PT975638E - Epothilons modificados nas cadeias laterais - Google Patents

Epothilons modificados nas cadeias laterais

Info

Publication number
PT975638E
PT975638E PT98912388T PT98912388T PT975638E PT 975638 E PT975638 E PT 975638E PT 98912388 T PT98912388 T PT 98912388T PT 98912388 T PT98912388 T PT 98912388T PT 975638 E PT975638 E PT 975638E
Authority
PT
Portugal
Prior art keywords
epothilons
modified
lateral chains
chains
lateral
Prior art date
Application number
PT98912388T
Other languages
English (en)
Inventor
Hofle Prof Dr Gerhard
Michael Sefkow
Original Assignee
Biotechnolog Forschung Mbh Gbf
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Biotechnolog Forschung Mbh Gbf filed Critical Biotechnolog Forschung Mbh Gbf
Publication of PT975638E publication Critical patent/PT975638E/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D493/00Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
    • C07D493/02Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains two hetero rings
    • C07D493/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Addition Polymer Or Copolymer, Post-Treatments, Or Chemical Modifications (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Other Resins Obtained By Reactions Not Involving Carbon-To-Carbon Unsaturated Bonds (AREA)
  • Silicon Polymers (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Polyesters Or Polycarbonates (AREA)
  • Epoxy Compounds (AREA)
PT98912388T 1997-02-25 1998-02-25 Epothilons modificados nas cadeias laterais PT975638E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19707505 1997-02-25

Publications (1)

Publication Number Publication Date
PT975638E true PT975638E (pt) 2002-12-31

Family

ID=7821415

Family Applications (1)

Application Number Title Priority Date Filing Date
PT98912388T PT975638E (pt) 1997-02-25 1998-02-25 Epothilons modificados nas cadeias laterais

Country Status (25)

Country Link
US (1) US6359140B1 (pt)
EP (2) EP1201666A3 (pt)
JP (1) JP2001513098A (pt)
KR (1) KR100494179B1 (pt)
CN (2) CN1544436A (pt)
AR (1) AR011878A1 (pt)
AT (1) ATE221888T1 (pt)
AU (1) AU736062B2 (pt)
BR (1) BR9807742B1 (pt)
CA (1) CA2281105A1 (pt)
CZ (1) CZ298027B6 (pt)
DE (2) DE19880193D2 (pt)
DK (1) DK0975638T3 (pt)
ES (1) ES2183338T3 (pt)
HK (1) HK1023774A1 (pt)
HU (1) HU228851B1 (pt)
IL (1) IL131343A (pt)
NO (1) NO327211B1 (pt)
NZ (1) NZ337195A (pt)
PL (1) PL190422B1 (pt)
PT (1) PT975638E (pt)
RU (1) RU2201932C2 (pt)
TW (1) TW480263B (pt)
WO (1) WO1998038192A1 (pt)
ZA (1) ZA981575B (pt)

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* Cited by examiner, † Cited by third party
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US6518421B1 (en) * 2000-03-20 2003-02-11 Bristol-Myers Squibb Company Process for the preparation of epothilone analogs
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US7649006B2 (en) 2002-08-23 2010-01-19 Sloan-Kettering Institute For Cancer Research Synthesis of epothilones, intermediates thereto and analogues thereof
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US7820702B2 (en) 2004-02-04 2010-10-26 Bristol-Myers Squibb Company Sulfonylpyrrolidine modulators of androgen receptor function and method
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US7696241B2 (en) 2004-03-04 2010-04-13 Bristol-Myers Squibb Company Bicyclic compounds as modulators of androgen receptor function and method
US7625923B2 (en) 2004-03-04 2009-12-01 Bristol-Myers Squibb Company Bicyclic modulators of androgen receptor function
BRPI0518286A2 (pt) * 2004-11-18 2008-11-11 Bristol Myers Squibb Co microesfera com revestimento entÉrico contendo ixabepilona e sua preparaÇço
US20060134214A1 (en) * 2004-11-18 2006-06-22 Ismat Ullah Enteric coated bead comprising epothilone or epothilone analog, and preparation and administration thereof
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BRPI0718360A2 (pt) 2006-12-04 2013-11-12 Univ Illinois "composições e métodos para o tratamento do câncer com cupredoxinas e dna rico em cpg"
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US8846006B2 (en) 2011-01-20 2014-09-30 Board Of Regents, The University Of Texas System MRI markers, delivery and extraction systems, and methods of manufacture and use thereof
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Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4138042C2 (de) * 1991-11-19 1993-10-14 Biotechnolog Forschung Gmbh Epothilone, deren Herstellungsverfahren sowie diese Verbindungen enthaltende Mittel
DE59609305D1 (de) * 1995-11-17 2002-07-11 Biotechnolog Forschung Gmbh Epothilon-Derivate und deren Herstellung
US6441186B1 (en) * 1996-12-13 2002-08-27 The Scripps Research Institute Epothilone analogs
EP1201666A3 (de) * 1997-02-25 2003-03-05 Gesellschaft für biotechnologische Forschung mbH (GBF) Seitenkettenmodifizierte Epothilone

Also Published As

Publication number Publication date
EP1201666A3 (de) 2003-03-05
ES2183338T3 (es) 2003-03-16
DE19880193D2 (de) 2000-08-24
EP1201666A2 (de) 2002-05-02
ZA981575B (en) 1998-09-08
CA2281105A1 (en) 1998-09-03
NZ337195A (en) 2001-05-25
US6359140B1 (en) 2002-03-19
CZ298027B6 (cs) 2007-05-30
CN1128803C (zh) 2003-11-26
BR9807742B1 (pt) 2010-12-14
CZ286599A3 (cs) 2000-03-15
IL131343A0 (en) 2001-01-28
RU2201932C2 (ru) 2003-04-10
IL131343A (en) 2004-03-28
KR100494179B1 (ko) 2005-06-10
KR20000075705A (ko) 2000-12-26
EP0975638A1 (de) 2000-02-02
HU228851B1 (en) 2013-06-28
BR9807742A (pt) 2000-02-22
NO327211B1 (no) 2009-05-11
HUP0002189A3 (en) 2001-12-28
TW480263B (en) 2002-03-21
NO994071D0 (no) 1999-08-24
AU6724998A (en) 1998-09-18
CN1248974A (zh) 2000-03-29
DK0975638T3 (da) 2002-11-18
DE59805110D1 (de) 2002-09-12
EP0975638B1 (de) 2002-08-07
WO1998038192A1 (de) 1998-09-03
PL190422B1 (pl) 2005-12-30
ATE221888T1 (de) 2002-08-15
AU736062B2 (en) 2001-07-26
JP2001513098A (ja) 2001-08-28
HK1023774A1 (en) 2000-09-22
PL335329A1 (en) 2000-04-25
NO994071L (no) 1999-10-21
CN1544436A (zh) 2004-11-10
HUP0002189A2 (hu) 2001-10-28
AR011878A1 (es) 2000-09-13

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