PT92628A - Processo de preparacao de acidos carboxilicos aza-heterociclicos n-substituidos e de composicoes farmaceuticas que os contem - Google Patents
Processo de preparacao de acidos carboxilicos aza-heterociclicos n-substituidos e de composicoes farmaceuticas que os contemInfo
- Publication number
- PT92628A PT92628A PT92628A PT9262889A PT92628A PT 92628 A PT92628 A PT 92628A PT 92628 A PT92628 A PT 92628A PT 9262889 A PT9262889 A PT 9262889A PT 92628 A PT92628 A PT 92628A
- Authority
- PT
- Portugal
- Prior art keywords
- preparation
- carboxylic acid
- pharmaceutical compositions
- substituted
- heterocyclic carboxylic
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/60—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/68—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
- C07D211/72—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D211/78—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Biomedical Technology (AREA)
- Public Health (AREA)
- Pain & Pain Management (AREA)
- Anesthesiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Cephalosporin Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Plural Heterocyclic Compounds (AREA)
- Steroid Compounds (AREA)
- Pyrrole Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Bipolar Transistors (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DK704488A DK704488D0 (da) | 1988-12-19 | 1988-12-19 | Nye n-substituerede azaheterocykliske carboxylsyrer |
Publications (2)
Publication Number | Publication Date |
---|---|
PT92628A true PT92628A (pt) | 1990-06-29 |
PT92628B PT92628B (pt) | 1995-09-12 |
Family
ID=8149197
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PT92628A PT92628B (pt) | 1988-12-19 | 1989-12-19 | Processo de preparacao de acidos carboxilicos aza-heterociclicos n-substituidos e de composicoes farmaceuticas que os contem |
Country Status (16)
Country | Link |
---|---|
US (1) | US5071859A (pt) |
EP (1) | EP0374801B1 (pt) |
JP (1) | JP2848534B2 (pt) |
AT (1) | ATE150455T1 (pt) |
AU (1) | AU634992B2 (pt) |
CA (1) | CA2005919C (pt) |
DE (1) | DE68927875T2 (pt) |
DK (1) | DK704488D0 (pt) |
ES (1) | ES2099067T3 (pt) |
FI (1) | FI93951C (pt) |
GR (1) | GR3023379T3 (pt) |
IL (1) | IL92652A0 (pt) |
NO (1) | NO177672C (pt) |
NZ (1) | NZ231836A (pt) |
PT (1) | PT92628B (pt) |
ZA (1) | ZA899736B (pt) |
Families Citing this family (27)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4910312A (en) * | 1985-11-08 | 1990-03-20 | Warner-Lambert Company | Various N-substituted 3-piperidine carboxylic acids or N-substituted 3-pyridinecarboxylic acids and derivatives thereof |
DE3609699A1 (de) * | 1986-03-20 | 1987-09-24 | Schering Ag | 5- oder 6-substituierte-(beta)-carbolin-3-carbonsaeureester |
US5214054A (en) * | 1988-05-18 | 1993-05-25 | Novo Nordisk A/S | Azacyclic carboxylic acid derivatives and their preparation and use |
FR2653123B1 (fr) * | 1989-10-17 | 1992-01-17 | Roussel Uclaf | Nouveaux derives de la pyridone, leur procede de preparation, les nouveaux intermediaires obtenus, leur application a titre de medicaments et les compositions pharmaceutiques les renfermant. |
DK588189D0 (da) * | 1989-11-22 | 1989-11-22 | Novo Nordisk As | Nye heterocykliske carboxylsyrer |
DE4017211A1 (de) * | 1990-05-29 | 1991-12-05 | Merck Patent Gmbh | Oxazolidinone |
