ES2067417A1 - Procedimiento para preparar nuevos derivados en n de (feniletil-beta-ol)-amina. - Google Patents
Procedimiento para preparar nuevos derivados en n de (feniletil-beta-ol)-amina.Info
- Publication number
- ES2067417A1 ES2067417A1 ES09301603A ES9301603A ES2067417A1 ES 2067417 A1 ES2067417 A1 ES 2067417A1 ES 09301603 A ES09301603 A ES 09301603A ES 9301603 A ES9301603 A ES 9301603A ES 2067417 A1 ES2067417 A1 ES 2067417A1
- Authority
- ES
- Spain
- Prior art keywords
- phenylethyl
- beta
- preparation
- same
- amine
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 150000001412 amines Chemical class 0.000 title 1
- 239000000203 mixture Substances 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/02—Non-specific cardiovascular stimulants, e.g. drugs for syncope, antihypotensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
- C07D307/04—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
- C07D307/10—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D307/14—Radicals substituted by nitrogen atoms not forming part of a nitro radical
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Pulmonology (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Furan Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
PROCEDIMIENTO PARA LA PREPARACION DE NUEVOS DERIVADOS DE N DE (FENILETIL-OL)-AMINA, CONCRETAMENTE DE UN DERIVADO DE N-(TETRAHIDROFURIL DISUSTITUIDO EN 2,4 O 2,5)-ALQUIL -N-(FENILETIL-OL)-AMINA BAJO UNA FORMA RACEMICA O ENANTIOMERA, DE FORMULA GENERAL I FORMULA EN QUE R REPRESENTA DIVERSOS RADICALES Y N ES DE 1 A 10, COMPRENDIENDO DICHO PROCEDIMIENTO UNA CONDENSACION DE UNA BENCILAMINA SUSTITUIDA DE FORMULA GENERAL II FORMULA CON 5-BROMOACETIL-SALICILATO DE METILO III, LUEGO REDUCCION Y, FINALMENTE, UNA DESBENCILACION.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB929215274A GB9215274D0 (en) | 1992-07-17 | 1992-07-17 | Derivatives of(phenylethyl-beta-ol)amine |
Publications (2)
Publication Number | Publication Date |
---|---|
ES2067417A1 true ES2067417A1 (es) | 1995-03-16 |
ES2067417B1 ES2067417B1 (es) | 1995-11-16 |
Family
ID=10718914
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES09301603A Expired - Fee Related ES2067417B1 (es) | 1992-07-17 | 1993-07-16 | Procedimiento para preparar nuevos derivados en n de (feniletil-beta-ol)-amina. |
Country Status (32)
Country | Link |
---|---|
US (1) | US5447942A (es) |
JP (1) | JP3204811B2 (es) |
AT (1) | AT403693B (es) |
AU (1) | AU672791B2 (es) |
BE (1) | BE1006429A3 (es) |
CA (1) | CA2100381C (es) |
CH (1) | CH687705A5 (es) |
DE (1) | DE4323976C2 (es) |
DK (1) | DK84793A (es) |
DZ (1) | DZ1704A1 (es) |
ES (1) | ES2067417B1 (es) |
FI (1) | FI933235A (es) |
FR (2) | FR2693723B1 (es) |
GB (2) | GB9215274D0 (es) |
GR (1) | GR1001565B (es) |
HK (1) | HK52596A (es) |
HU (1) | HUT64757A (es) |
IE (1) | IE73266B1 (es) |
IN (1) | IN183086B (es) |
LU (1) | LU88383A1 (es) |
MA (1) | MA22937A1 (es) |
MY (1) | MY109395A (es) |
NL (1) | NL9301241A (es) |
NO (1) | NO302946B1 (es) |
NZ (1) | NZ248041A (es) |
OA (1) | OA09838A (es) |
PL (1) | PL173783B1 (es) |
PT (1) | PT101308B (es) |
RU (1) | RU2060252C1 (es) |
SE (1) | SE503805C2 (es) |
TN (1) | TNSN93081A1 (es) |
ZA (1) | ZA934667B (es) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP1771435A4 (en) * | 2004-06-19 | 2008-02-13 | Human Biomolecular Res Inst | MODULATORS OF NEUROTRANSMITTERS OF THE CENTRAL NERVOUS SYSTEM |
WO2020148325A1 (en) | 2019-01-15 | 2020-07-23 | Phenex-Fxr Gmbh | Neutral lxr modulators |
Citations (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ES8505641A1 (es) * | 1983-04-18 | 1985-06-01 | Glaxo Group Ltd | Un procedimiento para la preparacion de derivados de fenetanolamina. |
