PT793671E - Derivados fluor-4-azasteroides substituidos por fenilo - Google Patents
Derivados fluor-4-azasteroides substituidos por fenilo Download PDFInfo
- Publication number
- PT793671E PT793671E PT96928436T PT96928436T PT793671E PT 793671 E PT793671 E PT 793671E PT 96928436 T PT96928436 T PT 96928436T PT 96928436 T PT96928436 T PT 96928436T PT 793671 E PT793671 E PT 793671E
- Authority
- PT
- Portugal
- Prior art keywords
- formula
- compound
- oxo
- aza
- group
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J73/00—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms
- C07J73/001—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom
- C07J73/005—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom by nitrogen as hetero atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/28—Antiandrogens
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Diabetes (AREA)
- Endocrinology (AREA)
- Steroid Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB9518858.7A GB9518858D0 (en) | 1995-09-14 | 1995-09-14 | Phenylsubstituted 4-azasteroid fluoroderivatives |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| PT793671E true PT793671E (pt) | 2000-07-31 |
Family
ID=10780746
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PT96928436T PT793671E (pt) | 1995-09-14 | 1996-08-09 | Derivados fluor-4-azasteroides substituidos por fenilo |
Country Status (28)
| Country | Link |
|---|---|
| US (2) | US5922728A (cs) |
| EP (1) | EP0793671B1 (cs) |
| JP (1) | JPH10509188A (cs) |
| KR (1) | KR100448745B1 (cs) |
| CN (1) | CN1104439C (cs) |
| AR (1) | AR004511A1 (cs) |
| AT (1) | ATE189681T1 (cs) |
| AU (1) | AU715858B2 (cs) |
| BR (1) | BR9606638A (cs) |
| CA (1) | CA2204002A1 (cs) |
| CZ (1) | CZ291450B6 (cs) |
| DE (1) | DE69606623T2 (cs) |
| DK (1) | DK0793671T3 (cs) |
| EA (1) | EA000362B1 (cs) |
| ES (1) | ES2144765T3 (cs) |
| GB (1) | GB9518858D0 (cs) |
| GR (1) | GR3033315T3 (cs) |
| HU (1) | HUP9702038A3 (cs) |
| IL (1) | IL120742A (cs) |
| MY (1) | MY116271A (cs) |
| NO (1) | NO309527B1 (cs) |
| NZ (1) | NZ316060A (cs) |
| PL (1) | PL185196B1 (cs) |
| PT (1) | PT793671E (cs) |
| TW (1) | TW357149B (cs) |
| UA (1) | UA66748C2 (cs) |
| WO (1) | WO1997010257A1 (cs) |
| ZA (1) | ZA967631B (cs) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6054446A (en) * | 1997-12-24 | 2000-04-25 | Sri International | Anti-estrogenic steroids, and associated pharmaceutical compositions and methods of use |
| US6548491B2 (en) * | 1997-12-24 | 2003-04-15 | Sri International | Anti-estrogenic steroids, and associated pharmaceutical compositions and methods of use |
| US7241753B2 (en) | 2000-02-25 | 2007-07-10 | Loria Roger M | Method of treatment of prostate cancer |
| US7402577B2 (en) * | 2001-10-03 | 2008-07-22 | Merck & Co., Inc. | Androstane 17-beta-carboxamides as androgen receptor modulators |
| AU2004255200A1 (en) * | 2003-06-30 | 2005-01-20 | Merck & Co., Inc. | 17-acetamido-4-azasteroid derivatives as androgen receptor modulators |
| WO2005005380A2 (en) * | 2003-06-30 | 2005-01-20 | Merck & Co., Inc. | 17-acetamido-4-azasteroid derivatives as androgen receptor modulators |