DK181190D0 (da) * | 1990-07-30 | 1990-07-30 | Lundbeck & Co As H | 3-aryl-indol- eller 3-aryl-indazolderivater |
DE4117904A1 (de) * | 1991-05-31 | 1992-12-03 | Basf Ag | Substituierte n-phenylpiperidine |
DK93791D0 (da) * | 1991-05-17 | 1991-05-17 | Novo Nordisk As | Nye heterocykliske carboxylsyrer |
EP0535496A1 (en) * | 1991-09-25 | 1993-04-07 | Hoechst-Roussel Pharmaceuticals Incorporated | (1-Indanon-2yl)methylpiperidines, intermediates and a process for their preparation and their use as medicaments |
EP0767174A1 (de) * | 1991-11-21 | 1997-04-09 | Ciba-Geigy Ag | Neue Aminoalkanphosphinsäuren und ihre Salze |
US5807872A (en) * | 1992-12-16 | 1998-09-15 | Schering Corporation | Imidazoylalkyl substituted with a six membered nitrogen containing heterocyclic ring |
US5932596A (en) * | 1991-12-18 | 1999-08-03 | Schering Corporation | Imidazoylalkyl substituted with a six membered nitrogen containing nitrogen containing heterocyclic ring |
US5633250A (en) * | 1991-12-18 | 1997-05-27 | Schering Corporation | Imidazoylalkyl substituted with a six or seven membered heterocyclic ring containing two nitrogen atoms |
DE69212844T2 (de) * | 1991-12-18 | 1997-01-09 | Schering Corp., Kenilworth, N.J. | Imidazolyl oder imidazolylalkyl substituiert mit einem 4- oder 5-gliedrigen stickstoff enthaltenden heterozyklischen ring |
GB9127306D0 (en) * | 1991-12-23 | 1992-02-19 | Boots Co Plc | Therapeutic agents |
US5284957A (en) * | 1992-09-03 | 1994-02-08 | Eli Lilly And Company | Excitatory amino acid receptor antagonists |
US5286733A (en) * | 1992-11-20 | 1994-02-15 | Sterling Winthrop Inc. | Substituted 3-piperidinealkanoates and alkanones and compositions and method of use thereof |
US5580877A (en) * | 1994-04-25 | 1996-12-03 | Merck Sharp & Dohme Ltd. | Pyrazolo-quinoline derivatives for treating cerebral ischemia |
US5962449A (en) | 1995-04-07 | 1999-10-05 | Novo Nordisk A/S | Tricyclic compounds in treating hyperalgesic conditions and NIDDM |
FR2735476B1 (fr) * | 1995-06-14 | 1997-07-18 | Rhone Poulenc Rorer Sa | Nouvelle application de derives du pyrrole |
US5747523A (en) * | 1996-01-24 | 1998-05-05 | Guilford Pharmaceuticals Inc. | Substituted ethyl α,α-diarylmethyl ether derivatives |
WO1999031056A1 (fr) * | 1997-12-12 | 1999-06-24 | Toyama Chemical Co., Ltd. | Derives d'ether alcoylique ou leurs sels, et antagonistes du calcium les contenant |
DE19840611A1 (de) * | 1998-09-05 | 2000-03-09 | Klaus Wanner | GABA-uptake-Inhibitoren mit Pyrrolidinstruktur |
US20040010010A1 (en) * | 2002-04-30 | 2004-01-15 | Ebetino Frank Hallock | Melanocortin receptor ligands |
US7026335B2 (en) * | 2002-04-30 | 2006-04-11 | The Procter & Gamble Co. | Melanocortin receptor ligands |
JP2023533387A (ja) * | 2020-07-02 | 2023-08-02 | シー ファーマシューティカルズ エルエルシー | 6‐(2‐(2h‐テトラゾール‐5‐イル)エチル)‐6‐フルオロデカヒドロイソキノリン‐3‐カルボキシル酸及びそのエステル誘導体の医薬組成物 |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU552050B2 (en) * | 1981-05-26 | 1986-05-22 | Smithkline Beckman Corporation | N-substituted azeheterocyclic carboxylic acids and their esters |
US4383999A (en) * | 1981-05-26 | 1983-05-17 | Smithkline Beckman Corporation | Inhibition of GABA uptake by N-substituted azaheterocyclic carboxylic acids and their esters |