EP0422889A2 (en) * | 1989-10-10 | 1991-04-17 | Glaxo Group Limited | Phenethanolamine compounds |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3700692A (en) | 1971-06-04 | 1972-10-24 | Colgate Palmolive Co | 1-(4{40 -hydroxy-3{40 -(hydroxy methyl)-phenyl)-1-hydroxy-2-aralkylaminoethanes |
GB2159151B (en) * | 1984-04-17 | 1987-10-07 | Glaxo Group Ltd | Phenethanolamine compounds |
DE3731198A1 (de) * | 1987-02-07 | 1988-08-18 | Bayer Ag | 2-aminomethyltetrahydrofurane |
EP0286242A3 (en) * | 1987-03-12 | 1989-08-09 | Glaxo Group Limited | Ethanolamine derivates, processes for their preparation and pharmaceutical compositions containing them |
GB2230525A (en) * | 1989-04-14 | 1990-10-24 | Glaxo Group Ltd | 1-(Hydroxyphenyl)-2-aminoethanol derivatives |
GB2230775A (en) * | 1989-04-24 | 1990-10-31 | Glaxo Group Ltd | Phenethanolamine compounds |
-
1992
- 1992-07-17 GB GB929215274A patent/GB9215274D0/en active Pending
-
1993
- 1993-06-24 IE IE930472A patent/IE73266B1/en not_active IP Right Cessation
- 1993-06-25 GR GR930100276A patent/GR1001565B/el not_active IP Right Cessation
- 1993-06-29 NO NO932383A patent/NO302946B1/no unknown
- 1993-06-29 ZA ZA934667A patent/ZA934667B/xx unknown
- 1993-06-30 IN IN678DE1993 patent/IN183086B/en unknown
- 1993-07-01 NZ NZ248041A patent/NZ248041A/xx unknown
- 1993-07-06 MY MYPI93001317A patent/MY109395A/en unknown
- 1993-07-09 FR FR9308452A patent/FR2693723B1/fr not_active Expired - Fee Related
- 1993-07-09 BE BE9300712A patent/BE1006429A3/fr not_active IP Right Cessation
- 1993-07-09 FR FR9308453A patent/FR2693653B1/fr not_active Expired - Fee Related
- 1993-07-09 CH CH02076/93A patent/CH687705A5/fr not_active IP Right Cessation
- 1993-07-12 DZ DZ930084A patent/DZ1704A1/fr active
- 1993-07-13 CA CA002100381A patent/CA2100381C/en not_active Expired - Fee Related
- 1993-07-13 US US08/091,589 patent/US5447942A/en not_active Expired - Lifetime
- 1993-07-15 PL PL93299693A patent/PL173783B1/pl unknown
- 1993-07-15 PT PT101308A patent/PT101308B/pt not_active IP Right Cessation
- 1993-07-15 GB GB9314718A patent/GB2268742B/en not_active Expired - Fee Related
- 1993-07-15 LU LU88383A patent/LU88383A1/fr unknown
- 1993-07-15 NL NL9301241A patent/NL9301241A/nl not_active Application Discontinuation
- 1993-07-16 MA MA23237A patent/MA22937A1/fr unknown
- 1993-07-16 RU RU9393046412A patent/RU2060252C1/ru active
- 1993-07-16 ES ES09301603A patent/ES2067417B1/es not_active Expired - Fee Related
- 1993-07-16 SE SE9302437A patent/SE503805C2/sv not_active IP Right Cessation
- 1993-07-16 TN TNTNSN93081A patent/TNSN93081A1/fr unknown
- 1993-07-16 DE DE4323976A patent/DE4323976C2/de not_active Expired - Fee Related
- 1993-07-16 AU AU42042/93A patent/AU672791B2/en not_active Ceased
- 1993-07-16 JP JP17693293A patent/JP3204811B2/ja not_active Expired - Fee Related
- 1993-07-16 FI FI933235A patent/FI933235A/fi unknown
- 1993-07-16 DK DK084793A patent/DK84793A/da not_active Application Discontinuation
- 1993-07-16 OA OA60392A patent/OA09838A/fr unknown
- 1993-07-16 HU HU9302057A patent/HUT64757A/hu unknown
- 1993-07-19 AT AT0142793A patent/AT403693B/de not_active IP Right Cessation
-
1996
- 1996-03-28 HK HK52596A patent/HK52596A/xx not_active IP Right Cessation
Patent Citations (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ES8505641A1 (es) * | 1983-04-18 | 1985-06-01 | Glaxo Group Ltd | Un procedimiento para la preparacion de derivados de fenetanolamina. |
EP0422889A2 (en) * | 1989-10-10 | 1991-04-17 | Glaxo Group Limited | Phenethanolamine compounds |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FD2A | Announcement of lapse in spain |
Effective date: 20180806 |