PL332648A1 - Derivatives of n-(2-benzothiazolyl)-1-piperidinethane mine, their production and application in medical therapy - Google Patents

Derivatives of n-(2-benzothiazolyl)-1-piperidinethane mine, their production and application in medical therapy

Info

Publication number
PL332648A1
PL332648A1 PL97332648A PL33264897A PL332648A1 PL 332648 A1 PL332648 A1 PL 332648A1 PL 97332648 A PL97332648 A PL 97332648A PL 33264897 A PL33264897 A PL 33264897A PL 332648 A1 PL332648 A1 PL 332648A1
Authority
PL
Poland
Prior art keywords
piperidinethane
benzothiazolyl
mine
derivatives
production
Prior art date
Application number
PL97332648A
Other languages
English (en)
Inventor
Gihad Dargazanli
Pascal George
Patrick Lardenois
Jonathan Frost
Johannes Schoemaker
Maria-Carmen Renones
Pascale Magat
Original Assignee
Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthelabo filed Critical Synthelabo
Publication of PL332648A1 publication Critical patent/PL332648A1/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
PL97332648A 1996-10-01 1997-09-26 Derivatives of n-(2-benzothiazolyl)-1-piperidinethane mine, their production and application in medical therapy PL332648A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9611925A FR2753970B1 (fr) 1996-10-01 1996-10-01 Derives de n-(benzothiazol-2-yl) piperidine-1-ethanamine, leur preparation et leur application en therapeutique
PCT/FR1997/001692 WO1998014444A1 (fr) 1996-10-01 1997-09-26 Derives de n-(benzothiazol-2-yl)piperidine-1-ethanamine, leur preparation et leur application en therapeutique

Publications (1)

Publication Number Publication Date
PL332648A1 true PL332648A1 (en) 1999-09-27

Family

ID=9496217

Family Applications (1)

Application Number Title Priority Date Filing Date
PL97332648A PL332648A1 (en) 1996-10-01 1997-09-26 Derivatives of n-(2-benzothiazolyl)-1-piperidinethane mine, their production and application in medical therapy

Country Status (23)

Country Link
EP (1) EP0929550A1 (no)
JP (1) JP2001501217A (no)
KR (1) KR20000048767A (no)
CN (1) CN1230959A (no)
AR (1) AR009105A1 (no)
AU (1) AU722147B2 (no)
BG (1) BG103271A (no)
BR (1) BR9711842A (no)
CA (1) CA2266510A1 (no)
CO (1) CO4650030A1 (no)
CZ (1) CZ112699A3 (no)
EE (1) EE9900135A (no)
FR (1) FR2753970B1 (no)
HU (1) HUP9904091A3 (no)
IL (1) IL128902A (no)
NO (1) NO991581L (no)
NZ (1) NZ334553A (no)
PL (1) PL332648A1 (no)
SK (1) SK42299A3 (no)
TR (1) TR199900634T2 (no)
TW (1) TW438800B (no)
WO (1) WO1998014444A1 (no)
ZA (1) ZA978772B (no)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9725541D0 (en) * 1997-12-02 1998-02-04 Pharmacia & Upjohn Spa Amino-benzothiazole derivatives
US6107313A (en) * 1998-10-02 2000-08-22 Combichem, Inc. Dopamine receptor antagonists
CZ2003182A3 (cs) 2000-06-21 2003-06-18 F. Hoffmann-La Roche Ag Deriváty benzothiazolu
US7087761B2 (en) 2003-01-07 2006-08-08 Hoffmann-La Roche Inc. Cyclization process for substituted benzothiazole derivatives
WO2005040129A2 (en) * 2003-10-24 2005-05-06 F. Hoffmann-La Roche Ag Ccr3 receptor antagonists
JP4668265B2 (ja) 2004-05-24 2011-04-13 エフ.ホフマン−ラ ロシュ アーゲー 4−ヒドロキシ−4−メチル−ピペリジン−1−カルボン酸(4−メトキシ−7−モルホリン−4−イル−ベンゾチアゾール−2−イル)−アミド
WO2006048172A1 (en) 2004-11-05 2006-05-11 F. Hoffmann-La Roche Ag Process for preparation of isonicotinic acid derivatives
KR100973609B1 (ko) 2005-03-23 2010-08-03 에프. 호프만-라 로슈 아게 mGluR2 길항제로서 아세틸렌일-피라졸로-피리미딘유도체
DE602006013493D1 (de) 2005-09-27 2010-05-20 Hoffmann La Roche Oxadiazolylpyrazolopyrimidine als mglur2-antagonisten

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1260474A (en) * 1984-12-03 1989-09-26 Raymond A. Stokbroekx Benzoxazol- and benzothiazolamine derivatives
KR930005004B1 (ko) * 1985-04-15 1993-06-11 쟈안센 파아마슈우티카 엔. 부이. 치환된 n-[(4-피페리디닐)알킬]이환 축합 옥사졸아민 및 티아졸아민의 제조방법

Also Published As

Publication number Publication date
BR9711842A (pt) 1999-08-24
BG103271A (en) 2000-05-31
KR20000048767A (ko) 2000-07-25
CA2266510A1 (en) 1998-04-09
CN1230959A (zh) 1999-10-06
FR2753970A1 (fr) 1998-04-03
JP2001501217A (ja) 2001-01-30
CO4650030A1 (es) 1998-09-03
IL128902A0 (en) 2000-02-17
SK42299A3 (en) 1999-12-10
AU4463897A (en) 1998-04-24
HUP9904091A2 (hu) 2000-05-28
NO991581L (no) 1999-06-01
AU722147B2 (en) 2000-07-20
HUP9904091A3 (en) 2000-07-28
FR2753970B1 (fr) 1998-10-30
ZA978772B (en) 1998-03-27
EP0929550A1 (fr) 1999-07-21
IL128902A (en) 2001-07-24
NO991581D0 (no) 1999-03-30
WO1998014444A1 (fr) 1998-04-09
CZ112699A3 (cs) 1999-06-16
AR009105A1 (es) 2000-03-08
TR199900634T2 (xx) 1999-06-21
TW438800B (en) 2001-06-07
NZ334553A (en) 2000-11-24
EE9900135A (et) 1999-12-15

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