PT1007039E - Novos analogos heterociclicos de compostos de difeniletileno - Google Patents

Novos analogos heterociclicos de compostos de difeniletileno

Info

Publication number
PT1007039E
PT1007039E PT99922836T PT99922836T PT1007039E PT 1007039 E PT1007039 E PT 1007039E PT 99922836 T PT99922836 T PT 99922836T PT 99922836 T PT99922836 T PT 99922836T PT 1007039 E PT1007039 E PT 1007039E
Authority
PT
Portugal
Prior art keywords
compounds
difenylethylene
new heterocyclic
heterocyclic analogs
levels
Prior art date
Application number
PT99922836T
Other languages
English (en)
Inventor
Partha Neogi
Bishwajit Nag
Satyanarayana Medicherla
Debendranath Dey
Original Assignee
Theracos Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US09/074,925 external-priority patent/US6245814B1/en
Application filed by Theracos Inc filed Critical Theracos Inc
Publication of PT1007039E publication Critical patent/PT1007039E/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/34—Oxygen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Diabetes (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Emergency Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Endocrinology (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Photoreceptors In Electrophotography (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
PT99922836T 1998-05-08 1999-05-07 Novos analogos heterociclicos de compostos de difeniletileno PT1007039E (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US09/074,925 US6245814B1 (en) 1998-05-08 1998-05-08 Diphenylethylene compounds
US09/287,237 US6331633B1 (en) 1998-05-08 1999-04-06 Heterocyclic analogs of diphenylethylene compounds

Publications (1)

Publication Number Publication Date
PT1007039E true PT1007039E (pt) 2004-07-30

Family

ID=26756222

Family Applications (1)

Application Number Title Priority Date Filing Date
PT99922836T PT1007039E (pt) 1998-05-08 1999-05-07 Novos analogos heterociclicos de compostos de difeniletileno

Country Status (14)

Country Link
US (1) US6331633B1 (pt)
EP (1) EP1007039B1 (pt)
JP (1) JP4577985B2 (pt)
KR (1) KR100595919B1 (pt)
CN (1) CN1151139C (pt)
AT (1) ATE260906T1 (pt)
AU (1) AU751235C (pt)
CA (1) CA2295599C (pt)
DE (1) DE69915223T2 (pt)
DK (1) DK1007039T3 (pt)
ES (1) ES2216513T3 (pt)
HK (1) HK1028348A1 (pt)
PT (1) PT1007039E (pt)
WO (1) WO1999058127A1 (pt)

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US7521465B2 (en) * 2003-01-17 2009-04-21 Bexel Pharmaceuticals, Inc. Diphenyl ether derivatives
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US8017634B2 (en) 2003-12-29 2011-09-13 President And Fellows Of Harvard College Compositions for treating obesity and insulin resistance disorders
AU2004312072B2 (en) * 2003-12-29 2011-06-23 President And Fellows Of Harvard College Compositions for treating or preventing obesity and insulin resistance disorders
CA2595486A1 (en) * 2005-01-20 2006-07-27 Sirtris Pharmaceuticals, Inc. Use of sirtuin-activating compounds for treating flushing and drug induced weight gain
US20080267888A1 (en) * 2005-05-26 2008-10-30 Pandey Surendrakumar Satyanara Heterocyclic Derivatives
WO2006138418A2 (en) 2005-06-14 2006-12-28 President And Fellows Of Harvard College Improvement of cognitive performance with sirtuin activators
WO2007042878A1 (en) * 2005-10-07 2007-04-19 Orchid Research Laboratories Limited Novel heterocyclic analogs of biphenyl ethers
KR101016875B1 (ko) * 2006-06-23 2011-02-22 현대중공업 주식회사 밀폐형 방청유 도포장치
CN112209896B (zh) * 2019-07-10 2023-05-16 苏州泽璟生物制药股份有限公司 噻唑烷二酮衍生物以及包含其的药物组合物
EP4205740A4 (en) * 2020-08-28 2024-09-04 Celros Biotech THIOHYDANTOIN DERIVATIVES AND THEIR USES

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Also Published As

Publication number Publication date
EP1007039B1 (en) 2004-03-03
CN1273528A (zh) 2000-11-15
DE69915223D1 (de) 2004-04-08
JP4577985B2 (ja) 2010-11-10
HK1028348A1 (en) 2001-02-16
ATE260906T1 (de) 2004-03-15
AU3974199A (en) 1999-11-29
DE69915223T2 (de) 2005-01-27
CA2295599C (en) 2009-01-20
WO1999058127A1 (en) 1999-11-18
EP1007039A1 (en) 2000-06-14
EP1007039A4 (en) 2002-05-22
CN1151139C (zh) 2004-05-26
US6331633B1 (en) 2001-12-18
CA2295599A1 (en) 1999-11-18
ES2216513T3 (es) 2004-10-16
KR20010021615A (ko) 2001-03-15
JP2002514598A (ja) 2002-05-21
AU751235B2 (en) 2002-08-08
AU751235C (en) 2004-06-24
KR100595919B1 (ko) 2006-07-03
DK1007039T3 (da) 2004-07-12

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