2007-03-26 2009-01-10 Юрий Георгиевич Жуковский Применение [дезамино-1, изолейцин-3, аргинин-8]вазопрессина в качестве средства для увеличения выведения почкой солей натрия и усиления обратного избирательного всасывания из почечных канальцев в кровь воды-растворителя
CN111253569B (zh) * 2020-02-26 2021-06-01 山东大学 一种聚合物、其制剂及其制备方法和应用

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1193509B (de) * 1960-06-02 1965-05-26 Hoechst Ag Verfahren zur Herstellung eines neuen Oktapeptids mit vasopressorischer Wirksamkeit
CH426861A (de) * 1963-06-06 1966-12-31 Sandoz Ag Verfahren zur Herstellung eines bisher unbekannten Polypeptids
CH442342A (de) * 1964-07-17 1967-08-31 Sandoz Ag Verfahren zur Herstellung eines neuen Polypeptids
CH460039A (de) * 1965-04-15 1968-07-31 Sandoz Ag Verfahren zur Herstellung eines neuen Polypeptids
CH495957A (de) * 1966-09-15 1970-09-15 Ceskoslovenska Akademie Ved Verfahren zur Herstellung eines antidiuretisch wirksamen Polypeptids
US4148787A (en) * 1976-05-24 1979-04-10 Ferring Ab Antidiuretically effective polypeptide and a process for preparing the same

Also Published As

Publication number Publication date
FI77047C (fi) 1989-01-10
NO820967L (no) 1982-09-27
DD202695A5 (de) 1983-09-28
CA1185235A (en) 1985-04-09
IE820465L (en) 1982-09-24
BG38487A3 (en) 1985-12-16
US4399125A (en) 1983-08-16
FI821019L (fi) 1982-09-25
EP0061356A3 (en) 1982-12-29
NZ199908A (en) 1985-09-13
PH19237A (en) 1986-02-14
RO84361B (ro) 1984-07-30
ZW4882A1 (en) 1983-02-23
IE52624B1 (en) 1988-01-06
DD212735A5 (de) 1984-08-22
PT74615A (en) 1982-04-01
ES8703489A1 (es) 1987-03-01
KR880000758B1 (ko) 1988-05-06
HU189127B (en) 1986-06-30
FI821019A0 (fi) 1982-03-23
AU546865B2 (en) 1985-09-26
NO162024C (no) 1989-10-25
YU63482A (en) 1985-10-31
FI77047B (fi) 1988-09-30
ES510579A0 (es) 1986-01-16
NO162024B (no) 1989-07-17
PT74615B (en) 1983-10-20
IL65211A0 (en) 1982-05-31
DE3264734D1 (en) 1985-08-22
KR830008683A (ko) 1983-12-14
EP0061356B1 (en) 1985-07-17
AU8161782A (en) 1982-09-30
IL65211A (en) 1986-02-28
ES8604264A1 (es) 1986-01-16
DK130182A (da) 1982-09-25
ES546137A0 (es) 1987-03-01
EP0061356A2 (en) 1982-09-29

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