PT3074384T - Derivados de amida para o agonista gpr119 - Google Patents
Derivados de amida para o agonista gpr119Info
- Publication number
- PT3074384T PT3074384T PT14866648T PT14866648T PT3074384T PT 3074384 T PT3074384 T PT 3074384T PT 14866648 T PT14866648 T PT 14866648T PT 14866648 T PT14866648 T PT 14866648T PT 3074384 T PT3074384 T PT 3074384T
- Authority
- PT
- Portugal
- Prior art keywords
- amide derivatives
- gpr119 agonist
- gpr119
- agonist
- amide
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
- A61K31/454—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/4965—Non-condensed pyrazines
- A61K31/497—Non-condensed pyrazines containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Diabetes (AREA)
- Epidemiology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Endocrinology (AREA)
- Emergency Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
KR20130144601 | 2013-11-26 |
Publications (1)
Publication Number | Publication Date |
---|---|
PT3074384T true PT3074384T (pt) | 2019-07-10 |
Family
ID=53199342
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PT14866648T PT3074384T (pt) | 2013-11-26 | 2014-11-25 | Derivados de amida para o agonista gpr119 |
Country Status (20)
Country | Link |
---|---|
US (1) | US9776987B2 (pt) |
EP (1) | EP3074384B1 (pt) |
JP (1) | JP6182269B2 (pt) |
KR (1) | KR101700906B1 (pt) |
CN (2) | CN105873916B (pt) |
AU (1) | AU2014354488B2 (pt) |
BR (1) | BR112016011999A2 (pt) |
CA (1) | CA2930850C (pt) |
DK (1) | DK3074384T3 (pt) |
ES (1) | ES2731823T3 (pt) |
HR (1) | HRP20191246T1 (pt) |
HU (1) | HUE045926T2 (pt) |
MX (1) | MX366297B (pt) |
NZ (1) | NZ720304A (pt) |
PH (1) | PH12016500980B1 (pt) |
PL (1) | PL3074384T3 (pt) |
PT (1) | PT3074384T (pt) |
RU (1) | RU2642429C2 (pt) |
TR (1) | TR201908098T4 (pt) |
WO (1) | WO2015080446A1 (pt) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA3178994A1 (en) | 2020-05-19 | 2021-11-25 | Iyassu Sebhat | Ampk activators |
JP2023531726A (ja) | 2020-06-26 | 2023-07-25 | キャリーオペ,インク. | Ampkアクチベーター |
Family Cites Families (25)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5109002A (en) | 1989-09-08 | 1992-04-28 | Du Pont Merck Pharmaceutical Company | Antipsychotic 1-cycloalkylpiperidines |
ES2204409T5 (es) | 2000-06-26 | 2008-04-16 | Saudi Basic Industries Corporation | Dimerizacion de isobuteno. |
EP1299334B1 (en) | 2000-07-13 | 2008-01-16 | MERCK PATENT GmbH | Chiral compounds i |
AU2002212282A1 (en) | 2000-10-20 | 2002-05-06 | Merck Patent G.M.B.H | Chiral binaphthol derivatives |
DE102004037515A1 (de) | 2003-08-22 | 2005-03-17 | Merck Patent Gmbh | Verfahren zur Herstellung von Aldehyden |
JP2010501629A (ja) * | 2006-08-30 | 2010-01-21 | ビオヴィトルム・アクチボラゲット(プブリクト) | Gpr119関連障害を治療するためのピリジン化合物 |
JP5330260B2 (ja) | 2006-12-06 | 2013-10-30 | スミスクライン ビーチャム コーポレーション | 二環式化合物ならびに抗糖尿病薬としての使用 |
PL2114933T3 (pl) | 2007-01-04 | 2012-02-29 | Prosidion Ltd | Piperydyny jako agoniści GPCR |
