PL3061821T3 - Kompozycje do leczenia zaburzeń łagodzonych przez aktywację receptora muskarynowego - Google Patents

Kompozycje do leczenia zaburzeń łagodzonych przez aktywację receptora muskarynowego

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Publication number
PL3061821T3
PL3061821T3 PL16151747T PL16151747T PL3061821T3 PL 3061821 T3 PL3061821 T3 PL 3061821T3 PL 16151747 T PL16151747 T PL 16151747T PL 16151747 T PL16151747 T PL 16151747T PL 3061821 T3 PL3061821 T3 PL 3061821T3
Authority
PL
Poland
Prior art keywords
compositions
treatment
receptor activation
muscarinic receptor
disorders ameliorated
Prior art date
Application number
PL16151747T
Other languages
English (en)
Inventor
Eric Elenko
Andrew C. Miller
Phillip E. MURRAY III
Original Assignee
PureTech Health LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by PureTech Health LLC filed Critical PureTech Health LLC
Publication of PL3061821T3 publication Critical patent/PL3061821T3/pl

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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/468-Azabicyclo [3.2.1] octane; Derivatives thereof, e.g. atropine, cocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/138Aryloxyalkylamines, e.g. propranolol, tamoxifen, phenoxybenzamine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/21Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A61K31/22Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin
    • A61K31/222Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin with compounds having aromatic groups, e.g. dipivefrine, ibopamine
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    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/4025Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil not condensed and containing further heterocyclic rings, e.g. cromakalim
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    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
    • A61K31/41781,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
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    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
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    • A61K31/47Quinolines; Isoquinolines
    • A61K31/472Non-condensed isoquinolines, e.g. papaverine
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    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/26Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
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    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • A61K47/38Cellulose; Derivatives thereof
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    • A61K9/4891Coated capsules; Multilayered drug free capsule shells
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PL16151747T 2009-07-22 2010-07-21 Kompozycje do leczenia zaburzeń łagodzonych przez aktywację receptora muskarynowego PL3061821T3 (pl)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US21385309P 2009-07-22 2009-07-22
US28265810P 2010-03-15 2010-03-15
PCT/US2010/002044 WO2011011060A1 (en) 2009-07-22 2010-07-21 Methods and compositions for treatment of disorders ameliorated by muscarinic receptor activation
EP16151747.9A EP3061821B1 (en) 2009-07-22 2010-07-21 Compositions for treatment of disorders ameliorated by muscarinic receptor activation
EP10802549.5A EP2456868A4 (en) 2009-07-22 2010-07-21 METHOD AND COMPOSITIONS FOR TREATING SUFFERING OF SUFFERING THROUGH MUSCARIN RECEPTOR ACTIVATION

Publications (1)

Publication Number Publication Date
PL3061821T3 true PL3061821T3 (pl) 2020-01-31

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PL16151747T PL3061821T3 (pl) 2009-07-22 2010-07-21 Kompozycje do leczenia zaburzeń łagodzonych przez aktywację receptora muskarynowego

Country Status (10)

Country Link
US (9) US20110020423A1 (pl)
EP (3) EP2456868A4 (pl)
JP (6) JP2012533621A (pl)
CA (1) CA2804215C (pl)
DK (1) DK3061821T3 (pl)
ES (1) ES2742728T3 (pl)
HU (1) HUE044653T2 (pl)
PL (1) PL3061821T3 (pl)
PT (1) PT3061821T (pl)
WO (1) WO2011011060A1 (pl)

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