PL94120B1 - - Google Patents

Download PDF

Info

Publication number
PL94120B1
PL94120B1 PL1974176207A PL17620774A PL94120B1 PL 94120 B1 PL94120 B1 PL 94120B1 PL 1974176207 A PL1974176207 A PL 1974176207A PL 17620774 A PL17620774 A PL 17620774A PL 94120 B1 PL94120 B1 PL 94120B1
Authority
PL
Poland
Prior art keywords
group
formula
compound
general formula
piperazinyl
Prior art date
Application number
PL1974176207A
Other languages
English (en)
Polish (pl)
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of PL94120B1 publication Critical patent/PL94120B1/pl

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/95Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in positions 2 and 4

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Cephalosporin Compounds (AREA)
PL1974176207A 1973-12-05 1974-12-05 PL94120B1 (forum.php)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/421,992 US3935213A (en) 1973-12-05 1973-12-05 Process for hypotensive 4-amino-2-(piperazin-1-yl) quinazoline derivatives

Publications (1)

Publication Number Publication Date
PL94120B1 true PL94120B1 (forum.php) 1977-07-30

Family

ID=23672938

Family Applications (1)

Application Number Title Priority Date Filing Date
PL1974176207A PL94120B1 (forum.php) 1973-12-05 1974-12-05

Country Status (32)

Country Link
US (1) US3935213A (forum.php)
JP (1) JPS5093987A (forum.php)
AR (1) AR207766A1 (forum.php)
AT (1) AT342598B (forum.php)
BE (1) BE822873A (forum.php)
CA (1) CA1010866A (forum.php)
CH (1) CH587843A5 (forum.php)
CS (1) CS189678B2 (forum.php)
DD (1) DD114950A5 (forum.php)
DE (1) DE2457911A1 (forum.php)
DK (1) DK135376B (forum.php)
EG (1) EG11404A (forum.php)
ES (1) ES432483A1 (forum.php)
FI (1) FI59799B (forum.php)
FR (1) FR2253750B1 (forum.php)
GB (1) GB1464583A (forum.php)
HK (1) HK28379A (forum.php)
IE (1) IE40204B1 (forum.php)
IL (1) IL46102A (forum.php)
IN (1) IN140460B (forum.php)
KE (1) KE2933A (forum.php)
LU (1) LU71427A1 (forum.php)
MY (1) MY7900247A (forum.php)
NL (1) NL7415793A (forum.php)
NO (1) NO141898C (forum.php)
PH (1) PH10594A (forum.php)
PL (1) PL94120B1 (forum.php)
RO (1) RO65957A (forum.php)
SE (1) SE411348B (forum.php)
SU (1) SU563914A3 (forum.php)
YU (1) YU36948B (forum.php)
ZA (1) ZA747593B (forum.php)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4001238A (en) * 1976-02-18 1977-01-04 Bristol-Myers Company 1,3,4-oxadiazole amides
US4060615A (en) * 1976-02-18 1977-11-29 Mead Johnson & Company 2-Piperazinyl-6,7-dimethoxyquinazolines
US4001237A (en) * 1976-02-18 1977-01-04 Bristol-Myers Company Oxazole, isoxazole, thiazole and isothiazole amides
SE435380B (sv) 1976-06-15 1984-09-24 Pfizer Forfarande for framstellning av kinazolinforeningar
US4062844A (en) * 1976-09-20 1977-12-13 Pfizer Inc. Process for preparing hypotensive 2-(4-aroylpiperazin-1-yl)-amino-6,7-dimethoxyquinazolines
FI58124C (fi) * 1976-12-15 1980-12-10 Orion Yhtymae Oy Ny mellanprodukt 3,4-dimetoxi-6-(4-(2-furoyl)-1-piperazinyltiokarbamido)-bensonitril foer framstaellning av 6,7-dimetoxi-4-amino-2-(4-(2-furoyl)-1-piperazinyl)kinazolin med blodtryckssaenkande verkan
FI58125C (fi) * 1976-12-15 1985-01-02 Orion Yhtymae Oy Foerfarande foer framstaellning av 6,7-dimetoxi-4-amino-2-(4-(2-furoyl)-1-piperazinyl)kinazolin med blodtryckssaenkande vekan
US4138561A (en) * 1977-09-30 1979-02-06 Bristol-Myers Company Cyanocarboxamidines and quinazoline process
DK153878C (da) * 1978-05-18 1989-02-06 Pfizer Fremgangsmaade til fremstilling af 2'-methyl-2'-hydroxy-propyl-piperazin-1-carboxylatforbindelser
FI67699C (fi) * 1979-01-31 1985-05-10 Orion Yhtymae Oy Foerfarande foer framstaellning av 6,7-dimetoxi-4-amino-2-(4-(2-furoyl)-1-piperazinyl)kinazolinhydroklorid med blodtryckssaenkande verkan
US4426382A (en) 1980-02-13 1984-01-17 Sankyo Company Limited 4-Amino-6,7-dimethoxy-2-piperazinylquinazoline derivatives, their preparation and use
US4333937A (en) * 1980-04-18 1982-06-08 American Home Products Corp. 2-(Piperazinyl)-4-pyrimioinamines
US4351832A (en) * 1980-04-18 1982-09-28 American Home Products Corporation 2-(Piperazinyl)-4-pyrimidinamines
FI70411C (fi) * 1980-12-29 1986-09-19 Pfizer Foerfarande foer framstaellning av nya antihypertensiva 4-amino-6,7-dimetoxi-2-piperazinokinazolin derivat
FI79107C (fi) * 1984-06-25 1989-11-10 Orion Yhtymae Oy Foerfarande foer framstaellning av stabil -form av prazosinhydroklorid.
CA2077252C (en) * 1992-08-31 2001-04-10 Khashayar Karimian Methods of making ureas and guanidines, and intermediates therefor
WO1996016946A1 (fr) * 1994-11-25 1996-06-06 Nippon Chemiphar Co., Ltd. Derive de quinazoline
US6313294B1 (en) 1998-02-04 2001-11-06 Development Center For Biotechnology Process for preparing amides
US20070086958A1 (en) * 2005-10-14 2007-04-19 Medafor, Incorporated Formation of medically useful gels comprising microporous particles and methods of use
US20070087061A1 (en) * 2005-10-14 2007-04-19 Medafor, Incorporated Method and composition for creating and/or activating a platelet-rich gel by contact with a porous particulate material, for use in wound care, tissue adhesion, or as a matrix for delivery of therapeutic components