AU2008279447A1 (en) | 2007-07-19 | 2009-01-29 | Metabolex, Inc. | N-azacyclic substituted pyrrole, pyrazole, imidazole, triazole and tetrazole derivatives as agonists of the RUP3 or GPR119 receptor for the treatment of diabetes and metabolic disorders |
ES2499018T3 (es) | 2007-09-20 | 2014-09-26 | Irm Llc | Compuestos y composiciones como moduladores de la actividad de GPR119 |
WO2009106565A1 (en) | 2008-02-27 | 2009-09-03 | Biovitrum Ab (Publ) | Agonists of gpr119 |
WO2009106561A1 (en) * | 2008-02-27 | 2009-09-03 | Biovitrum Ab (Publ) | Pyrazine compounds for treating gpr119 related disorders |
JP5309216B2 (ja) * | 2008-07-11 | 2013-10-09 | アイアールエム・リミテッド・ライアビリティ・カンパニー | Gpr119活性のモジュレーターとしての4−フェノキシメチルピペリジン類 |
WO2010048149A2 (en) | 2008-10-20 | 2010-04-29 | Kalypsys, Inc. | Heterocyclic modulators of gpr119 for treatment of disease |
AR077642A1 (es) | 2009-07-09 | 2011-09-14 | Arena Pharm Inc | Moduladores del metabolismo y el tratamiento de trastornos relacionados con el mismo |
AR077638A1 (es) * | 2009-07-15 | 2011-09-14 | Lilly Co Eli | Compuesto de (metanosulfonil -piperidin )-( alcoxi-aril) -tetrahidro- piridina , composicion farmaceutica que lo comprende y su uso para preparar un medicamento util para el tratamiento de diabetes u obesidad |
JP2013523819A (ja) * | 2010-04-06 | 2013-06-17 | アリーナ ファーマシューティカルズ, インコーポレイテッド | Gpr119レセプターのモジュレーターおよびそれに関連する障害の処置 |
WO2011145718A1 (ja) * | 2010-05-21 | 2011-11-24 | 田辺三菱製薬株式会社 | 新規ピロロ[2,3-d]ピリミジン化合物 |
TW201202230A (en) * | 2010-05-24 | 2012-01-16 | Mitsubishi Tanabe Pharma Corp | Novel quinazoline compound |
CN102432598A (zh) | 2010-09-29 | 2012-05-02 | 江苏恒瑞医药股份有限公司 | 三环化合物、其制备方法及其在医药上的应用 |
AU2011333472A1 (en) * | 2010-11-26 | 2013-06-06 | Lupin Limited | Bicyclic GPR119 modulators |
WO2012077655A1 (ja) | 2010-12-07 | 2012-06-14 | 塩野義製薬株式会社 | Gpr119アゴニスト活性を有するスピロ誘導体 |
JP2014159376A (ja) * | 2011-06-17 | 2014-09-04 | Taisho Pharmaceutical Co Ltd | アザスピロアルカン化合物 |
ES2759010T3 (es) * | 2012-06-12 | 2020-05-07 | Chong Kun Dang Pharmaceutical Corp | Derivados de piperidina como agonistas del GPR119 |
EP2862763B1 (en) * | 2012-06-13 | 2015-12-09 | Nissan Motor Co., Ltd. | Driving force controller for vehicle |
-
2014
- 2014-11-25 PT PT14866648T patent/PT3074384T/pt unknown
- 2014-11-25 HU HUE14866648A patent/HUE045926T2/hu unknown
- 2014-11-25 BR BR112016011999A patent/BR112016011999A2/pt active Search and Examination
- 2014-11-25 DK DK14866648.0T patent/DK3074384T3/da active
- 2014-11-25 MX MX2016006904A patent/MX366297B/es active IP Right Grant
- 2014-11-25 ES ES14866648T patent/ES2731823T3/es active Active
- 2014-11-25 TR TR2019/08098T patent/TR201908098T4/tr unknown
- 2014-11-25 US US15/039,226 patent/US9776987B2/en active Active
- 2014-11-25 AU AU2014354488A patent/AU2014354488B2/en not_active Ceased
- 2014-11-25 CN CN201480064763.0A patent/CN105873916B/zh not_active Expired - Fee Related
