PT3452463T - Derivados de piridiniltriazol substituído com amida e utilizações dos mesmos - Google Patents

Derivados de piridiniltriazol substituído com amida e utilizações dos mesmos

Info

Publication number
PT3452463T
PT3452463T PT177201472T PT17720147T PT3452463T PT 3452463 T PT3452463 T PT 3452463T PT 177201472 T PT177201472 T PT 177201472T PT 17720147 T PT17720147 T PT 17720147T PT 3452463 T PT3452463 T PT 3452463T
Authority
PT
Portugal
Prior art keywords
pyridinyltriazole
amide
derivatives
substituted
substituted pyridinyltriazole
Prior art date
Application number
PT177201472T
Other languages
English (en)
Original Assignee
Bayer Pharma AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Pharma AG filed Critical Bayer Pharma AG
Publication of PT3452463T publication Critical patent/PT3452463T/pt

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/08Drugs for disorders of the urinary system of the prostate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/10Drugs for disorders of the urinary system of the bladder
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/12Drugs for disorders of the urinary system of the kidneys
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/02Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • A61P27/06Antiglaucoma agents or miotics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/04Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/06Antiarrhythmics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
PT177201472T 2016-05-03 2017-05-02 Derivados de piridiniltriazol substituído com amida e utilizações dos mesmos PT3452463T (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP16168165 2016-05-03

Publications (1)

Publication Number Publication Date
PT3452463T true PT3452463T (pt) 2021-04-28

Family

ID=55910850

Family Applications (1)

Application Number Title Priority Date Filing Date
PT177201472T PT3452463T (pt) 2016-05-03 2017-05-02 Derivados de piridiniltriazol substituído com amida e utilizações dos mesmos

Country Status (42)

Country Link
US (4) US9988367B2 (pt)
EP (1) EP3452463B1 (pt)
JP (1) JP6932140B2 (pt)
KR (1) KR20190003655A (pt)
CN (2) CN109415347B (pt)
AR (1) AR108262A1 (pt)
AU (1) AU2017259870B2 (pt)
BR (1) BR112018072542A2 (pt)
CA (1) CA3022749A1 (pt)
CL (1) CL2018003105A1 (pt)
CO (1) CO2018011933A2 (pt)
CR (1) CR20180522A (pt)
CU (1) CU24567B1 (pt)
CY (1) CY1124084T1 (pt)
DK (1) DK3452463T3 (pt)
DO (1) DOP2018000240A (pt)
EA (1) EA035596B1 (pt)
EC (1) ECSP18081881A (pt)
ES (1) ES2866109T3 (pt)
GE (1) GEP20207158B (pt)
HR (1) HRP20210648T1 (pt)
HU (1) HUE053908T2 (pt)
IL (1) IL262557B (pt)
JO (1) JOP20170105B1 (pt)
LT (1) LT3452463T (pt)
MA (1) MA44851B1 (pt)
MX (1) MX2018013335A (pt)
NI (1) NI201800115A (pt)
PE (1) PE20190116A1 (pt)
PH (1) PH12018502268A1 (pt)
PL (1) PL3452463T3 (pt)
PT (1) PT3452463T (pt)
RS (1) RS61771B1 (pt)
SG (1) SG11201809752VA (pt)
SI (1) SI3452463T1 (pt)
SV (1) SV2018005771A (pt)
TN (1) TN2018000368A1 (pt)
TW (1) TWI772295B (pt)
UA (1) UA123791C2 (pt)
UY (1) UY37220A (pt)
WO (1) WO2017191102A1 (pt)
ZA (1) ZA201808131B (pt)

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Also Published As

Publication number Publication date
SV2018005771A (es) 2019-01-04
TWI772295B (zh) 2022-08-01
DOP2018000240A (es) 2019-03-15
CN113121504A (zh) 2021-07-16
US9988367B2 (en) 2018-06-05
TN2018000368A1 (en) 2020-06-15
TW201806941A (zh) 2018-03-01
IL262557A (en) 2018-12-31
RS61771B1 (sr) 2021-05-31
EP3452463B1 (en) 2021-03-24
LT3452463T (lt) 2021-04-26
ES2866109T3 (es) 2021-10-19
GEP20207158B (en) 2020-10-12
CU24567B1 (es) 2022-01-13
US20200017473A1 (en) 2020-01-16
MX2018013335A (es) 2019-05-09
CL2018003105A1 (es) 2019-02-15
AU2017259870B2 (en) 2021-07-15
MA44851B1 (fr) 2021-09-30
MA44851A (fr) 2019-03-13
EA201892505A1 (ru) 2019-04-30
JP6932140B2 (ja) 2021-09-08
UA123791C2 (uk) 2021-06-02
UY37220A (es) 2017-11-30
PL3452463T3 (pl) 2021-08-09
JOP20170105B1 (ar) 2022-03-14
US20180251447A1 (en) 2018-09-06
NI201800115A (es) 2019-03-14
WO2017191102A1 (en) 2017-11-09
HUE053908T2 (hu) 2021-07-28
CN109415347A (zh) 2019-03-01
US20170320854A1 (en) 2017-11-09
EA035596B1 (ru) 2020-07-14
CA3022749A1 (en) 2017-11-09
CY1124084T1 (el) 2022-05-27
DK3452463T3 (da) 2021-04-26
SG11201809752VA (en) 2018-12-28
HRP20210648T1 (hr) 2021-05-28
SI3452463T1 (sl) 2021-07-30
ZA201808131B (en) 2021-05-26
BR112018072542A2 (pt) 2019-03-26
EP3452463A1 (en) 2019-03-13
US20190144423A1 (en) 2019-05-16
JP2019514945A (ja) 2019-06-06
PE20190116A1 (es) 2019-01-16
IL262557B (en) 2022-01-01
ECSP18081881A (es) 2018-11-30
CR20180522A (es) 2019-01-15
US11091463B2 (en) 2021-08-17
AR108262A1 (es) 2018-08-01
US10472348B2 (en) 2019-11-12
CO2018011933A2 (es) 2018-11-22
CN109415347B (zh) 2021-05-07
AU2017259870A1 (en) 2018-11-15
KR20190003655A (ko) 2019-01-09
CU20180134A7 (es) 2019-06-04
PH12018502268A1 (en) 2019-07-15

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