| EP1641464A4 (en) * | 2003-06-30 | 2008-05-14 | Merck & Co Inc | 17-ACETAMIDO-4-AZASTEROID DERIVATIVES AS MODULATORS OF THE ANDROGEN RECEPTOR |
| WO2005005606A2 (en) | 2003-06-30 | 2005-01-20 | Merck & Co., Inc. | 17-acetamido-4-azasteroid derivatives as androgen receptor modulators |
| CN103787894B (zh) * | 2014-02-08 | 2015-09-16 | 济南大学 | 从甲苯二异氰酸酯制备过程中形成的残渣废料中回收甲苯二胺的方法 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9002922D0 (en) * | 1990-02-09 | 1990-04-04 | Erba Carlo Spa | 17 beta-substituted-4-aza-5 alpha-androstan-3-one derivatives and process for their preparation |
| GB9216284D0 (en) * | 1992-07-31 | 1992-09-16 | Erba Carlo Spa | Fluorinated 17beta-substituted 4-aza-5alpha-androstane-3-one derivatives |
| GB9216329D0 (en) * | 1992-07-31 | 1992-09-16 | Erba Carlo Spa | 17beta-substituted 4-aza-5alpha-androstan-3-one derivatives |
| GB9608045D0 (en) * | 1996-04-18 | 1996-06-19 | Pharmacia Spa | Process for preparing steroids having a carboxamide side-chain |
| US5686501A (en) * | 1996-04-19 | 1997-11-11 | Foamex L.P. | Breathable open cell urethane polymers |
-
1995
- 1995-09-14 GB GBGB9518858.7A patent/GB9518858D0/en active Pending
-
1996
- 1996-08-09 IL IL12074296A patent/IL120742A/en not_active IP Right Cessation
- 1996-08-09 EA EA199700063A patent/EA000362B1/ru not_active IP Right Cessation
- 1996-08-09 PL PL96320114A patent/PL185196B1/pl not_active IP Right Cessation
- 1996-08-09 CZ CZ19971460A patent/CZ291450B6/cs not_active IP Right Cessation
- 1996-08-09 CA CA002204002A patent/CA2204002A1/en not_active Abandoned
- 1996-08-09 CN CN96191076A patent/CN1104439C/zh not_active Expired - Fee Related
- 1996-08-09 NZ NZ316060A patent/NZ316060A/xx unknown
- 1996-08-09 KR KR1019970703203A patent/KR100448745B1/ko not_active IP Right Cessation
- 1996-08-09 ES ES96928436T patent/ES2144765T3/es not_active Expired - Lifetime
- 1996-08-09 AT AT96928436T patent/ATE189681T1/de not_active IP Right Cessation
- 1996-08-09 DE DE69606623T patent/DE69606623T2/de not_active Expired - Fee Related
- 1996-08-09 BR BR9606638A patent/BR9606638A/pt not_active Application Discontinuation
- 1996-08-09 DK DK96928436T patent/DK0793671T3/da active
- 1996-08-09 EP EP96928436A patent/EP0793671B1/en not_active Expired - Lifetime
- 1996-08-09 PT PT96928436T patent/PT793671E/pt unknown
- 1996-08-09 US US08/836,052 patent/US5922728A/en not_active Expired - Fee Related
- 1996-08-09 JP JP9511593A patent/JPH10509188A/ja not_active Withdrawn
- 1996-08-09 AU AU68205/96A patent/AU715858B2/en not_active Ceased
- 1996-08-09 WO PCT/EP1996/003518 patent/WO1997010257A1/en active IP Right Grant
- 1996-08-09 UA UA97062805A patent/UA66748C2/xx unknown
- 1996-08-09 HU HU9702038A patent/HUP9702038A3/hu unknown
- 1996-09-05 TW TW085110841A patent/TW357149B/zh active
- 1996-09-09 AR ARP960104280A patent/AR004511A1/es unknown
- 1996-09-10 ZA ZA967631A patent/ZA967631B/xx unknown
- 1996-09-13 MY MYPI96003782A patent/MY116271A/en unknown
-
1997
- 1997-05-13 NO NO972186A patent/NO309527B1/no unknown
-
1999
- 1999-04-28 US US09/300,454 patent/US6114345A/en not_active Expired - Fee Related
-
2000
- 2000-04-26 GR GR20000400999T patent/GR3033315T3/el not_active IP Right Cessation
Also Published As
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