PT1888080E - Composiães farmacuticas de um esterëide neuroactivo e as suas utilizaães - Google Patents
Composiães farmacuticas de um esterëide neuroactivo e as suas utilizaães Download PDFInfo
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- PT1888080E PT1888080E PT06754274T PT06754274T PT1888080E PT 1888080 E PT1888080 E PT 1888080E PT 06754274 T PT06754274 T PT 06754274T PT 06754274 T PT06754274 T PT 06754274T PT 1888080 E PT1888080 E PT 1888080E
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- pregnan
- imidazolyl
- methoxymethyl
- pharmaceutical composition
- hydroxy
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Classifications
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Landscapes
- Health & Medical Sciences (AREA)
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Steroid Compounds (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
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| US68890505P | 2005-06-09 | 2005-06-09 |
Publications (1)
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| PT1888080E true PT1888080E (pt) | 2010-07-06 |
Family
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| PT10000305T PT2168585E (pt) | 2005-06-09 | 2006-06-09 | Composições farmacêuticas de um esteróide neuroactivo e as suas utilizações |
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| US (2) | US20090131383A1 (de) |
| EP (3) | EP1888080B1 (de) |
| JP (2) | JP2008542419A (de) |
| KR (3) | KR20100095661A (de) |
| CN (1) | CN101193640A (de) |
| AT (2) | ATE464054T1 (de) |
| AU (1) | AU2006256851C1 (de) |
| BR (1) | BRPI0612921A2 (de) |
| CA (1) | CA2611430C (de) |
| CY (2) | CY1110199T1 (de) |
| DE (1) | DE602006013622D1 (de) |
| DK (2) | DK1888080T3 (de) |
| EA (1) | EA013744B1 (de) |
| ES (2) | ES2344313T3 (de) |
| HK (2) | HK1140947A1 (de) |
| HR (2) | HRP20100372T1 (de) |
| IL (3) | IL187813A (de) |
| NO (1) | NO20076319L (de) |
| NZ (1) | NZ562979A (de) |
| PL (2) | PL1888080T3 (de) |
| PT (2) | PT1888080E (de) |
| RS (2) | RS52199B (de) |
| SI (2) | SI1888080T1 (de) |
| UA (1) | UA94909C2 (de) |
| WO (1) | WO2006131392A1 (de) |
| ZA (1) | ZA200709188B (de) |
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| US20150291654A1 (en) | 2011-10-14 | 2015-10-15 | Sage Therapeutics, Inc. | 3,3 disubstituted 19-nor pregnane compounds, compositions, and uses thereof |
| EP2986624B1 (de) | 2013-04-17 | 2020-03-25 | Sage Therapeutics, Inc. | Neuroaktive 19-nor-steroide zur verwendung zur behandlung von krankheiten |
| EP3909966A1 (de) | 2013-04-17 | 2021-11-17 | Sage Therapeutics, Inc. | 19-nor c3,3-disubstituiertes c21-n-pyrazolyl-steroid zur verwendung in der therapie |
| WO2014169831A1 (en) | 2013-04-17 | 2014-10-23 | Sage Therapeutics, Inc. | 19-nor c3,3-disubstituted c21-c-bound heteroaryl steroids and methods of use thereof |
| US20160068563A1 (en) | 2013-04-17 | 2016-03-10 | Boyd L. Harrison | 19-nor neuroactive steroids and methods of use thereof |
| RS61733B1 (sr) | 2013-07-19 | 2021-05-31 | Sage Therapeutics Inc | Neuroaktivni steroidi, njihove kompozicije i upotrebe |
| PT3488852T (pt) | 2013-08-23 | 2021-02-03 | Sage Therapeutics Inc | Esteroides neuroativos, composições e seus usos |
| WO2015195962A1 (en) | 2014-06-18 | 2015-12-23 | Sage Therapeutics, Inc. | Neuroactive steroids, compositions, and uses thereof |
| NZ731034A (en) * | 2014-10-16 | 2024-02-23 | Sage Therapeutics Inc | Compositions and methods for treating cns disorders |
| NZ731095A (en) | 2014-10-16 | 2023-12-22 | Sage Therapeutics Inc | Compositions and methods for treating cns disorders |
| HUE049014T2 (hu) | 2014-11-27 | 2020-09-28 | Sage Therapeutics Inc | Készítmények és módszerek a központi idegrendszer rendellenességeinek kezelésére |
| JP6745274B2 (ja) | 2015-01-26 | 2020-08-26 | セージ セラピューティクス， インコーポレイテッド | Ｃｎｓ障害を処置するための組成物および方法 |
| US10329320B2 (en) | 2015-02-20 | 2019-06-25 | Sage Therapeutics, Inc. | Neuroactive steroids, compositions, and uses thereof |
| EP3481845B1 (de) | 2016-07-11 | 2023-09-13 | Sage Therapeutics, Inc. | C17-, c20- und c21-substituierte neuroaktive steroide und deren verfahren zur verwendung |
| CN117771252A (zh) * | 2017-09-07 | 2024-03-29 | 萨奇治疗股份有限公司 | 神经活性甾类及其使用方法 |
| US10562930B1 (en) * | 2018-08-31 | 2020-02-18 | Praxis Precision Medicines, Inc. | Salts and crystal forms of GABAA positive allosteric modulator |
