PT2270005E - Pró-fármaco de um inibidor de ice - Google Patents
Pró-fármaco de um inibidor de ice Download PDFInfo
- Publication number
- PT2270005E PT2270005E PT101775377T PT10177537T PT2270005E PT 2270005 E PT2270005 E PT 2270005E PT 101775377 T PT101775377 T PT 101775377T PT 10177537 T PT10177537 T PT 10177537T PT 2270005 E PT2270005 E PT 2270005E
- Authority
- PT
- Portugal
- Prior art keywords
- prodrug
- ice inhibitor
- inhibitor
- ice
- Prior art date
Links
- 101000828805 Cowpox virus (strain Brighton Red) Serine proteinase inhibitor 2 Proteins 0.000 title 1
- 229940002612 prodrug Drugs 0.000 title 1
- 239000000651 prodrug Substances 0.000 title 1
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- C07K5/06—Dipeptides
- C07K5/06008—Dipeptides with the first amino acid being neutral
- C07K5/06017—Dipeptides with the first amino acid being neutral and aliphatic
- C07K5/06034—Dipeptides with the first amino acid being neutral and aliphatic the side chain containing 2 to 4 carbon atoms
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- C07—ORGANIC CHEMISTRY
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- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06008—Dipeptides with the first amino acid being neutral
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06191—Dipeptides containing heteroatoms different from O, S, or N
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/08—Tripeptides
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/08—Tripeptides
- C07K5/0802—Tripeptides with the first amino acid being neutral
- C07K5/0804—Tripeptides with the first amino acid being neutral and aliphatic
- C07K5/0808—Tripeptides with the first amino acid being neutral and aliphatic the side chain containing 2 to 4 carbon atoms, e.g. Val, Ile, Leu
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
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- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
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2001
- 2001-05-15 PE PE2001000436A patent/PE20011350A1/es not_active Application Discontinuation
- 2001-05-18 ES ES01939230T patent/ES2380915T3/es not_active Expired - Lifetime
- 2001-05-18 AT AT01939230T patent/ATE543814T1/de active
- 2001-05-18 EP EP01939230A patent/EP1286989B1/en not_active Expired - Lifetime
- 2001-05-18 US US09/860,750 patent/US7417029B2/en not_active Expired - Lifetime
- 2001-05-18 SK SK102-2002A patent/SK287070B6/sk not_active IP Right Cessation
- 2001-05-18 ES ES10177537.7T patent/ES2548869T3/es not_active Expired - Lifetime
- 2001-05-18 DK DK01939230.7T patent/DK1286989T3/da active
- 2001-05-18 EP EP10177537.7A patent/EP2270005B1/en not_active Expired - Lifetime
- 2001-05-18 EP EP03020900A patent/EP1396492B1/en not_active Expired - Lifetime
- 2001-05-18 AP APAP/P/2002/002406A patent/AP2002002406A0/en unknown
- 2001-05-18 PL PL365171A patent/PL207575B1/pl unknown
- 2001-05-18 PT PT01939230T patent/PT1286989E/pt unknown
- 2001-05-18 WO PCT/US2001/016441 patent/WO2001090063A2/en active IP Right Grant
- 2001-05-18 CA CA002379972A patent/CA2379972C/en not_active Expired - Lifetime
- 2001-05-18 JP JP2001586252A patent/JP4890719B2/ja not_active Expired - Lifetime
- 2001-05-18 KR KR1020027000779A patent/KR100863144B1/ko active IP Right Grant
- 2001-05-18 NZ NZ516703A patent/NZ516703A/en not_active IP Right Cessation
- 2001-05-18 AU AU2001264770A patent/AU2001264770A1/en not_active Abandoned
- 2001-05-18 DK DK10177537.7T patent/DK2270005T3/en active
- 2001-05-18 PT PT101775377T patent/PT2270005E/pt unknown
- 2001-05-18 MX MXPA02000751A patent/MXPA02000751A/es active IP Right Grant
- 2001-05-18 TR TR2002/00769T patent/TR200200769T1/xx unknown
- 2001-06-12 TW TW090111976A patent/TWI285642B/zh not_active IP Right Cessation
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2002
- 2002-01-18 NO NO20020287A patent/NO324354B1/no not_active IP Right Cessation
- 2002-01-23 ZA ZA200200610A patent/ZA200200610B/xx unknown
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2004
- 2004-05-28 HK HK04103839.5A patent/HK1060881A1/xx not_active IP Right Cessation
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2008
- 2008-07-01 US US12/165,838 patent/US8022041B2/en not_active Expired - Fee Related
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2011
- 2011-07-25 JP JP2011162436A patent/JP5285130B2/ja not_active Expired - Lifetime
- 2011-08-16 US US13/210,712 patent/US8329662B2/en not_active Expired - Lifetime
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2012
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- 2012-12-10 US US13/709,610 patent/US9156880B2/en not_active Expired - Fee Related
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2015
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2016
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2018
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