US4514414A (en) * | 1982-10-25 | 1985-04-30 | Smithkline Beckman Corporation | N-Substituted pyrrolidineacetic acids and their esters |
FI83957C (fi) * | 1984-09-28 | 1991-09-25 | Byk Gulden Lomberg Chem Fab | Foerfarande foer framstaellning av nya, terapeutiskt anvaendbara diarylfoereningar. |
DK288385D0 (da) * | 1985-06-26 | 1985-06-26 | Novo Industri As | Aminosyrederivater |
FI864246A (fi) * | 1985-11-08 | 1987-05-09 | Warner Lambert Co | N-substituerade 3-piperidin- eller 3-pyridinkarboxylsyror samt deras derivat. |
US4910312A (en) * | 1985-11-08 | 1990-03-20 | Warner-Lambert Company | Various N-substituted 3-piperidine carboxylic acids or N-substituted 3-pyridinecarboxylic acids and derivatives thereof |
IL81179A (en) * | 1986-01-07 | 1992-02-16 | Novo Nordisk As | N-phenylbutenyl substituted azaheterocyclic carboxylic acids,their preparation and pharmaceutical compositions comprising them |
DK270488D0 (da) * | 1988-05-18 | 1988-05-18 | Novo Industri As | Hidtil ukendte o-substituerede ketoximer |
-
1988
- 1988-12-19 DK DK704488A patent/DK704488D0/da not_active Application Discontinuation
-
1989
- 1989-12-12 IL IL92652A patent/IL92652A0/xx not_active IP Right Cessation
- 1989-12-14 US US07/450,805 patent/US5071859A/en not_active Expired - Fee Related
- 1989-12-18 NZ NZ231836A patent/NZ231836A/xx unknown
- 1989-12-18 ES ES89123400T patent/ES2099067T3/es not_active Expired - Lifetime
- 1989-12-18 AT AT89123400T patent/ATE150455T1/de not_active IP Right Cessation
- 1989-12-18 EP EP89123400A patent/EP0374801B1/en not_active Expired - Lifetime
- 1989-12-18 DE DE68927875T patent/DE68927875T2/de not_active Expired - Fee Related
- 1989-12-18 AU AU46889/89A patent/AU634992B2/en not_active Ceased
- 1989-12-18 NO NO895093A patent/NO177672C/no unknown
- 1989-12-19 FI FI896084A patent/FI93951C/fi not_active IP Right Cessation
- 1989-12-19 PT PT92628A patent/PT92628B/pt not_active IP Right Cessation
- 1989-12-19 ZA ZA899736A patent/ZA899736B/xx unknown
- 1989-12-19 CA CA002005919A patent/CA2005919C/en not_active Expired - Fee Related
- 1989-12-19 JP JP1327463A patent/JP2848534B2/ja not_active Expired - Lifetime
-
1997
- 1997-05-09 GR GR970401032T patent/GR3023379T3/el unknown
Also Published As
Publication number | Publication date |
---|---|
NO177672B (no) | 1995-07-24 |
CA2005919C (en) | 1997-01-07 |
FI93951B (fi) | 1995-03-15 |
US5071859A (en) | 1991-12-10 |
DK704488D0 (da) | 1988-12-19 |
DE68927875D1 (de) | 1997-04-24 |
EP0374801A2 (en) | 1990-06-27 |
EP0374801A3 (en) | 1991-08-07 |
FI93951C (fi) | 1995-06-26 |
NO895093L (no) | 1990-06-20 |
NO895093D0 (no) | 1989-12-18 |
IL92652A0 (en) | 1990-08-31 |
DE68927875T2 (de) | 1997-06-26 |
GR3023379T3 (en) | 1997-08-29 |
EP0374801B1 (en) | 1997-03-19 |
AU634992B2 (en) | 1993-03-11 |
ES2099067T3 (es) | 1997-05-16 |
JPH02223551A (ja) | 1990-09-05 |
ZA899736B (en) | 1990-09-26 |
ATE150455T1 (de) | 1997-04-15 |
CA2005919A1 (en) | 1990-06-19 |
JP2848534B2 (ja) | 1999-01-20 |
NO177672C (no) | 1995-11-01 |
FI896084A0 (fi) | 1989-12-19 |
PT92628B (pt) | 1995-09-12 |
NZ231836A (en) | 1992-11-25 |
AU4688989A (en) | 1990-06-21 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FG3A | Patent granted, date of granting |
Effective date: 19950504 |
|
MM3A | Annulment or lapse |
Free format text: LAPSE DUE TO NON-PAYMENT OF FEES Effective date: 20001130 |