- 2014-11-25 CN CN201910451096.6A patent/CN110028494A/zh active Pending
- 2014-11-25 JP JP2016534127A patent/JP6182269B2/ja not_active Expired - Fee Related
- 2014-11-25 PL PL14866648T patent/PL3074384T3/pl unknown
- 2014-11-25 NZ NZ720304A patent/NZ720304A/en not_active IP Right Cessation
- 2014-11-25 WO PCT/KR2014/011356 patent/WO2015080446A1/en active Application Filing
- 2014-11-25 CA CA2930850A patent/CA2930850C/en not_active Expired - Fee Related
- 2014-11-25 EP EP14866648.0A patent/EP3074384B1/en active Active
- 2014-11-25 RU RU2016125492A patent/RU2642429C2/ru active
- 2014-11-25 KR KR1020140164986A patent/KR101700906B1/ko active IP Right Grant
-
2016
- 2016-05-26 PH PH12016500980A patent/PH12016500980B1/en unknown
-
2019
- 2019-07-11 HR HRP20191246TT patent/HRP20191246T1/hr unknown
Also Published As
Publication number | Publication date |
---|---|
JP2016538296A (ja) | 2016-12-08 |
EP3074384B1 (en) | 2019-05-22 |
PH12016500980A1 (en) | 2016-06-20 |
CA2930850C (en) | 2017-05-16 |
AU2014354488A1 (en) | 2016-06-09 |
US20170129875A1 (en) | 2017-05-11 |
MX366297B (es) | 2019-07-04 |
KR20150060573A (ko) | 2015-06-03 |
CN110028494A (zh) | 2019-07-19 |
MX2016006904A (es) | 2016-10-28 |
KR101700906B1 (ko) | 2017-01-31 |
PL3074384T3 (pl) | 2019-09-30 |
CN105873916A (zh) | 2016-08-17 |
CA2930850A1 (en) | 2015-06-04 |
EP3074384A1 (en) | 2016-10-05 |
PH12016500980B1 (en) | 2016-06-20 |
ES2731823T3 (es) | 2019-11-19 |
TR201908098T4 (tr) | 2019-06-21 |
HRP20191246T1 (hr) | 2019-12-27 |
DK3074384T3 (da) | 2019-07-15 |
JP6182269B2 (ja) | 2017-08-16 |
RU2016125492A (ru) | 2018-01-09 |
RU2642429C2 (ru) | 2018-01-25 |
WO2015080446A1 (en) | 2015-06-04 |
NZ720304A (en) | 2017-08-25 |
CN105873916B (zh) | 2019-08-27 |
AU2014354488B2 (en) | 2017-08-24 |
BR112016011999A2 (pt) | 2017-08-08 |
EP3074384A4 (en) | 2017-04-19 |
US9776987B2 (en) | 2017-10-03 |
HUE045926T2 (hu) | 2020-01-28 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
HK1215795A1 (zh) | 鵝膏毒素衍生物 | |
SG11201506100XA (en) | Pyridazinone-amides derivatives | |
EP2858986A4 (en) | GPR119 AGONIST PIPERIDINE DERIVATIVES | |
ZA201601333B (en) | Oxoquinazolinyl-butanamide derivatives | |
IL245737B (en) | Glucosylceramide synthase inhibitors | |
EP3006444A4 (en) | HETEROCYCLIC AMIDE COMPOUND | |
SG11201605189YA (en) | Imidazopyrazinone derivatives | |
GB2510914B (en) | Cases for cigarette packets | |
PL3074384T3 (pl) | Pochodne amidowe dla agonisty gpr119 | |
IL243730A0 (en) | Vasopressin-2 receptor agonists | |
PL2981678T3 (pl) | Przyrząd przytrzymujący | |
GB201312010D0 (en) | Receptor Agonists | |
GB201309343D0 (en) | Device for holding apparel | |
TH1601003052A (th) | อนุพันธ์เอไมด์ สำหรับ gpr119 อะโกนิสต์ | |
GB201304105D0 (en) | Agonist | |
TH1401007264A (th) | อนุพันธ์พิเพอริดีน สำหรับเป็น gpr119 อะโกนิสท์ | |
GB201313108D0 (en) | Peptide agonist | |
TWM475331U (en) | Unclamping cylinder device |