PT1761533E - 1-aza-biciclo[3.3.1] nonanos - Google Patents

1-aza-biciclo[3.3.1] nonanos Download PDF

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Publication number
PT1761533E
PT1761533E PT05771214T PT05771214T PT1761533E PT 1761533 E PT1761533 E PT 1761533E PT 05771214 T PT05771214 T PT 05771214T PT 05771214 T PT05771214 T PT 05771214T PT 1761533 E PT1761533 E PT 1761533E
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PT
Portugal
Prior art keywords
nonanes
aza
bicyclo
Prior art date
Application number
PT05771214T
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English (en)
Inventor
Thomas J Troxler
Konstanze Hurth
Dominik Feuerbach
Werner Mueller
Bernard Lucien Roy
Mathias Frederiksen
Original Assignee
Novartis Ag
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Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of PT1761533E publication Critical patent/PT1761533E/pt

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/08—Bridged systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/439—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom the ring forming part of a bridged ring system, e.g. quinuclidine
    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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    • A61P9/06—Antiarrhythmics
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    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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    • A61P9/12—Antihypertensives
PT05771214T 2004-06-18 2005-06-17 1-aza-biciclo[3.3.1] nonanos PT1761533E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US58102004P 2004-06-18 2004-06-18

Publications (1)

Publication Number Publication Date
PT1761533E true PT1761533E (pt) 2011-06-01

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Family Applications (1)

Application Number Title Priority Date Filing Date
PT05771214T PT1761533E (pt) 2004-06-18 2005-06-17 1-aza-biciclo[3.3.1] nonanos

Country Status (33)

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US (3) US20070249657A1 (pt)
EP (2) EP1761533B8 (pt)
JP (1) JP4944772B2 (pt)
KR (3) KR20120047317A (pt)
CN (1) CN1964968A (pt)
AR (1) AR049401A1 (pt)
AT (1) ATE506362T1 (pt)
AU (1) AU2005254689B2 (pt)
BR (1) BRPI0510940A (pt)
CA (1) CA2566155C (pt)
CY (1) CY1111528T1 (pt)
DE (1) DE602005027567D1 (pt)
DK (1) DK1761533T3 (pt)
EC (1) ECSP067053A (pt)
ES (1) ES2364971T3 (pt)
HK (1) HK1107559A1 (pt)
HR (1) HRP20110535T1 (pt)
IL (2) IL179611A (pt)
MA (1) MA28684B1 (pt)
MX (1) MXPA06014697A (pt)
MY (1) MY147262A (pt)
NO (1) NO20070339L (pt)
NZ (1) NZ551198A (pt)
PE (1) PE20060437A1 (pt)
PL (1) PL1761533T3 (pt)
PT (1) PT1761533E (pt)
RU (1) RU2445313C2 (pt)
SG (1) SG153834A1 (pt)
SI (1) SI1761533T1 (pt)
TN (1) TNSN06407A1 (pt)
TW (1) TWI370128B (pt)
WO (1) WO2005123732A1 (pt)
ZA (1) ZA200609255B (pt)

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JO3766B1 (ar) 2011-10-20 2021-01-31 Novartis Ag منشط مستقبل أسيتيل كولين الفا - 7 النيكوتيني
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WO2014111751A1 (en) 2013-01-15 2014-07-24 Novartis Ag Use of alpha 7 nicotinic receptor agonists for the treatment of narcolepsy
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WO2020163405A1 (en) 2019-02-05 2020-08-13 Skyhawk Therapeutics, Inc. Methods and compositions for modulating splicing
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IL225968A0 (en) 2013-06-27
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