PT101308B - Processo para a preparcao de novos n-derivados de (feniletil-beta-ol)-aminas - Google Patents

Processo para a preparcao de novos n-derivados de (feniletil-beta-ol)-aminas Download PDF

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Publication number
PT101308B
PT101308B PT101308A PT10130893A PT101308B PT 101308 B PT101308 B PT 101308B PT 101308 A PT101308 A PT 101308A PT 10130893 A PT10130893 A PT 10130893A PT 101308 B PT101308 B PT 101308B
Authority
PT
Portugal
Prior art keywords
compound
trans
cis
nmr
meoh
Prior art date
Application number
PT101308A
Other languages
English (en)
Portuguese (pt)
Other versions
PT101308A (pt
Inventor
Pierre Braquet
Colette Broquet
Serge Auvin
Original Assignee
Scras
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Scras filed Critical Scras
Publication of PT101308A publication Critical patent/PT101308A/pt
Publication of PT101308B publication Critical patent/PT101308B/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/08—Bronchodilators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/02—Non-specific cardiovascular stimulants, e.g. drugs for syncope, antihypotensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
    • C07D307/04—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C07D307/10—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D307/14—Radicals substituted by nitrogen atoms not forming part of a nitro radical

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Furan Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
PT101308A 1992-07-17 1993-07-15 Processo para a preparcao de novos n-derivados de (feniletil-beta-ol)-aminas PT101308B (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB929215274A GB9215274D0 (en) 1992-07-17 1992-07-17 Derivatives of(phenylethyl-beta-ol)amine

Publications (2)

Publication Number Publication Date
PT101308A PT101308A (pt) 1994-05-31
PT101308B true PT101308B (pt) 1999-10-29

Family

ID=10718914

Family Applications (1)

Application Number Title Priority Date Filing Date
PT101308A PT101308B (pt) 1992-07-17 1993-07-15 Processo para a preparcao de novos n-derivados de (feniletil-beta-ol)-aminas

Country Status (32)

Country Link
US (1) US5447942A (OSRAM)
JP (1) JP3204811B2 (OSRAM)
AT (1) AT403693B (OSRAM)
AU (1) AU672791B2 (OSRAM)
BE (1) BE1006429A3 (OSRAM)
CA (1) CA2100381C (OSRAM)
CH (1) CH687705A5 (OSRAM)
DE (1) DE4323976C2 (OSRAM)
DK (1) DK84793A (OSRAM)
DZ (1) DZ1704A1 (OSRAM)
ES (1) ES2067417B1 (OSRAM)
FI (1) FI933235L (OSRAM)
FR (2) FR2693653B1 (OSRAM)
GB (2) GB9215274D0 (OSRAM)
GR (1) GR1001565B (OSRAM)
HK (1) HK52596A (OSRAM)
HU (1) HUT64757A (OSRAM)
IE (1) IE73266B1 (OSRAM)
IN (1) IN183086B (OSRAM)
LU (1) LU88383A1 (OSRAM)
MA (1) MA22937A1 (OSRAM)
MY (1) MY109395A (OSRAM)
NL (1) NL9301241A (OSRAM)
NO (1) NO302946B1 (OSRAM)
NZ (1) NZ248041A (OSRAM)
OA (1) OA09838A (OSRAM)
PL (1) PL173783B1 (OSRAM)
PT (1) PT101308B (OSRAM)
RU (1) RU2060252C1 (OSRAM)
SE (1) SE503805C2 (OSRAM)
TN (1) TNSN93081A1 (OSRAM)
ZA (1) ZA934667B (OSRAM)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1771435A4 (en) * 2004-06-19 2008-02-13 Human Biomolecular Res Inst MODULATORS OF NEUROTRANSMITTERS OF THE CENTRAL NERVOUS SYSTEM
WO2020148325A1 (en) 2019-01-15 2020-07-23 Phenex-Fxr Gmbh Neutral lxr modulators
GB202304652D0 (en) * 2023-03-29 2023-05-10 Atrogi Ab New compounds and medical uses thereof

