PL3068786T3 - Związki pirazolopirymidynowe - Google Patents

Związki pirazolopirymidynowe

Info

Publication number
PL3068786T3
PL3068786T3 PL14861448T PL14861448T PL3068786T3 PL 3068786 T3 PL3068786 T3 PL 3068786T3 PL 14861448 T PL14861448 T PL 14861448T PL 14861448 T PL14861448 T PL 14861448T PL 3068786 T3 PL3068786 T3 PL 3068786T3
Authority
PL
Poland
Prior art keywords
pyrazolopyrimidine compounds
pyrazolopyrimidine
compounds
Prior art date
Application number
PL14861448T
Other languages
English (en)
Inventor
Radoslaw Laufer
Grace Ng
Sze-Wan Li
Heinz W. Pauls
Yong Liu
Narendra Kumar B. Patel
Original Assignee
University Health Network
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by University Health Network filed Critical University Health Network
Publication of PL3068786T3 publication Critical patent/PL3068786T3/pl

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D519/00Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
PL14861448T 2012-11-16 2014-11-14 Związki pirazolopirymidynowe PL3068786T3 (pl)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201261727581P 2012-11-16 2012-11-16
US201361808152P 2013-04-03 2013-04-03
PCT/CA2013/000957 WO2014075168A1 (en) 2012-11-16 2013-11-15 Pyrazolopyrimidine compounds
EP14861448.0A EP3068786B1 (en) 2012-11-16 2014-11-14 Pyrazolopyrimidine compounds
PCT/CA2014/051091 WO2015070349A1 (en) 2012-11-16 2014-11-14 Pyrazolopyrimidine compounds

Publications (1)

Publication Number Publication Date
PL3068786T3 true PL3068786T3 (pl) 2018-10-31

Family

ID=50730425

Family Applications (1)

Application Number Title Priority Date Filing Date
PL14861448T PL3068786T3 (pl) 2012-11-16 2014-11-14 Związki pirazolopirymidynowe

Country Status (24)

Country Link
US (9) US9573954B2 (pl)
EP (2) EP2920181B1 (pl)
JP (1) JP6377068B2 (pl)
CN (1) CN105793261B (pl)
AU (1) AU2013344716B2 (pl)
BR (1) BR112016010080B1 (pl)
CA (1) CA2889919C (pl)
CY (1) CY1120480T1 (pl)
DK (1) DK3068786T3 (pl)
ES (1) ES2686097T3 (pl)
HR (1) HRP20181041T1 (pl)
HU (1) HUE039351T2 (pl)
IL (1) IL245187B (pl)
LT (1) LT3068786T (pl)
ME (1) ME03093B (pl)
MX (1) MX373713B (pl)
NZ (1) NZ707432A (pl)
PL (1) PL3068786T3 (pl)
PT (1) PT3068786T (pl)
RS (1) RS57481B1 (pl)
SG (1) SG11201603102TA (pl)
SI (1) SI3068786T1 (pl)
TW (1) TWI679201B (pl)
WO (2) WO2014075168A1 (pl)

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AU2019273871A1 (en) * 2018-05-23 2020-12-10 University Health Network Methods of treating cancers characterized by a high expression level of spindle and kinetochore associated complex subunit 3 (SKA3) gene
IL282254B2 (en) 2018-10-30 2025-08-01 Kronos Bio Inc Compounds, compositions, and methods for modulating cdk9 activity
CN111377925B (zh) * 2018-12-28 2024-03-12 四川科伦博泰生物医药股份有限公司 嘌呤类衍生物、其制备方法及其在医药上的应用
CN112142744A (zh) * 2019-06-28 2020-12-29 上海瑛派药业有限公司 取代的稠合杂芳双环化合物作为激酶抑制剂及其应用
TW202146416A (zh) * 2019-12-11 2021-12-16 德商拜耳廠股份有限公司 吡唑并三𠯤
CN113773324B (zh) * 2021-09-07 2022-07-26 武汉九州钰民医药科技有限公司 抗肿瘤药cfi-402257的合成制备工艺
CN116396298A (zh) * 2023-06-06 2023-07-07 四川维亚本苑生物科技有限公司 CDK Ligand-1的中间体XII及CDK Ligand-1的制备方法

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Also Published As

Publication number Publication date
TWI679201B (zh) 2019-12-11
US20170217966A1 (en) 2017-08-03
PT3068786T (pt) 2018-07-26
RS57481B1 (sr) 2018-10-31
SI3068786T1 (sl) 2018-09-28
AU2013344716A1 (en) 2015-05-14
US20210009595A1 (en) 2021-01-14
US9573954B2 (en) 2017-02-21
CY1120480T1 (el) 2019-07-10
SG11201603102TA (en) 2016-05-30
CN105793261B (zh) 2018-11-30
TW201605860A (zh) 2016-02-16
US10106545B2 (en) 2018-10-23
EP2920181B1 (en) 2019-01-09
HRP20181041T1 (hr) 2018-09-21
US9657025B2 (en) 2017-05-23
US20150299203A1 (en) 2015-10-22
BR112016010080A8 (pt) 2020-04-14
JP2015537008A (ja) 2015-12-24
ME03093B (me) 2019-01-20
BR112016010080B1 (pt) 2020-12-29
IL245187A0 (en) 2016-06-30
US10570143B2 (en) 2020-02-25
US10167289B2 (en) 2019-01-01
US20160137651A1 (en) 2016-05-19
EP3068786A4 (en) 2017-04-12
MX373713B (es) 2020-05-08
HUE039351T2 (hu) 2018-12-28
CN105793261A (zh) 2016-07-20
US20240287077A1 (en) 2024-08-29
IL245187B (en) 2019-12-31
WO2014075168A1 (en) 2014-05-22
EP3068786B1 (en) 2018-06-06
US20170320881A1 (en) 2017-11-09
NZ707432A (en) 2020-01-31
CA2889919A1 (en) 2014-05-22
WO2015070349A1 (en) 2015-05-21
ES2686097T3 (es) 2018-10-16
AU2013344716B2 (en) 2018-03-01
EP2920181A1 (en) 2015-09-23
EP2920181A4 (en) 2016-07-27
US20190322669A1 (en) 2019-10-24
EP3068786A1 (en) 2016-09-21
DK3068786T3 (en) 2018-07-16
MX2016006336A (es) 2016-09-06
JP6377068B2 (ja) 2018-08-22
US20190040074A1 (en) 2019-02-07
US20220204511A1 (en) 2022-06-30
LT3068786T (lt) 2018-08-27
CA2889919C (en) 2021-08-17

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