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3511836A (en) * 1967-12-13 1970-05-12 Pfizer & Co C 2,4,6,7-tetra substituted quinazolines

Also Published As

Publication number Publication date
EG11404A (en) 1978-03-29
IL46102A0 (en) 1975-02-10
IL46102A (en) 1977-12-30
US3935213A (en) 1976-01-27
LU71427A1 (forum.php) 1975-08-20
AT342598B (de) 1978-04-10
AR207766A1 (es) 1976-10-29
DK135376C (forum.php) 1977-09-26
CA1010866A (en) 1977-05-24
ATA970274A (de) 1977-08-15
IE40204L (en) 1975-06-05
NO141898B (no) 1980-02-18
DK135376B (da) 1977-04-18
SE7413960L (forum.php) 1975-06-06
FR2253750A1 (forum.php) 1975-07-04
YU36948B (en) 1984-08-31
DE2457911A1 (de) 1975-06-12
PH10594A (en) 1977-07-15
SE411348B (sv) 1979-12-17
KE2933A (en) 1979-03-30
BE822873A (fr) 1975-06-03
CH587843A5 (forum.php) 1977-05-13
FI351474A7 (forum.php) 1975-06-06
CS189678B2 (en) 1979-04-30
SU563914A3 (ru) 1977-06-30
GB1464583A (en) 1977-02-16
FR2253750B1 (forum.php) 1977-10-28
ES432483A1 (es) 1976-11-16
FI59799B (fi) 1981-06-30
MY7900247A (en) 1979-12-31
NO744382L (forum.php) 1975-06-30
HK28379A (en) 1979-05-11
IE40204B1 (en) 1979-04-11
IN140460B (forum.php) 1976-11-13
ZA747593B (en) 1975-12-31
AU7553874A (en) 1976-05-20
NL7415793A (nl) 1975-06-09
YU317874A (en) 1982-06-18
NO141898C (no) 1980-06-04
DD114950A5 (forum.php) 1975-09-05
DK629874A (forum.php) 1975-07-21
RO65957A (fr) 1979-07-15
JPS5093987A (forum.php) 1975-07-26

