DE69606623T2 - Phenyl-substituierte 4-azasteroid-fluorderivate - Google Patents

Phenyl-substituierte 4-azasteroid-fluorderivate

Info

Publication number
DE69606623T2
DE69606623T2 DE69606623T DE69606623T DE69606623T2 DE 69606623 T2 DE69606623 T2 DE 69606623T2 DE 69606623 T DE69606623 T DE 69606623T DE 69606623 T DE69606623 T DE 69606623T DE 69606623 T2 DE69606623 T2 DE 69606623T2
Authority
DE
Germany
Prior art keywords
azasteroid
phenyl
substituted
fluor
derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
DE69606623T
Other languages
English (en)
Other versions
DE69606623D1 (de
Inventor
Achille Panzeri
Marcella Nesi
Salle Enrico Di
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Italia SRL
Original Assignee
Pharmacia and Upjohn SpA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmacia and Upjohn SpA filed Critical Pharmacia and Upjohn SpA
Application granted granted Critical
Publication of DE69606623D1 publication Critical patent/DE69606623D1/de
Publication of DE69606623T2 publication Critical patent/DE69606623T2/de
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J73/00—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms
    • C07J73/001—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom
    • C07J73/005—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom by nitrogen as hetero atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/28—Antiandrogens

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DE69606623T 1995-09-14 1996-08-09 Phenyl-substituierte 4-azasteroid-fluorderivate Expired - Fee Related DE69606623T2 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9518858.7A GB9518858D0 (en) 1995-09-14 1995-09-14 Phenylsubstituted 4-azasteroid fluoroderivatives
PCT/EP1996/003518 WO1997010257A1 (en) 1995-09-14 1996-08-09 Phenylsubstituted 4-azasteroid fluoroderivatives

Publications (2)

Publication Number Publication Date
DE69606623D1 DE69606623D1 (de) 2000-03-16
DE69606623T2 true DE69606623T2 (de) 2000-08-31

Family

ID=10780746

Family Applications (1)

Application Number Title Priority Date Filing Date
DE69606623T Expired - Fee Related DE69606623T2 (de) 1995-09-14 1996-08-09 Phenyl-substituierte 4-azasteroid-fluorderivate

Country Status (28)

Country Link
US (2) US5922728A (de)
EP (1) EP0793671B1 (de)
JP (1) JPH10509188A (de)
KR (1) KR100448745B1 (de)
CN (1) CN1104439C (de)
AR (1) AR004511A1 (de)
AT (1) ATE189681T1 (de)
AU (1) AU715858B2 (de)
BR (1) BR9606638A (de)
CA (1) CA2204002A1 (de)
CZ (1) CZ291450B6 (de)
DE (1) DE69606623T2 (de)
DK (1) DK0793671T3 (de)
EA (1) EA000362B1 (de)
ES (1) ES2144765T3 (de)
GB (1) GB9518858D0 (de)
GR (1) GR3033315T3 (de)
HU (1) HUP9702038A3 (de)
IL (1) IL120742A (de)
MY (1) MY116271A (de)
NO (1) NO309527B1 (de)
NZ (1) NZ316060A (de)
PL (1) PL185196B1 (de)
PT (1) PT793671E (de)
TW (1) TW357149B (de)
UA (1) UA66748C2 (de)
WO (1) WO1997010257A1 (de)
ZA (1) ZA967631B (de)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6548491B2 (en) * 1997-12-24 2003-04-15 Sri International Anti-estrogenic steroids, and associated pharmaceutical compositions and methods of use
US6054446A (en) * 1997-12-24 2000-04-25 Sri International Anti-estrogenic steroids, and associated pharmaceutical compositions and methods of use
AU2001241779A1 (en) 2000-02-25 2001-09-03 Hollis-Eden Pharmaceuticals, Inc. Method of treatment of prostate cancer
CA2462456C (en) * 2001-10-03 2010-05-04 Merck & Co., Inc. Androstane 17-beta-carboxamides as androgen receptor modulators
EP1641761A4 (de) * 2003-06-30 2008-05-14 Merck & Co Inc 17-acetamido-4-azasteroidderivate als androgenrezeptormodulatoren
US7482357B2 (en) 2003-06-30 2009-01-27 Merck & Co., Inc. 17-acetamido-4-azasteroid derivatives as androgen receptor modulators
CN100528168C (zh) * 2003-06-30 2009-08-19 麦克公司 作为雄激素受体调节剂的17-乙酰氨基-4-氮杂甾类衍生物
CA2530025A1 (en) * 2003-06-30 2005-01-20 William P. Dankulich 17-acetamido-4-azasteroid derivatives as androgen receptor modulators
CN103787894B (zh) * 2014-02-08 2015-09-16 济南大学 从甲苯二异氰酸酯制备过程中形成的残渣废料中回收甲苯二胺的方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9002922D0 (en) * 1990-02-09 1990-04-04 Erba Carlo Spa 17 beta-substituted-4-aza-5 alpha-androstan-3-one derivatives and process for their preparation
GB9216284D0 (en) * 1992-07-31 1992-09-16 Erba Carlo Spa Fluorinated 17beta-substituted 4-aza-5alpha-androstane-3-one derivatives
GB9216329D0 (en) * 1992-07-31 1992-09-16 Erba Carlo Spa 17beta-substituted 4-aza-5alpha-androstan-3-one derivatives
GB9608045D0 (en) * 1996-04-18 1996-06-19 Pharmacia Spa Process for preparing steroids having a carboxamide side-chain
US5686501A (en) * 1996-04-19 1997-11-11 Foamex L.P. Breathable open cell urethane polymers

Also Published As

Publication number Publication date
US6114345A (en) 2000-09-05
NO309527B1 (no) 2001-02-12
MY116271A (en) 2003-12-31
EA000362B1 (ru) 1999-06-24
IL120742A (en) 2002-04-21
CN1165520A (zh) 1997-11-19
CA2204002A1 (en) 1997-03-20
ZA967631B (en) 1997-04-16
NO972186L (no) 1997-07-02
US5922728A (en) 1999-07-13
AU715858B2 (en) 2000-02-10
CN1104439C (zh) 2003-04-02
HUP9702038A2 (hu) 1998-03-30
GB9518858D0 (en) 1995-11-15
PL185196B1 (pl) 2003-03-31
GR3033315T3 (en) 2000-09-29
TW357149B (en) 1999-05-01
DK0793671T3 (da) 2000-07-17
WO1997010257A1 (en) 1997-03-20
NZ316060A (en) 1999-08-30
IL120742A0 (en) 1997-08-14
AU6820596A (en) 1997-04-01
DE69606623D1 (de) 2000-03-16
AR004511A1 (es) 1998-12-16
PT793671E (pt) 2000-07-31
PL320114A1 (en) 1997-09-15
EA199700063A1 (ru) 1997-12-30
MX9703464A (es) 1997-07-31
EP0793671A1 (de) 1997-09-10
ATE189681T1 (de) 2000-02-15
CZ291450B6 (cs) 2003-03-12
UA66748C2 (en) 2004-06-15
KR100448745B1 (ko) 2004-12-14
ES2144765T3 (es) 2000-06-16
BR9606638A (pt) 1997-11-11
NO972186D0 (no) 1997-05-13
HUP9702038A3 (en) 1998-11-30
CZ146097A3 (en) 1997-10-15
JPH10509188A (ja) 1998-09-08
EP0793671B1 (de) 2000-02-09

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Legal Events

Date Code Title Description
8364 No opposition during term of opposition
8339 Ceased/non-payment of the annual fee