| CN113226326A (zh) * | 2018-12-17 | 2021-08-06 | 细胞内治疗公司 | 有机化合物 |
| CN113891715A (zh) * | 2019-03-04 | 2022-01-04 | 普拉西斯精密医药公司 | 围绝经期和绝经期的治疗方法 |
| JOP20210293A1 (ar) | 2019-05-31 | 2023-01-30 | Sage Therapeutics Inc | ستيرويدات ذات فعالية عصبية وتركيبات منها |
| WO2021067702A1 (en) * | 2019-10-02 | 2021-04-08 | Praxis Precision Medicines, Inc. | Combinations of gaba-a receptor positive allosteric modulators and nmda antagonists, nmda negative allosteric modulators or nmda partial agonists |
| WO2021168106A1 (en) * | 2020-02-18 | 2021-08-26 | Praxis Precision Medicines, Inc. | Deuterated neurosteroid |
| WO2022177718A1 (en) | 2021-02-18 | 2022-08-25 | Sage Therapeutics, Inc. | Use of neuroactive steroid for treatment of sexual dysfunction |
| WO2022178000A1 (en) * | 2021-02-18 | 2022-08-25 | Praxis Precision Medicines, Inc. | Hemi-citrate salts of gaba-a positive allosteric modulator and crystalline form thereof |
| WO2022232104A1 (en) * | 2021-04-26 | 2022-11-03 | Praxis Precision Medicines, Inc. | Methods of treatment with neuroactive steroids |
| WO2023159035A1 (en) | 2022-02-16 | 2023-08-24 | Sage Therapeutics, Inc. | Neuroactive steroids for treatment of cns-related disorders |
| WO2023159094A2 (en) * | 2022-02-16 | 2023-08-24 | Praxis Precision Medicines, Inc. | PROCESS OF MAKING 3α-HYDROXY-3β-METHOXYMETHYL-21-(1'- IMIDAZOLYL)-5α-PREGNAN-20-ONE |
| WO2023164386A1 (en) | 2022-02-28 | 2023-08-31 | Sage Therapeutics, Inc. | Neuroactive steroids for treatment of gastrointestinal diseases or conditions |
Family Cites Families (14)
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|---|---|---|---|---|
| FR2535202B1 (fr) * | 1982-11-03 | 1985-08-09 | Fabre Sa Pierre | Comprimes de theophylline a liberation controlee et leur procede de fabrication |
| US4861598A (en) * | 1986-07-18 | 1989-08-29 | Euroceltique, S.A. | Controlled release bases for pharmaceuticals |
| GB8626098D0 (en) * | 1986-10-31 | 1986-12-03 | Euro Celtique Sa | Controlled release hydromorphone composition |
| US4884909A (en) | 1986-12-25 | 1989-12-05 | Canon Kabushiki Kaisha | Recording apparatus |
| US5939545A (en) * | 1994-02-14 | 1999-08-17 | Cocensys, Inc. | Method, compositions, and compounds for allosteric modulation of the gaba receptor by members of the androstane and pregnane series |
| JP4066272B2 (ja) * | 1994-02-14 | 2008-03-26 | ユーロ‐セルティック エス． ア． | Ｇａｂａ受容体のアロステリックな調節のためのアンドロスタン及びプレグナン類 |
| US5478572A (en) * | 1994-09-06 | 1995-12-26 | Bristol-Myers Squibb Co. | Gepirone dosage form |
| US5965161A (en) * | 1994-11-04 | 1999-10-12 | Euro-Celtique, S.A. | Extruded multi-particulates |
| US7083808B2 (en) * | 1998-12-17 | 2006-08-01 | Euro-Celtique S.A. | Controlled/modified release oral methylphenidate formulations |
| EP1177206A1 (de) * | 1999-04-29 | 2002-02-06 | Purdue Pharma Ltd. | 3alpha-hydroxy-3beta methoxymethyl-21-heterozyklish substituierte steroide mit anesthetische aktivität |
| CO5210862A1 (es) * | 1999-09-15 | 2002-10-30 | Alza Corp | Formas de dosificacion y metodos para proporcionar efectiva terapia de reboxetina con dosificacion de una vez al dia |
| US6080736A (en) * | 1999-10-27 | 2000-06-27 | Janus Pharmaceuticals, Inc. | Methods and compositions for treating and preventing anxiety and anxiety disorders using optically pure (R) tofisopam |
| GB0218876D0 (en) * | 2002-08-13 | 2002-09-25 | Merck Sharp & Dohme | Therapeutic agents |
| US20060074059A1 (en) * | 2004-08-26 | 2006-04-06 | Goliber Philip A | Isomorphic crystalline habits of 3alpha-hydroxy-21-(1'-imidazolyl)-3beta-methoxymethyl-5alpha-pregnane-20-one |
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2007
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2008
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-
2010
- 2010-07-02 HR HR20100372T patent/HRP20100372T1/hr unknown
- 2010-07-09 CY CY20101100642T patent/CY1110199T1/el unknown
-
2011
- 2011-02-08 IL IL211114A patent/IL211114A/en not_active IP Right Cessation
- 2011-11-07 IL IL216194A patent/IL216194A/en not_active IP Right Cessation
-
2012
- 2012-03-21 CY CY20121100298T patent/CY1112499T1/el unknown
- 2012-03-23 HR HR20120264T patent/HRP20120264T1/hr unknown
- 2012-05-04 US US13/464,369 patent/US20120276196A1/en not_active Abandoned
- 2012-07-23 JP JP2012162303A patent/JP2012229261A/ja active Pending
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