Similar Documents

Publication Publication Date Title
PL94120B1 (forum.php)
DK1797037T3 (en) PROCESS FOR THE PREPARATION OF 4- {4 - [({[4-chloro-3- (trifluoromethyl) phenyl] AMINO} CARBONYL) AMINO] PHENYOXY} N-methylpyridine-2-carboxamide
US4973695A (en) Process for preparing pyridine-2,3-dicarboxylic acid compounds
AU2013293974B2 (en) Method for Producing 4-[5-(Pyridin-4-yl)-1H-1,2,4-Triazol-3-yl]Pyridin-2-Carbonitrile, and Intermediate thereof
AU2002217089B2 (en) Method for producing sulfonamide-substituted imidazotriazinones
CZ20032654A3 (cs) Způsob výroby 4,6-diaminopyrimido(5,4-d)pyrimidinů
Sondhi et al. Synthesis, anti-inflammatory and analgesic activity evaluation of some pyrimidine derivatives
JPH0219829B2 (forum.php)
US4650892A (en) Process for the preparation of herbicidal sulfonamides
CS203172B2 (en) Method of producing 2-/4-furoylpiperazin-1-yl-/4-amino-6,7-dimethoxyquinazoline derivatives
FI66853C (fi) Mellanprodukt foer anvaendning vid framstaellning av hypotensivt 2-(4-(2-furoyl)piperazin-1-yl)-6,7-dimetoxikinazolin
Alagarsamy et al. Synthesis and pharmacological investigation of novel 4‐(4‐Ethyl phenyl)‐1‐substituted‐4H‐[1, 2, 4] triazolo [4, 3‐a]‐quinazolin‐5‐ones as new class of H1‐antihistaminic agents
US4493838A (en) Medicaments containing derivatives of 3-chloro-quinoline
JP3338872B2 (ja) 1,2−ベンゾイソチアゾリノン化合物の製造方法
JPS5982366A (ja) ケト中間体ならびにその用法および製造方法
JP5079809B2 (ja) (3−アルキル−5−ピペリジン−1−イル−3,3a−ジヒドロ−ピラゾロ[1,5−a]ピリミジン−7−イル)−アミノ誘導体および中間体の合成のための方法および合成のための中間体
CA2307080C (en) Process for preparing 8-cyclopentyl-6-ethyl-3-¬substituted|-5,8-dihydro-4h-1,2,3a,7,8-pentaaza-as-indacenes and intermediates useful therein
EP0188225A1 (en) Process for the preparation of herbicidal sulfonamides derived from substituted 2-amino-1,2,4 triazolo (1,5-a) pyrimidines and novel intermediates provided therein
Eldin 2-Amino-1, 1, 3-tricyanopropene in heterocyclic synthesis: novel synthesis of thiopyran pyridinethiones and nicotinonitrile derivatives
CZ111898A3 (cs) Nové deriváty naftylpiperazinu
PL164340B1 (pl) Sposób wytwarzania nowych pochodnych benzotiazyny PL PL
Cowden et al. Pyrimidine N-Oxides. II. The Synthesis of Some Amino-and Imino-pyrimidine N-Oxides and Related Compounds
EP1380585B1 (en) Pyrazolopyridinone as intermediate
Sun et al. A rapid parallel synthesis of 2-dialkylamino-5, 6, 7, 8-tetrahydro-benzothieno [2, 3-d] pyrimidin-4 (3h)-ones
Tarshits et al. Synthesis and transformations of 1, 4-diethynyl-2-nitrobenzene