PL3061821T3 - Kompozycje do leczenia zaburzeń łagodzonych przez aktywację receptora muskarynowego - Google Patents
Kompozycje do leczenia zaburzeń łagodzonych przez aktywację receptora muskarynowegoInfo
- Publication number
- PL3061821T3 PL3061821T3 PL16151747T PL16151747T PL3061821T3 PL 3061821 T3 PL3061821 T3 PL 3061821T3 PL 16151747 T PL16151747 T PL 16151747T PL 16151747 T PL16151747 T PL 16151747T PL 3061821 T3 PL3061821 T3 PL 3061821T3
- Authority
- PL
- Poland
- Prior art keywords
- compositions
- treatment
- receptor activation
- muscarinic receptor
- disorders ameliorated
- Prior art date
Links
Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/46—8-Azabicyclo [3.2.1] octane; Derivatives thereof, e.g. atropine, cocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
- A61K31/138—Aryloxyalkylamines, e.g. propranolol, tamoxifen, phenoxybenzamine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
- A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
- A61K31/22—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin
- A61K31/222—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin with compounds having aromatic groups, e.g. dipivefrine, ibopamine
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/4025—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil not condensed and containing further heterocyclic rings, e.g. cromakalim
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4178—1,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/438—The ring being spiro-condensed with carbocyclic or heterocyclic ring systems
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
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- A—HUMAN NECESSITIES
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/472—Non-condensed isoquinolines, e.g. papaverine
- A61K31/4725—Non-condensed isoquinolines, e.g. papaverine containing further heterocyclic rings
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- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
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- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/26—Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
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- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
- A61K47/38—Cellulose; Derivatives thereof
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- A61K9/4816—Wall or shell material
- A61K9/4825—Proteins, e.g. gelatin
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- A61K9/4891—Coated capsules; Multilayered drug free capsule shells
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- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
Applications Claiming Priority (5)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US21385309P | 2009-07-22 | 2009-07-22 | |
US28265810P | 2010-03-15 | 2010-03-15 | |
PCT/US2010/002044 WO2011011060A1 (en) | 2009-07-22 | 2010-07-21 | Methods and compositions for treatment of disorders ameliorated by muscarinic receptor activation |
EP16151747.9A EP3061821B1 (en) | 2009-07-22 | 2010-07-21 | Compositions for treatment of disorders ameliorated by muscarinic receptor activation |
EP10802549.5A EP2456868A4 (en) | 2009-07-22 | 2010-07-21 | METHOD AND COMPOSITIONS FOR TREATING SUFFERING OF SUFFERING THROUGH MUSCARIN RECEPTOR ACTIVATION |
Publications (1)
Publication Number | Publication Date |
---|---|
PL3061821T3 true PL3061821T3 (pl) | 2020-01-31 |
Family
ID=43497520
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PL16151747T PL3061821T3 (pl) | 2009-07-22 | 2010-07-21 | Kompozycje do leczenia zaburzeń łagodzonych przez aktywację receptora muskarynowego |
Country Status (10)
Country | Link |
---|---|
US (9) | US20110020423A1 (pl) |
EP (3) | EP2456868A4 (pl) |
JP (6) | JP2012533621A (pl) |
CA (1) | CA2804215C (pl) |
DK (1) | DK3061821T3 (pl) |
ES (1) | ES2742728T3 (pl) |
HU (1) | HUE044653T2 (pl) |
PL (1) | PL3061821T3 (pl) |
PT (1) | PT3061821T (pl) |
WO (1) | WO2011011060A1 (pl) |
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CA2804215C (en) | 2019-10-01 |
JP2012533621A (ja) | 2012-12-27 |
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WO2011011060A1 (en) | 2011-01-27 |
JP2018002738A (ja) | 2018-01-11 |
EP3061821B1 (en) | 2019-07-10 |
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JP2015083612A (ja) | 2015-04-30 |
US20140099356A1 (en) | 2014-04-10 |
US10369144B2 (en) | 2019-08-06 |
DK3061821T3 (da) | 2019-08-26 |
JP2020023494A (ja) | 2020-02-13 |
US20110020423A1 (en) | 2011-01-27 |
US20190307739A1 (en) | 2019-10-10 |
JP7136545B2 (ja) | 2022-09-13 |
EP2456868A4 (en) | 2013-11-06 |
JP2022168136A (ja) | 2022-11-04 |
HUE044653T2 (hu) | 2019-11-28 |
EP3646870A1 (en) | 2020-05-06 |
ES2742728T3 (es) | 2020-02-17 |
PT3061821T (pt) | 2019-09-05 |
JP2016164201A (ja) | 2016-09-08 |
US10369143B2 (en) | 2019-08-06 |
US10238643B2 (en) | 2019-03-26 |
US20190192500A1 (en) | 2019-06-27 |
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