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3700692A (en) 1971-06-04 1972-10-24 Colgate Palmolive Co 1-(4{40 -hydroxy-3{40 -(hydroxy methyl)-phenyl)-1-hydroxy-2-aralkylaminoethanes
ZW6584A1 (en) * 1983-04-18 1985-04-17 Glaxo Group Ltd Phenethanolamine derivatives
NZ211822A (en) * 1984-04-17 1988-11-29 Glaxo Group Ltd Phenethanolamine derivatives and pharmaceutical compositions
DE3731198A1 (de) * 1987-02-07 1988-08-18 Bayer Ag 2-aminomethyltetrahydrofurane
US4937268A (en) * 1987-03-12 1990-06-26 Glaxo Group Limited Chemical compounds
GB2230525A (en) * 1989-04-14 1990-10-24 Glaxo Group Ltd 1-(Hydroxyphenyl)-2-aminoethanol derivatives
GB2230775A (en) * 1989-04-24 1990-10-31 Glaxo Group Ltd Phenethanolamine compounds
JPH03133946A (ja) * 1989-10-10 1991-06-07 Glaxo Group Ltd フェンエタノールアミン化合物

Also Published As

Publication number Publication date
FR2693723B1 (fr) 1994-10-28
IN183086B (OSRAM) 1999-09-04
FI933235A0 (fi) 1993-07-16
PT101308A (pt) 1994-05-31
NO932383D0 (no) 1993-06-29
IE930472A1 (en) 1994-01-26
ES2067417A1 (es) 1995-03-16
RU2060252C1 (ru) 1996-05-20
MA22937A1 (fr) 1994-04-01
FI933235A7 (fi) 1994-01-18
GB2268742B (en) 1995-11-08
AU4204293A (en) 1994-01-20
CH687705A5 (fr) 1997-01-31
NL9301241A (nl) 1994-02-16
LU88383A1 (fr) 1994-04-01
IE73266B1 (en) 1997-05-21
DE4323976A1 (de) 1994-01-20
DK84793A (da) 1994-01-18
JP3204811B2 (ja) 2001-09-04
FR2693653B1 (fr) 1994-10-28
FR2693723A1 (fr) 1994-01-21
GB2268742A (en) 1994-01-19
SE9302437L (sv) 1994-01-18
NO302946B1 (no) 1998-05-11
NO932383L (no) 1994-01-18
AT403693B (de) 1998-04-27
GB9314718D0 (en) 1993-08-25
GB9215274D0 (en) 1992-09-02
CA2100381A1 (en) 1994-01-18
NZ248041A (en) 1994-06-27
PL299693A1 (en) 1994-03-21
PL173783B1 (pl) 1998-04-30
HUT64757A (en) 1994-02-28
SE9302437D0 (sv) 1993-07-16
MY109395A (en) 1997-01-31
SE503805C2 (sv) 1996-09-09
GR1001565B (el) 1994-05-31
AU672791B2 (en) 1996-10-17
ZA934667B (en) 1994-01-25
OA09838A (fr) 1994-08-15
DK84793D0 (da) 1993-07-16
FR2693653A1 (fr) 1994-01-21
DZ1704A1 (fr) 2002-02-17
JPH06157492A (ja) 1994-06-03
ES2067417B1 (es) 1995-11-16
DE4323976C2 (de) 2003-05-28
BE1006429A3 (fr) 1994-08-23
CA2100381C (en) 2004-09-21
ATA142793A (de) 1997-09-15
US5447942A (en) 1995-09-05
FI933235L (fi) 1994-01-18
HK52596A (en) 1996-04-03
TNSN93081A1 (fr) 1994-03-17
HU9302057D0 (en) 1993-10-28

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BB1A Laying open of patent application

Effective date: 19931018

FG3A Patent granted, date of granting

Effective date: 19990708

MM4A Annulment/lapse due to non-payment of fees, searched and examined patent

Free format text: LAPSE DUE TO NON-PAYMENT OF FEES

Effective date: 20100108